AAAAAA

   
Results: 1-20 |
Results: 20
Central effects of urotensin-II following ICV administration in rats
Authors: Gartlon, J Parker, F Harrison, DC Douglas, SA Ashmeade, TE Riley, GJ Hughes, ZA Taylor, SG Munton, RP Hagan, JJ Hunter, JA Jones, DNC
Citation: J. Gartlon et al., Central effects of urotensin-II following ICV administration in rats, PSYCHOPHAR, 155(4), 2001, pp. 426-433
Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinityand selectivity for the dopamine D-3 receptor
Authors: Austin, NE Avenell, KY Boyfield, I Branch, CL Hadley, MS Jeffrey, P Johnson, CN Macdonald, GJ Nash, DJ Riley, GJ Smith, AB Stemp, G Thewlis, KM Vong, AKK Wood, MD
Citation: Ne. Austin et al., Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinityand selectivity for the dopamine D-3 receptor, BIOORG MED, 11(5), 2001, pp. 685-688
Evaluation of a series of anticonvulsant 1,2,3,4-tetrahydroisoquinolinyl-benzamides
Authors: Chan, WN Hadley, MS Darling, JD Herdon, HJ Orlek, BS Riley, GJ Stead, REA Stean, TO Thompson, M Upton, N Ward, RW
Citation: Wn. Chan et al., Evaluation of a series of anticonvulsant 1,2,3,4-tetrahydroisoquinolinyl-benzamides, BIO MED CH, 8(8), 2000, pp. 2085-2094
Novel 2,3,4,5-tetrahydro-1H-3-benzazepines with high affinity and selectivity for the dopamine D-3 receptor
Authors: Austin, NE Avenell, KY Boyfield, I Branch, CL Hadley, MS Jeffrey, P Johnson, CN Macdonald, GJ Nash, DJ Riley, GJ Smith, AB Stemp, G Thewlis, KM Vong, AKK Wood, M
Citation: Ne. Austin et al., Novel 2,3,4,5-tetrahydro-1H-3-benzazepines with high affinity and selectivity for the dopamine D-3 receptor, BIOORG MED, 10(22), 2000, pp. 2553-2555
1-[2-[(heteroaryloxy)heteroaryl]carbamoyl]indolines: Novel and selective 5-HT2C receptor inverse agonists with potential as antidepressant/anxiolyticagents
Authors: Bromidge, SM Dabbs, S Davies, S Duckworth, DM Forbes, IT Jones, GE Jones, J King, FD Saunders, DV Blackburn, TP Holland, V Kennett, GA Lightowler, S Middlemiss, DN Riley, GJ Trail, B Wood, MD
Citation: Sm. Bromidge et al., 1-[2-[(heteroaryloxy)heteroaryl]carbamoyl]indolines: Novel and selective 5-HT2C receptor inverse agonists with potential as antidepressant/anxiolyticagents, BIOORG MED, 10(16), 2000, pp. 1863-1866
1-[2-[(heteroarylmethoxy)aryl]carbamoyl]indolines are selective and orallyactive 5-HT2C receptor inverse agonists
Authors: Bromidge, SM Davies, S Duckworth, DM Forbes, IT Jones, GE Jones, J King, FD Blackburn, TP Holland, V Kennett, GA Lightowler, S Middlemiss, DN Riley, GJ Trail, B Wood, MD
Citation: Sm. Bromidge et al., 1-[2-[(heteroarylmethoxy)aryl]carbamoyl]indolines are selective and orallyactive 5-HT2C receptor inverse agonists, BIOORG MED, 10(16), 2000, pp. 1867-1870
Pharmacological actions of a novel, high-affinity, and selective human dopamine D-3 receptor antagonist, SB-277011-A
Authors: Reavill, C Taylor, SG Wood, MD Ashmeade, T Austin, NE Avenell, KY Boyfield, I Branch, CL Cilia, J Coldwell, MC Hadley, MS Hunter, AJ Jeffrey, P Jewitt, F Johnson, CN Jones, DNC Medhurst, AD Middlemiss, DN Nash, DJ Riley, GJ Routledge, C Stemp, G Thewlis, KM Trail, B Vong, AKK Hagan, JJ
Citation: C. Reavill et al., Pharmacological actions of a novel, high-affinity, and selective human dopamine D-3 receptor antagonist, SB-277011-A, J PHARM EXP, 294(3), 2000, pp. 1154-1165
Design and synthesis of trans-N-[4-[2-(6-cyano-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A potent and selective dopamine D-3 receptor antagonist with high oral bioavailability and CNS penetration in the rat
Authors: Stemp, G Ashmeade, T Branch, CL Hadley, MS Hunter, AJ Johnson, CN Nash, DJ Thewlis, KM Vong, AKK Austin, NE Jeffrey, P Avenell, KY Boyfield, I Hagan, JJ Middlemiss, DN Reavill, C Riley, GJ Routledge, C Wood, M
Citation: G. Stemp et al., Design and synthesis of trans-N-[4-[2-(6-cyano-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A potent and selective dopamine D-3 receptor antagonist with high oral bioavailability and CNS penetration in the rat, J MED CHEM, 43(9), 2000, pp. 1878-1885
Biarylcarbamoylindolines are novel and selective 5-HT2C receptor inverse agonists: Identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent
Authors: Bromidge, SM Dabbs, S Davies, DT Davies, S Duckworth, DM Forbes, IT Gaster, LM Ham, P Jones, GE King, FD Mulholland, KR Saunders, DV Wyman, PA Blaney, FE Clarke, SE Blackburn, TP Holland, V Kennett, GA Lightowler, S Middlemiss, DN Trail, B Riley, GJ Wood, MD
Citation: Sm. Bromidge et al., Biarylcarbamoylindolines are novel and selective 5-HT2C receptor inverse agonists: Identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent, J MED CHEM, 43(6), 2000, pp. 1123-1134
A novel, potent, and selective 5-HT7 antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)-ethyl)pyrrolidine-1-sulfonyl)phenol (SB-269970)
Authors: Lovell, PJ Bromidge, SM Dabbs, S Duckworth, DM Forbes, IT Jennings, AJ King, FD Middlemiss, DN Rahman, SK Saunders, DV Collin, LL Hagan, JJ Riley, GJ Thomas, DR
Citation: Pj. Lovell et al., A novel, potent, and selective 5-HT7 antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)-ethyl)pyrrolidine-1-sulfonyl)phenol (SB-269970), J MED CHEM, 43(3), 2000, pp. 342-345
Evidence for antagonist activity of the dopamine D3 receptor partial agonist, BP 897, at human dopamine D3 receptor
Authors: Wood, MD Boyfield, I Nash, DJ Jewitt, FR Avenell, KY Riley, GJ
Citation: Md. Wood et al., Evidence for antagonist activity of the dopamine D3 receptor partial agonist, BP 897, at human dopamine D3 receptor, EUR J PHARM, 407(1-2), 2000, pp. 47-51
Characterization of SB-269970-A, a selective 5-HT7 receptor antagonist
Authors: Hagan, JJ Price, GW Jeffrey, P Deeks, NJ Stean, T Piper, D Smith, MI Upton, N Medhurst, AD Middlemiss, DN Riley, GJ Lovell, PJ Bromidge, SM Thomas, DR
Citation: Jj. Hagan et al., Characterization of SB-269970-A, a selective 5-HT7 receptor antagonist, BR J PHARM, 130(3), 2000, pp. 539-548
Selective serotonin receptor uptake inhibitors can reduce restless legs symptoms
Authors: Dimmitt, SB Riley, GJ
Citation: Sb. Dimmitt et Gj. Riley, Selective serotonin receptor uptake inhibitors can reduce restless legs symptoms, ARCH IN MED, 160(5), 2000, pp. 712-712
Model studies on a synthetically facile series of N-substituted phenyl-N '-pyridin-3-yl ureas leading to 1-(3-pyridylcarbamoyl) indolines that are potent and selective 5-HT2C/2B receptor antagonists
Authors: Bromidge, SM Dabbs, S Davies, DT Davies, S Duckworth, DM Forbes, IT Gadre, A Ham, P Jones, GE King, FD Saunders, DV Thewlis, KM Vyas, D Blackburn, TP Holland, V Kennett, GA Riley, GJ Wood, MD
Citation: Sm. Bromidge et al., Model studies on a synthetically facile series of N-substituted phenyl-N '-pyridin-3-yl ureas leading to 1-(3-pyridylcarbamoyl) indolines that are potent and selective 5-HT2C/2B receptor antagonists, BIO MED CH, 7(12), 1999, pp. 2767-2773
Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D-3 receptor
Authors: Austin, NE Avenell, KY Boyfield, I Branch, CL Coldwell, MC Hadley, MS Jeffrey, P Johns, A Johnson, CN Nash, DJ Riley, GJ Smith, SA Stacey, RC Stemp, G Thewlis, KM Vong, AKK
Citation: Ne. Austin et al., Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D-3 receptor, BIOORG MED, 9(2), 1999, pp. 179-184
Heterocyclic analogues of 2-aminotetralins with high affinity and selectivity for the dopamine D-3 receptor
Authors: Avenell, KY Boyfield, I Hadley, MS Johnson, CN Nash, DJ Riley, GJ Stemp, G
Citation: Ky. Avenell et al., Heterocyclic analogues of 2-aminotetralins with high affinity and selectivity for the dopamine D-3 receptor, BIOORG MED, 9(18), 1999, pp. 2715-2720
Placental protein 14 functions as a direct T-cell inhibitor
Authors: Rachmilewitz, J Riley, GJ Tykocinski, ML
Citation: J. Rachmilewitz et al., Placental protein 14 functions as a direct T-cell inhibitor, CELL IMMUN, 191(1), 1999, pp. 26-33
An empirical model for predicting the foundation modulus of wood for metal-plate connector teeth
Authors: Riley, GJ Gebremedhin, KG
Citation: Gj. Riley et Kg. Gebremedhin, An empirical model for predicting the foundation modulus of wood for metal-plate connector teeth, T ASAE, 42(3), 1999, pp. 755-760
Axial and rotational stiffness model of metal-plate-connected wood truss joints
Authors: Riley, GJ Gebremedhin, KG
Citation: Gj. Riley et Kg. Gebremedhin, Axial and rotational stiffness model of metal-plate-connected wood truss joints, T ASAE, 42(3), 1999, pp. 761-770
Functional effects of the muscarinic receptor agonist, xanomeline, at 5-HT1 and 5-HT2 receptors
Authors: Watson, J Brough, S Coldwell, MC Gager, T Ho, M Hunter, AJ Jerman, J Middlemiss, DN Riley, GJ Brown, AM
Citation: J. Watson et al., Functional effects of the muscarinic receptor agonist, xanomeline, at 5-HT1 and 5-HT2 receptors, BR J PHARM, 125(7), 1998, pp. 1413-1420
Risultati: 1-20 |