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Results: 1-17 |
Results: 17
A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor
Authors: DeVita, RJ Walsh, TF Young, JR Jiang, JL Ujjainwalla, F Toupence, RB Parikh, M Huang, SX Fair, JA Goulet, MT Wyvratt, MJ Lo, JL Ren, N Yudkovitz, JB Yang, YT Cheng, K Cui, JS Mount, G Rohrer, SP Schaeffer, JM Rhodes, L Drisko, JE McGowan, E MacIntyre, DE Vincent, S Carlin, JR Cameron, J Smith, RG
Citation: Rj. Devita et al., A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor, J MED CHEM, 44(6), 2001, pp. 917-922
Inactivation of the mouse melanocortin-3 receptor results in increased fatmass and reduced lean body mass
Authors: Chen, AS Marsh, DJ Trumbauer, ME Frazier, EG Guan, XM Yu, H Rosenblum, CI Vongs, A Feng, Y Cao, LH Metzger, JM Strack, AM Camacho, RE Mellin, TN Nunes, CN Min, W Fisher, J Gopal-Truter, S MacIntyre, DE Chen, HY Van der Ploeg, LHT
Citation: As. Chen et al., Inactivation of the mouse melanocortin-3 receptor results in increased fatmass and reduced lean body mass, NAT GENET, 26(1), 2000, pp. 97-102
Role of the melanocortin-4 receptor in metabolic rate and food intake in mice
Authors: Chen, AS Metzger, JM Trumbauer, ME Guan, XM Yu, H Frazier, EG Marsh, DJ Forrest, MJ Gopal-Truter, S Fisher, J Camacho, RE Strack, AM Mellin, TN MacIntyre, DE Chen, HY Van der Ploeg, LHT
Citation: As. Chen et al., Role of the melanocortin-4 receptor in metabolic rate and food intake in mice, TRANSGEN RE, 9(2), 2000, pp. 145-154
Human beta 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
Authors: Brockunier, LL Parmee, ER Ok, HO Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Ll. Brockunier et al., Human beta 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides, BIOORG MED, 10(18), 2000, pp. 2111-2114
Potent, selective 3-pyridylethanolamine beta(3) adrenergic receptor agonists possessing a thiazole benzenesulfonamide pharmacophore
Authors: Mathvink, RJ Tolman, JS Chitty, D Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Rj. Mathvink et al., Potent, selective 3-pyridylethanolamine beta(3) adrenergic receptor agonists possessing a thiazole benzenesulfonamide pharmacophore, BIOORG MED, 10(17), 2000, pp. 1971-1973
Substituted oxazole benzenesulfonamides as potent human beta(3) adrenergicreceptor agonists
Authors: Ok, HO Reigle, LB Candelore, MR Cascieri, MA Colwell, LF Deng, L Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Strader, CD Tota, L Wang, P Wyvratt, MJ Fisher, MH Weber, AE
Citation: Ho. Ok et al., Substituted oxazole benzenesulfonamides as potent human beta(3) adrenergicreceptor agonists, BIOORG MED, 10(14), 2000, pp. 1531-1534
Discovery of an orally bioavailable alkyl oxadiazole beta(3) adrenergic receptor agonist
Authors: Feng, DQD Biftu, T Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Dqd. Feng et al., Discovery of an orally bioavailable alkyl oxadiazole beta(3) adrenergic receptor agonist, BIOORG MED, 10(13), 2000, pp. 1427-1429
Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective beta(3) adrenergic receptor agonist antiobesity agents
Authors: Biftu, T Feng, DD Liang, GB Kuo, H Qian, XX Naylor, EM Colandrea, VJ Candelore, MR Cascieri, MA Colwell, LF Forrest, MJ Hom, GJ MacIntyre, DE Stearns, RA Strader, CD Wyvratt, MJ Fisher, MH Weber, AE
Citation: T. Biftu et al., Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective beta(3) adrenergic receptor agonist antiobesity agents, BIOORG MED, 10(13), 2000, pp. 1431-1434
The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L758,298, inhibit acute and delayed cisplatin-inducedemesis in ferrets
Authors: Tattersall, FD Rycroft, W Cumberbatch, M Mason, G Tye, S Williamson, DJ Hale, JJ Mills, SG Finke, PE MacCoss, M Sadowski, S Ber, E Cascieri, M Hill, RG MacIntyre, DE Hargreaves, RJ
Citation: Fd. Tattersall et al., The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L758,298, inhibit acute and delayed cisplatin-inducedemesis in ferrets, NEUROPHARM, 39(4), 2000, pp. 652-663
Phosphorylated morpholine acetal human neurokinin-1 receptor antagonists as water-soluble prodrugs
Authors: Hale, JJ Mills, SG MacCoss, M Dorn, CP Finke, PE Budhu, RJ Reamer, RA Huskey, SEW Luffer-Atlas, D Dean, BJ McGowan, EM Feeney, WP Chiu, SHL Cascieri, MA Chicchi, GG Kurtz, MM Sadowski, S Ber, E Tattersall, FD Rupniak, NMJ Williams, AR Rycroft, W Hargreaves, R Metzger, JM MacIntyre, DE
Citation: Jj. Hale et al., Phosphorylated morpholine acetal human neurokinin-1 receptor antagonists as water-soluble prodrugs, J MED CHEM, 43(6), 2000, pp. 1234-1241
Discovery of a potent, orally bioavailable beta(3) adrenergic receptor agonist, (R)-N-[4-[2-[[2-hydroxy-2-(3-pyridinyl)ethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide
Authors: Mathvink, RJ Tolman, JS Chitty, D Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Rj. Mathvink et al., Discovery of a potent, orally bioavailable beta(3) adrenergic receptor agonist, (R)-N-[4-[2-[[2-hydroxy-2-(3-pyridinyl)ethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide, J MED CHEM, 43(21), 2000, pp. 3832-3836
L-770,644: A potent and selective human beta(3) adrenergic receptor agonist with improved oral bioavailability
Authors: Shih, TL Candelore, MR Cascieri, MA Chiu, SHL Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Tl. Shih et al., L-770,644: A potent and selective human beta(3) adrenergic receptor agonist with improved oral bioavailability, BIOORG MED, 9(9), 1999, pp. 1251-1254
Human beta(3) adrenergic receptor agonists containing cyclic ureidobenzenesulfonamides
Authors: Parmee, ER Naylor, EM Perkins, L Colandrea, VJ Ok, HO Candelore, MR Cascieri, MA Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Er. Parmee et al., Human beta(3) adrenergic receptor agonists containing cyclic ureidobenzenesulfonamides, BIOORG MED, 9(5), 1999, pp. 749-754
Human beta(3) adrenergic receptor agonists containing imidazolidinone and imidazolone benzenesulfonamides
Authors: Naylor, EM Parmee, ER Colandrea, VJ Perkins, L Brockunier, L Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Strader, CD Tota, L Wang, PR Wyvratt, MJ Fisher, MH Weber, AE
Citation: Em. Naylor et al., Human beta(3) adrenergic receptor agonists containing imidazolidinone and imidazolone benzenesulfonamides, BIOORG MED, 9(5), 1999, pp. 755-758
The effects of IB4, a monoclonal antibody to the CD18 leukocyte integrin on phorbol myristate acetate (PMA)-induced polymorphonuclear leukocyte (PMN)accumulation and endothelial injury in rabbit lungs
Authors: Meurer, RD Forrest, MJ MacIntyre, DE
Citation: Rd. Meurer et al., The effects of IB4, a monoclonal antibody to the CD18 leukocyte integrin on phorbol myristate acetate (PMA)-induced polymorphonuclear leukocyte (PMN)accumulation and endothelial injury in rabbit lungs, INFLAMMATIO, 23(1), 1999, pp. 51-62
Production of leptin in Escherichia coli: A comparison of methods
Authors: Varnerin, JP Smith, T Rosenblum, CI Vongs, A Murphy, BA Nunes, C Mellin, TN King, JJ Burgess, BW Junker, B Chou, M Hey, P Frazier, E MacIntyre, DE Van der Ploeg, LHT Tota, MR
Citation: Jp. Varnerin et al., Production of leptin in Escherichia coli: A comparison of methods, PROT EX PUR, 14(3), 1998, pp. 335-342
Melanocortin mediated inhibition of feeding behavior in rats
Authors: Murphy, B Nunes, CN Ronan, JJ Harper, CM Beall, MJ Hanaway, M Fairhurst, AM Van der Ploeg, LHT MacIntyre, DE Mellin, TN
Citation: B. Murphy et al., Melanocortin mediated inhibition of feeding behavior in rats, NEUROPEPTID, 32(6), 1998, pp. 491-497
Risultati: 1-17 |