Authors:
van Muijlwijk-Koezen, JE
Timmerman, H
van der Sluis, RP
van de Stolpe, AC
Menge, WMPB
Beukers, MW
van der Graaf, PH
de Groote, M
IJzerman, AP
Citation: Je. Van Muijlwijk-koezen et al., Synthesis and use of FSCPX, an irreversible adenosine A(1) antagonist, as a 'receptor knock-down' tool, BIOORG MED, 11(6), 2001, pp. 815-818
Authors:
Gao, ZG
Van Muijlwijk-Koezen, JE
Chen, AS
Muller, CE
IJzerman, AP
Jacobson, KA
Citation: Zg. Gao et al., Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives, MOLEC PHARM, 60(5), 2001, pp. 1057-1063
Authors:
van Tilburg, EW
van der Klein, PAM
von Frijtag, J
Kunzel, D
de Groote, M
Stannek, C
Lorenzen, A
IJzerman, AP
Citation: Ew. Van Tilburg et al., 5 '-O-alkyl ethers of N,2-substituted adenosine derivatives: Partial agonists for the adenosine A(1) and A(3) receptors, J MED CHEM, 44(18), 2001, pp. 2966-2975
Authors:
Kourounakis, A
Visser, C
de Groote, M
IJzerman, AP
Citation: A. Kourounakis et al., Differential effects of the allosteric enhancer (2-amino-4,5-dimethyl-trienyl)[3-(trifluoromethyl) phenyl]methanone (PD81,723) on agonist and antagonist binding and function at the human wild-type and a mutant (T277A) adenosine A(1) receptor, BIOCH PHARM, 61(2), 2001, pp. 137-144
Authors:
Wanner, MJ
Kunzel, JKVD
IJzerman, AP
Koomen, GJ
Citation: Mj. Wanner et al., 2-nitro analogues of adenosine and 1-deazaadenosine: Synthesis and bindingstudies at the adenosine A(1), A(2A) and A(3) receptor subtypes, BIOORG MED, 10(18), 2000, pp. 2141-2144
Authors:
Kourounakis, AP
Visser, C
de Groote, M
IJzerman, AP
Citation: Ap. Kourounakis et al., Allosteric modulation of the rat adenosine A(1) receptor: Differential effects on agonist and antagonist binding, DRUG DEV R, 51(4), 2000, pp. 207-215
Citation: K. Ingkaninan et al., Luteolin, a compound with adenosine A(1) receptor-binding activity, and chromone and dihydronaphthalenone constituents from Senna siamea, J NAT PROD, 63(3), 2000, pp. 315-317
Authors:
van Muijlwijk-Koezen, JE
Timmerman, H
van der Goot, H
Menge, WMPB
Kunzel, JFV
de Groote, M
IJzerman, AP
Citation: Je. Van Muijlwijk-koezen et al., Isoquinoline and quinazoline urea analogues as antagonists for the human adenosine A(3) receptor, J MED CHEM, 43(11), 2000, pp. 2227-2238
Authors:
Gao, ZG
Jiang, QL
Jacobson, KA
IJzerman, AP
Citation: Zg. Gao et al., Site-directed mutagenesis studies of human A(2A) adenosine receptors - Involvement of Glu(13) and His(278) in ligand binding and sodium modulation, BIOCH PHARM, 60(5), 2000, pp. 661-668
Citation: Zg. Gao et Ap. Ijzerman, Allosteric modulation of A(2A) adenosine receptors by amiloride analogues and sodium ions, BIOCH PHARM, 60(5), 2000, pp. 669-676
Authors:
Dalpiaz, A
Scatturin, A
Pavan, B
Varani, K
IJzerman, AP
Borea, PA
Citation: A. Dalpiaz et al., Thermodynamic in vitro studies as a method to investigate the pharmacodynamic behavior of adenosine A(1) receptor ligands, PHARM RES, 16(7), 1999, pp. 1054-1058
Authors:
van Tilburg, EW
Kunzel, JVD
de Groote, M
Vollinga, RC
Lorenzen, A
IJzerman, AP
Citation: Ew. Van Tilburg et al., N-6,5 '-disubstituted adenosine derivatives as partial agonists for the human adenosine A(3) receptor, J MED CHEM, 42(8), 1999, pp. 1393-1400
Authors:
van der Klein, PAM
Kourounakis, AP
IJzerman, AP
Citation: Pam. Van Der Klein et al., Allosteric modulation of the adenosine A(1) receptor. Synthesis and biological evaluation of novel 2-amino-3-benzoylthiophenes as allosteric enhancers of agonist binding, J MED CHEM, 42(18), 1999, pp. 3629-3635
Citation: Sa. Rivkees et al., Identification of the adenine binding site of the human A(1) adenosine receptor, J BIOL CHEM, 274(6), 1999, pp. 3617-3621