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Results: 1-13 |
Results: 13

Authors: MEDERSKI WWKR DORSCH D OSSWALD M ANZALI S CHRISTADLER M SCHMITGES CJ SCHELLING P WILM C FLUCK M
Citation: Wwkr. Mederski et al., 3 - ENDOTHELIN ANTAGONISTS - DISCOVERY OF EMD-122946, A HIGHLY POTENTAND ORALLY-ACTIVE ETA SELECTIVE ANTAGONIST, Bioorganic & medicinal chemistry letters, 8(13), 1998, pp. 1771-1776

Authors: ANZALI S MEDERSKI WWKR OSSWALD M DORSCH D
Citation: S. Anzali et al., 1 - ENDOTHELIN ANTAGONISTS - SEARCH FOR SURROGATES OF METHYLENDIOXYPHENYL BY MEANS OF A KOHONEN NEURAL-NETWORK, Bioorganic & medicinal chemistry letters, 8(1), 1998, pp. 11-16

Authors: MEDERSKI WWKR OSSWALD M DORSCH D ANZALI S CHRISTADLER M SCHMITGES CJ WILM C
Citation: Wwkr. Mederski et al., 2 - ENDOTHELIN ANTAGONISTS - EVALUATION OF 2,1,3-BENZOTHIADIAZOLE AS A METHYLENDIOXYPHENYL BIOISOSTER, Bioorganic & medicinal chemistry letters, 8(1), 1998, pp. 17-22

Authors: DORSCH D MEDERSKI WWKR OSSWALD M DEVANT RM SCHMITGES CJ CHRISTADLER M WILM C
Citation: D. Dorsch et al., PYRIDAZINONES WITH A PENDANT ACYLSULFONAMIDE MOIETY AS ENDOTHELIN RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 7(3), 1997, pp. 275-280

Authors: MEDERSKI WWKR OSSWALD M DORSCH D CHRISTADLER M SCHMITGES CJ WILM C
Citation: Wwkr. Mederski et al., ,4-DIARYL-2-OXO-1,2-DIHYRDO-QUINOLINE-3-CARBOXYLIC ACIDS AS ENDOTHELIN RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 7(14), 1997, pp. 1883-1886

Authors: MEDERSKI WWKR DORSCH D OSSWALD M SCHWARTZ H BEIER N CHRISTADLER M MINCK KO SCHELLING P SCHMITGES CJ
Citation: Wwkr. Mederski et al., NOVEL 4,5-DIHYDRO-4-OXO-3H-IMIDAZO[4,5-C]PYRIDINES - POTENT ANGIOTENSIN-II RECEPTOR ANTAGONISTS WITH HIGH-AFFINITY FOR BOTH THE AT(1) AND AT(2) SUBTYPES, European journal of medicinal chemistry, 32(6), 1997, pp. 479-491

Authors: MEDERSKI WWKR DORSCH D OSSWALD M BEIER N LUES I MINCK KO SCHELLING P LADSTETTER BJ
Citation: Wwkr. Mederski et al., 4,5-DIHYDRO-4-OXO-3H-IMIDAZO[4,5-C]PYRIDINES - POTENT ARYLACETIC ACID-DERIVED AT(1) ANTAGONISTS WITH IMPROVED AFFINITY FOR THE AT(2) RECEPTOR, Bioorganic & medicinal chemistry letters, 5(22), 1995, pp. 2665-2670

Authors: DORSCH D MEDERSKI WWKR OSSWALD M BEIER N SCHELLING P
Citation: D. Dorsch et al., URACIL-BASED ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 5(18), 1995, pp. 2071-2076

Authors: KOPPE T MEDERSKI WWKR OSSWALD M SCHWARZ M
Citation: T. Koppe et al., ON THE REGIOCHEMISTRY OF THE ALKYLATION OF TERT-BUTYL -BUTYL-1,2-DIHYDRO-2-OXO-3-PYRIDYLMETHYL]CARBAMATE - PRECURSOR OF A SERIES OF POTENT ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Tetrahedron letters, 36(3), 1995, pp. 377-380

Authors: OSSWALD M MEDERSKI WWKR SCHWARZ M BEIER N LUES I MINCK KO
Citation: M. Osswald et al., 3-SUBSTITUTED 6-BUTYL-1,2-DIHYDROPYRIDIN-2-ONES - A NEW SERIES OF POTENT NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(5), 1994, pp. 683-688

Authors: DORSCH D MEDERSKI WWKR BEIER N LUES I MINCK KO SCHELLING P
Citation: D. Dorsch et al., (6-OXO-3-PYRIDAZINYL)-BENZIMIDAZOLES AS POTENT ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(11), 1994, pp. 1297-1302

Authors: BEIER N LABITZKE E MEDERSKI WWKR RADUNZ HE RAUSCHENBACHRUESS K SCHNEIDER B
Citation: N. Beier et al., SYNTHESIS OF 7-ETHYL-1,2-DIHYDROQUINOLIN-2-ONES AS ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Heterocycles, 39(1), 1994, pp. 117-131

Authors: MEDERSKI WWKR DORSCH D BOKEL HH BEIER N LUES I SCHELLING P
Citation: Wwkr. Mederski et al., NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A SERIES OF NOVEL 4,5-DIHYDRO-4-OXO-3H-IMIDAZO[4,5-C]PYRIDINE DERIVATIVES, Journal of medicinal chemistry, 37(11), 1994, pp. 1632-1645
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