Authors:
ELLIOTT JM
CASCIERI MA
CHICCHI G
DAVIES S
KELLEHER FJ
KURTZ M
LADDUWAHETTY T
LEWIS RT
MACLEOD AM
MERCHANT KJ
SADOWSKI S
STEVENSON GI
Citation: Jm. Elliott et al., SERINE DERIVED NK1 ANTAGONISTS 1 - THE EFFECT OF MODIFICATIONS TO THESERINE SUBSTITUENTS, Bioorganic & medicinal chemistry letters, 8(14), 1998, pp. 1845-1850
Authors:
STEVENSON GI
HUSCROFT I
MACLEOD AM
SWAIN CJ
CASCIERI MA
CHICCHI GG
GRAHAM MI
HARRISON T
KELLEHER FJ
KURTZ M
LADDUWAHETTY T
MERCHANT KJ
METZGER JM
MACINTYRE DE
SADOWSKI S
SOHAL B
OWENS AP
Citation: Gi. Stevenson et al., 4,4-DISUBSTITUTED PIPERIDINE HIGH-AFFINITY NK1 ANTAGONISTS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND IN-VIVO ACTIVITY, Journal of medicinal chemistry, 41(23), 1998, pp. 4623-4635
Authors:
LEWIS RT
MACLEOD AM
MERCHANT KJ
KELLEHER F
SANDERSON I
HERBERT RH
CASCIERI MA
SADOWSKI S
BALL RG
HOOGSTEEN K
Citation: Rt. Lewis et al., TRYPTOPHAN-DERIVED NK1 ANTAGONISTS - CONFORMATIONALLY CONSTRAINED HETEROCYCLIC BIOISOSTERES OF THE ESTER LINKAGE, Journal of medicinal chemistry, 38(6), 1995, pp. 923-933
Authors:
MACLEOD AM
CASCIERI MA
MERCHANT KJ
SADOWSKI S
HARDWICKE S
LEWIS RT
MACINTYRE DE
METZGER JM
FONG TM
SHEPHEARD S
TATTERSALL FD
HARGREAVES R
BAKER R
Citation: Am. Macleod et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF NK1 ANTAGONISTS DERIVED FROM L-TRYPTOPHAN, Journal of medicinal chemistry, 38(6), 1995, pp. 934-941
Authors:
SWAIN CJ
SEWARD EM
CASCIERI MA
FONG TM
HERBERT R
MACINTYRE DE
MERCHANT KJ
OWEN SN
OWENS AP
SABIN V
TEALL M
VANNIEL MB
WILLIAMS BJ
SADOWSKI S
STRADER C
BALL RG
BAKER R
Citation: Cj. Swain et al., IDENTIFICATION OF A SERIES OF 3-(BENZYLOXY)-1-AZABICYCLO[2.2.2]OCTANEHUMAN NK1 ANTAGONISTS, Journal of medicinal chemistry, 38(24), 1995, pp. 4793-4805
Authors:
MACLEOD M
MERCHANT KJ
BROOKFIELD F
KELLEHER F
STEVENSON G
OWENS AP
SWAIN CJ
BAKER R
CASCIERI MA
SADOWSKI S
BER E
STRADER CD
MACINTYRE DE
METZGER JM
BALL RG
Citation: M. Macleod et al., IDENTIFICATION OF L-TRYPTOPHAN DERIVATIVES WITH POTENT AND SELECTIVE ANTAGONIST ACTIVITY AT THE NK1 RECEPTOR, Journal of medicinal chemistry, 37(9), 1994, pp. 1269-1274
Authors:
CASCIERI MA
MACLEOD AM
UNDERWOOD D
SHIAO LL
BER E
SADOWSKI S
YU H
MERCHANT KJ
SWAIN CJ
STRADER CD
FONG TM
Citation: Ma. Cascieri et al., CHARACTERIZATION OF THE INTERACTION OF N-ACYL-L-TRYPTOPHAN BENZYL ESTER NEUROKININ ANTAGONISTS WITH THE HUMAN NEUROKININ-1 RECEPTOR, The Journal of biological chemistry, 269(9), 1994, pp. 6587-6591