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Results: 1-19 |
Results: 19
SYNTHESIS OF 9-BETA-METHYL-2-ALKYL-7-OXO-5-ARYLMORPHANS
Authors: THOMAS JB ZHENG XL BRIEADDY LE BURGESS JP MASCARELLA SW FIX SE CANTRELL BE ZIMMERMAN DM CARROLL FI
Citation: Jb. Thomas et al., SYNTHESIS OF 9-BETA-METHYL-2-ALKYL-7-OXO-5-ARYLMORPHANS, Tetrahedron letters, 39(39), 1998, pp. 7001-7004
N-SUBSTITUTED 9-BETA-METHYL-5-(3-HYDROXYPHENYL)MORPHANS ARE OPIOID RECEPTOR PURE ANTAGONISTS
Authors: THOMAS JB ZHENG XL MASCARELLA SW ROTHMAN RB DERSCH CM PARTILLA JS FLIPPENANDERSON JL GEORGE CF CANTRELL BE ZIMMERMAN DM CARROLL FI
Citation: Jb. Thomas et al., N-SUBSTITUTED 9-BETA-METHYL-5-(3-HYDROXYPHENYL)MORPHANS ARE OPIOID RECEPTOR PURE ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4143-4149
INVESTIGATION OF THE N-SUBSTITUENT CONFORMATION GOVERNING POTENCY ANDMU-RECEPTOR SUBTYPE-SELECTIVITY IN (-(3R,4R)-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE OPIOID ANTAGONISTS())
Authors: THOMAS JB MASCARELLA SW ROTHMAN RB PARTILLA JS XU H MCCULLOUGH KB DERSCH CN CANTRELL BE ZIMMERMAN DM CARROLL FI
Citation: Jb. Thomas et al., INVESTIGATION OF THE N-SUBSTITUENT CONFORMATION GOVERNING POTENCY ANDMU-RECEPTOR SUBTYPE-SELECTIVITY IN (-(3R,4R)-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE OPIOID ANTAGONISTS()), Journal of medicinal chemistry, 41(11), 1998, pp. 1980-1990
SYNTHESIS AND TRANSPORTER BINDING-PROPERTIES OF 2,3-DIPHENYLTROPANE STEREOISOMERS - COMPARISON TO 3-BETA-PHENYLTROPANE-2-BETA-CARBOXYLIC ACID-ESTERS
Authors: CHANG AC BURGESS JP MASCARELLA SW ABRAHAM P KUHAR MJ CARROLL FI
Citation: Ac. Chang et al., SYNTHESIS AND TRANSPORTER BINDING-PROPERTIES OF 2,3-DIPHENYLTROPANE STEREOISOMERS - COMPARISON TO 3-BETA-PHENYLTROPANE-2-BETA-CARBOXYLIC ACID-ESTERS, Journal of medicinal chemistry, 40(8), 1997, pp. 1247-1251
STRUCTURE-ACTIVITY ANALYSIS OF ANANDAMIDE ANALOGS - RELATIONSHIP TO ACANNABINOID PHARMACOPHORE
Authors: THOMAS BF ADAMS IB MASCARELLA SW MARTIN BR RAZDAN RK
Citation: Bf. Thomas et al., STRUCTURE-ACTIVITY ANALYSIS OF ANANDAMIDE ANALOGS - RELATIONSHIP TO ACANNABINOID PHARMACOPHORE, Journal of medicinal chemistry, 39(2), 1996, pp. 471-479
SYNTHESIS, LIGAND-BINDING, AND QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP STUDY OF 3-BETA-(4-SUBSTITUTED PHENYL)-2-BETA-HETEROCYCLIC TROPANES - EVIDENCE FOR AN ELECTROSTATIC INTERACTION AT THE 2-BETA-POSITION
Authors: KOTIAN P MASCARELLA SW ABRAHAM P LEWIN AH BOJA JW KUHAR MJ CARROLL FI
Citation: P. Kotian et al., SYNTHESIS, LIGAND-BINDING, AND QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP STUDY OF 3-BETA-(4-SUBSTITUTED PHENYL)-2-BETA-HETEROCYCLIC TROPANES - EVIDENCE FOR AN ELECTROSTATIC INTERACTION AT THE 2-BETA-POSITION, Journal of medicinal chemistry, 39(14), 1996, pp. 2753-2763
EFFECTS OF SPHINGOSINE STEREOISOMERS ON P-GLYCOPROTEIN PHOSPHORYLATION AND VINBLASTINE ACCUMULATION IN MULTIDRUG-RESISTANT MCF-7 CELLS
Authors: SACHS CW BALLAS LM MASCARELLA SW SAFA AR LEWIN AH LOOMIS C CARROLL FI BELL RM FINE RL
Citation: Cw. Sachs et al., EFFECTS OF SPHINGOSINE STEREOISOMERS ON P-GLYCOPROTEIN PHOSPHORYLATION AND VINBLASTINE ACCUMULATION IN MULTIDRUG-RESISTANT MCF-7 CELLS, Biochemical pharmacology, 52(4), 1996, pp. 603-612
(-CIS-N-(PARA, META, AND ORTHO SUBSTITUTED BENZYL)-N-NORMETAZOCINES SYNTHESIS AND BINDING-AFFINITY AT THE [H-3] (+)-PENTAZOCINE-LABELED (SIGMA-1)-SITE AND QUANTITATIVE STRUCTURE-AFFINITY RELATIONSHIP STUDIES())
Authors: MASCARELLA SW BAI X WILLIAMS W SINE B BOWEN WD CARROLL FI
Citation: Sw. Mascarella et al., (-CIS-N-(PARA, META, AND ORTHO SUBSTITUTED BENZYL)-N-NORMETAZOCINES SYNTHESIS AND BINDING-AFFINITY AT THE [H-3] (+)-PENTAZOCINE-LABELED (SIGMA-1)-SITE AND QUANTITATIVE STRUCTURE-AFFINITY RELATIONSHIP STUDIES()), Journal of medicinal chemistry, 38(3), 1995, pp. 565-569
SYNTHESIS AND LIGAND-BINDING STUDY OF 3-BETA-(4'-SUBSTITUTED PHENYL)-2-BETA-(HETEROCYCLIC)TROPANES
Authors: KOTIAN P ABRAHAM P LEWIN AH MASCARELLA SW BOJA JW KUHAR MJ CARROLL FI
Citation: P. Kotian et al., SYNTHESIS AND LIGAND-BINDING STUDY OF 3-BETA-(4'-SUBSTITUTED PHENYL)-2-BETA-(HETEROCYCLIC)TROPANES, Journal of medicinal chemistry, 38(18), 1995, pp. 3451-3453
SYNTHESIS AND SIGMA-BINDING-PROPERTIES OF 2'-SUBSTITUTED 5,9-ALPHA-DIMETHYL-6,7-BENZOMORPHANS
Authors: DANSODANQUAH R BAI X ZHANG X MASCARELLA SW WILLIAMS W SINE B BOWEN WD CARROLL FI
Citation: R. Dansodanquah et al., SYNTHESIS AND SIGMA-BINDING-PROPERTIES OF 2'-SUBSTITUTED 5,9-ALPHA-DIMETHYL-6,7-BENZOMORPHANS, Journal of medicinal chemistry, 38(15), 1995, pp. 2978-2985
SYNTHESIS AND SIGMA-BINDING PROPERTIES OF 1'-HALO-N-NORMETAZOCINE AND3'-HALO-N-NORMETAZOCINE AND 1',3'-DIHALO-N-NORMETAZOCINE ANALOGS
Authors: DANSODANQUAH R BAI X ZHANG X MASCARELLA SW WILLIAMS W SINE B BOWEN WD CARROLL FI
Citation: R. Dansodanquah et al., SYNTHESIS AND SIGMA-BINDING PROPERTIES OF 1'-HALO-N-NORMETAZOCINE AND3'-HALO-N-NORMETAZOCINE AND 1',3'-DIHALO-N-NORMETAZOCINE ANALOGS, Journal of medicinal chemistry, 38(15), 1995, pp. 2986-2989
STIMULATION OF RAT STRIATAL TYROSINE-HYDROXYLASE ACTIVITY FOLLOWING INTRANIGRAL ADMINISTRATION OF SIGMA-RECEPTOR LIGANDS
Authors: WEISER SD PATRICK SL MASCARELLA SW DOWNINGPARK J BAI X CARROLL FI WALKER JM PATRICK RL
Citation: Sd. Weiser et al., STIMULATION OF RAT STRIATAL TYROSINE-HYDROXYLASE ACTIVITY FOLLOWING INTRANIGRAL ADMINISTRATION OF SIGMA-RECEPTOR LIGANDS, European journal of pharmacology, 275(1), 1995, pp. 1-7
RTI-4793-14, A NEW LIGAND WITH HIGH-AFFINITY AND SELECTIVITY FOR THE (-MK801-INSENSITIVE [H-3] 1-[1-(2-THIENYL)CYCLOHEXYL]PIPERIDINE BINDING-SITE (PCP SITE-2) OF GUINEA-PIG BRAIN())
Authors: GOODMAN CB THOMAS DN PERT A EMILIEN B CADET JL CARROLL FI BLOUGH BE MASCARELLA SW ROGAWSKI MA SUBRAMANIAM S ROTHMAN RB
Citation: Cb. Goodman et al., RTI-4793-14, A NEW LIGAND WITH HIGH-AFFINITY AND SELECTIVITY FOR THE (-MK801-INSENSITIVE [H-3] 1-[1-(2-THIENYL)CYCLOHEXYL]PIPERIDINE BINDING-SITE (PCP SITE-2) OF GUINEA-PIG BRAIN()), Synapse, 16(1), 1994, pp. 59-65
A NOVEL STEREOSELECTIVE AND ENANTIOSELECTIVE SYNTHESIS OF TRANS-9-ALKYL-2-BENZYL-5-METHYL-6,7-BENZOMORPHANS
Authors: DEHGHANI A BAI X MASCARELLA SW BOWEN WD CARROLL FI
Citation: A. Dehghani et al., A NOVEL STEREOSELECTIVE AND ENANTIOSELECTIVE SYNTHESIS OF TRANS-9-ALKYL-2-BENZYL-5-METHYL-6,7-BENZOMORPHANS, Tetrahedron letters, 35(48), 1994, pp. 8969-8972
A NOVEL ASYMMETRIC-SYNTHESIS OF ,5,6-HEXAHYDRO-11-ALKYL-2,6-METHANO-3-BENZAZOCINES
Authors: BAI X MASCARELLA SW BOWEN WD CARROLL FI
Citation: X. Bai et al., A NOVEL ASYMMETRIC-SYNTHESIS OF ,5,6-HEXAHYDRO-11-ALKYL-2,6-METHANO-3-BENZAZOCINES, Journal of the Chemical Society, Chemical Communications, (20), 1994, pp. 2401-2402
SYNTHESIS, LIGAND-BINDING, AND QSAR (COMFA AND CLASSICAL) STUDY OF 3-BETA-(3'-SUBSTITUTED PHENYL), 3-BETA-(4'-SUBSTITUTED PHENYL), AND 3-BETA-(3',4'-DISUBSTITUTED PHENYL)TROPANE-2-BETA-CARBOXYLIC ACID METHYL-ESTERS
Authors: CARROLL FI MASCARELLA SW KUZEMKO MA GAO YG ABRAHAM P LEWIN AH BOJA JW KUHAR MJ
Citation: Fi. Carroll et al., SYNTHESIS, LIGAND-BINDING, AND QSAR (COMFA AND CLASSICAL) STUDY OF 3-BETA-(3'-SUBSTITUTED PHENYL), 3-BETA-(4'-SUBSTITUTED PHENYL), AND 3-BETA-(3',4'-DISUBSTITUTED PHENYL)TROPANE-2-BETA-CARBOXYLIC ACID METHYL-ESTERS, Journal of medicinal chemistry, 37(18), 1994, pp. 2865-2873
SYNTHESIS AND STRUCTURAL DETERMINATION OF 5H-BENZOCYCLOHEPTEN-5,8-IMINES
Authors: DICESARE JC BURGESS JP MASCARELLA SW CARROLL FI ROTHMAN RB
Citation: Jc. Dicesare et al., SYNTHESIS AND STRUCTURAL DETERMINATION OF 5H-BENZOCYCLOHEPTEN-5,8-IMINES, Journal of heterocyclic chemistry, 31(1), 1994, pp. 187-192
SYNTHESIS OF L-2,3,4,5-TETRAHYDRO-2,5-METHANO-1H-2-BENZAZEPINES AND THEIR REARRANGEMENT TO O-1,2,3,4,5,6-HEXAHYDRO-2,6-METHANO-2-BENZAZOCINES
Authors: BLOUGH BE MASCARELLA SW ROTHMAN RB CARROLL FI
Citation: Be. Blough et al., SYNTHESIS OF L-2,3,4,5-TETRAHYDRO-2,5-METHANO-1H-2-BENZAZEPINES AND THEIR REARRANGEMENT TO O-1,2,3,4,5,6-HEXAHYDRO-2,6-METHANO-2-BENZAZOCINES, Journal of the Chemical Society, Chemical Communications, (9), 1993, pp. 758-760
A COMPARISON OF (-)-DEOXYBENZOMORPHANS DEVOID OF OPIATE ACTIVITY WITHTHEIR DEXTROROTATORY PHENOLIC COUNTERPARTS SUGGESTS ROLE OF SIGMA(2) RECEPTORS IN MOTOR FUNCTION (VOL 231, PG 61, 1993)
Authors: WALKER JM BOWEN WD PATRICK SL WILLIAMS WE MASCARELLA SW BAI X CARROLL FI
Citation: Jm. Walker et al., A COMPARISON OF (-)-DEOXYBENZOMORPHANS DEVOID OF OPIATE ACTIVITY WITHTHEIR DEXTROROTATORY PHENOLIC COUNTERPARTS SUGGESTS ROLE OF SIGMA(2) RECEPTORS IN MOTOR FUNCTION (VOL 231, PG 61, 1993), European journal of pharmacology, 236(3), 1993, pp. 495-495
Risultati: 1-19 |