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Citation: Na. Powell et Wr. Roush, Studies on the total synthesis of formamicin: Synthesis of the C(1)-C(11) fragment, ORG LETT, 3(3), 2001, pp. 453-456
Citation: Bm. Savall et al., Highly diastereoselective synthesis of propargylic 1,2-anti-diol derivatives using alpha-alkoxypropargylstannanes, ORG LETT, 3(19), 2001, pp. 3057-3060
Citation: Gc. Micalizio et Wr. Roush, Studies on the synthesis of pectenotoxin II: Synthesis of a C(11)-C(26) fragment precursor via [3+2]-annulation reactions of chiral allylsilanes, ORG LETT, 3(12), 2001, pp. 1949-1952
Authors:
Menard, R
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Citation: R. Menard et al., Cathepsins X and B display distinct activity profiles that can be exploited for inhibitor design, BIOL CHEM, 382(5), 2001, pp. 839-845
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Roush, WR
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Citation: Wr. Roush et al., Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain, BIOORG MED, 11(20), 2001, pp. 2759-2762
Citation: Wr. Roush et Gj. Dilley, Studies on the synthesis of 2,6-disubstituted dihydropyrans: Intervention of oxonia-Cope rearrangements in the Lewis acid mediated cyclodehydrative reactions of aldehydes and beta-hydroxyallylsilanes, SYNLETT, 2001, pp. 955-959
Citation: Wr. Roush et al., Studies on the synthesis of landomycin A: Synthesis and glycosidation reactions of L-rhodinosyl acetate derivatives, J ORG CHEM, 66(19), 2001, pp. 6389-6393
Authors:
Therrien, C
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Citation: C. Therrien et al., Cathepsins X and B can be differentiated through their respective mono- and dipeptidyl carboxypeptidase activities, BIOCHEM, 40(9), 2001, pp. 2702-2711
Citation: Gc. Micalizio et Wr. Roush, A three-component coupling strategy for tetrahydrofuran synthesis: Application of the diisopropyl tartrate modified (E)-gamma-(dimethylphenylsilyl)allylboronate as an alpha,gamma-allyl dianion equivalent, ORG LETT, 2(4), 2000, pp. 461-464
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Brinen, LS
Hansell, E
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Citation: Ls. Brinen et al., A target within the target: probing Cruzain's P1 ' site to define structural determinants for the Chagas' disease protease, STRUCT F D, 8(8), 2000, pp. 831-840
Citation: Wr. Roush et al., [(E)-gamma-(dimethylphenylsilyl)allyl]diisopinocampheylborane: a highly enantioselective reagent for the synthesis of anti-beta-hydroxyallylsilanes, TETRAHEDR L, 41(49), 2000, pp. 9413-9417
Authors:
Roush, WR
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Hansell, E
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Citation: Wr. Roush et al., Design, synthesis and evaluation of D-homophenylalanyl epoxysuccinate inhibitors of the trypanosomal cysteine protease cruzain, TETRAHEDRON, 56(50), 2000, pp. 9747-9762
Citation: Gc. Micalizio et al., Synthesis of the C(29)-C(45) bis-pyran subunit (E-F) of spongistatin 1 (altohyrtin A), J ORG CHEM, 65(25), 2000, pp. 8730-8736
Citation: Sa. Frank et al., Studies on the synthesis of the decahydro-as-indacene ring system of (-)-spinosyn A via transannular Diels-Alder reactions of substituted (E,E,E)-cyclododeca-1,6,8-trienes, CAN J CHEM, 78(6), 2000, pp. 757-771
Citation: Wr. Roush et Ce. Bennett, A highly stereoselective synthesis of the landomycin A hexasaccharide unit, J AM CHEM S, 122(25), 2000, pp. 6124-6125
Citation: Wr. Roush et al., 2-Deoxy-2-iodo- and 2-deoxy-2-bromo-alpha-glucopyranosyl trichloroacetimidates: Highly reactive and stereoselective donors for the synthesis of 2-deoxy-beta-glycosides, ORG LETT, 1(6), 1999, pp. 891-893
Authors:
Roush, WR
Narayan, S
Bennett, CE
Briner, K
Citation: Wr. Roush et al., Iodoacetoxylation of glycals using cerium(IV) ammonium nitrate, sodium iodide, and acetic acid: Stereoselective synthesis of 2-deoxy-2-iodo-alpha-mannopyranosyl acetates, ORG LETT, 1(6), 1999, pp. 895-897
Citation: Wr. Roush et S. Narayan, 2-deoxy-2-iodo-alpha-mannopyranosyl and -talopyranosyl acetates: Highly stereoselective glycosyl donors for the synthesis of 2-deoxy-alpha-glycosides, ORG LETT, 1(6), 1999, pp. 899-902
Citation: Wr. Roush et Gc. Lane, Studies on the synthesis of tedanolide: Synthesis of the C(5)-C(21) segment via a highly stereoselective fragment assembly aldol reaction of a chiralbeta,gamma-unsaturated methyl ketone, ORG LETT, 1(1), 1999, pp. 95-98
Authors:
Scheidt, KA
Tasaka, A
Bannister, TD
Wendt, MD
Roush, WR
Citation: Ka. Scheidt et al., Total synthesis of (-)-bafilomycin A(1): Application of diastereoselectivecrotylboration and methyl ketone aldol reactions, ANGEW CHEM, 38(11), 1999, pp. 1652-1655
Citation: Sr. Chemler et al., An improved synthesis of the (E,Z)-Dienoate precursor of (+)-damavaricin Dvia a vinylogous Horner-Eadsworth-Emmons reaction, TETRAHEDR L, 40(7), 1999, pp. 1269-1272
Citation: Wr. Roush et Gj. Dilley, Studies of fragment assembly aldol reactions of chiral aldehydes and chiral methyl ketones: stereoselective synthesis of the C(13)-C(25) segment of scytophycin C, TETRAHEDR L, 40(27), 1999, pp. 4955-4959