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Results: 1-23 |
Results: 23
Potent and specific inhibitors of trypanothione reductase from Trypanosomacruzi: Bis(2-aminodiphenylsulfides) for fluorescent labeling studies
Authors: Girault, S Davioud-Charvet, E Maes, L Dubremetz, JF Debreu, MA Landry, V Sergheraert, C
Citation: S. Girault et al., Potent and specific inhibitors of trypanothione reductase from Trypanosomacruzi: Bis(2-aminodiphenylsulfides) for fluorescent labeling studies, BIO MED CH, 9(4), 2001, pp. 837-846
A role for MAP kinase in regulating ectodomain shedding of APLP2 in corneal epithelial cells
Authors: Xu, KP Zoukhri, D Zieske, JD Dartt, DA Sergheraert, C Loing, E Yu, FSX
Citation: Kp. Xu et al., A role for MAP kinase in regulating ectodomain shedding of APLP2 in corneal epithelial cells, AM J P-CELL, 281(2), 2001, pp. C603-C614
Evidence for an endocannabinoid system in the central nervous system of the leech Hirudo medicinalis
Authors: Matias, I Bisogno, T Melck, D Vandenbulcke, F Verger-Bocquet, M De Petrocellis, L Sergheraert, C Breton, C Di Marzo, V Salzet, M
Citation: I. Matias et al., Evidence for an endocannabinoid system in the central nervous system of the leech Hirudo medicinalis, MOL BRAIN R, 87(2), 2001, pp. 145-159
Convenient synthesis of tetrahydroisoquinoline-hydantoins
Authors: Charton, J Delarue, S Vendeville, S Debreu-Fontaine, MA Girault-Mizzi, S Sergheraert, C
Citation: J. Charton et al., Convenient synthesis of tetrahydroisoquinoline-hydantoins, TETRAHEDR L, 42(43), 2001, pp. 7559-7561
Antimalarial in-vivo activity of bis(9-amino-6-chloro-2-methoxyacridines)
Authors: Girault, S Delarue, S Grellier, P Berecibar, A Maes, L Quirijnen, L Lemiere, P Debreu-Fontaine, MA Sergheraert, C
Citation: S. Girault et al., Antimalarial in-vivo activity of bis(9-amino-6-chloro-2-methoxyacridines), J PHARM PHA, 53(7), 2001, pp. 935-938
2-and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: Synthesis and correlation between redox cycling activities and in vitro cytotoxicity
Authors: Salmon-Chemin, L Buisine, E Yardley, V Kohler, S Debreu, MA Landry, V Sergheraert, C Croft, SL Krauth-Siegel, RL Davioud-Charvet, E
Citation: L. Salmon-chemin et al., 2-and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: Synthesis and correlation between redox cycling activities and in vitro cytotoxicity, J MED CHEM, 44(4), 2001, pp. 548-565
A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline
Authors: Davioud-Charvet, E Delarue, S Biot, C Schwobel, B Boehme, CC Mussigbrodt, A Maes, L Sergheraert, C Grellier, P Schirmer, RH Becker, K
Citation: E. Davioud-charvet et al., A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline, J MED CHEM, 44(24), 2001, pp. 4268-4276
Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines
Authors: Delarue, S Girault, S Maes, L Debreu-Fontaine, MA Labaeid, M Grellier, P Sergheraert, C
Citation: S. Delarue et al., Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines, J MED CHEM, 44(17), 2001, pp. 2827-2833
Antiplasmodial activity and cytotoxicity of bis-, tris-, and tetraquinolines with linear or cyclic amino linkers
Authors: Girault, S Grellier, P Berecibar, A Maes, L Lemiere, P Mouray, E Davioud-Charvet, E Sergheraert, C
Citation: S. Girault et al., Antiplasmodial activity and cytotoxicity of bis-, tris-, and tetraquinolines with linear or cyclic amino linkers, J MED CHEM, 44(11), 2001, pp. 1658-1665
Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4-bis{3-[N-(cyclohexyl methyl)amino]propyl}piperazine (vol 484, pg 246, 2000)
Authors: Florent, I Mouray, E Ali, FD Drobecq, H Girault, S Schrevel, J Sergheraert, C Grellier, P
Citation: I. Florent et al., Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4-bis{3-[N-(cyclohexyl methyl)amino]propyl}piperazine (vol 484, pg 246, 2000), FEBS LETTER, 490(1-2), 2001, pp. 102-102
"One-pot" synthesis and antimalarial activity of formamidine derivatives of 4-anilinoquinoline
Authors: Delarue, S Girault, S Ali, FD Maes, L Grellier, P Sergheraert, C
Citation: S. Delarue et al., "One-pot" synthesis and antimalarial activity of formamidine derivatives of 4-anilinoquinoline, CHEM PHARM, 49(8), 2001, pp. 933-937
Trypanothione reductase inhibition/trypanocidal activity relationships in a 1,4-bis(3-aminopropyl)piperazine series
Authors: Bonnet, B Soullez, D Girault, S Maes, L Landry, V Davioud-Charvet, E Sergheraert, C
Citation: B. Bonnet et al., Trypanothione reductase inhibition/trypanocidal activity relationships in a 1,4-bis(3-aminopropyl)piperazine series, BIO MED CH, 8(1), 2000, pp. 95-103
Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi
Authors: Salmon-Chemin, L Lemaire, A De Freitas, S Deprez, B Sergheraert, C Davioud-Charvet, E
Citation: L. Salmon-chemin et al., Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi, BIOORG MED, 10(7), 2000, pp. 631-635
Cholinergic-induced Ca2+ elevation in rat lacrimal gland acini is negatively modulated by PKC delta and PKC epsilon
Authors: Zoukhri, D Hodges, RR Sergheraert, C Dartt, DA
Citation: D. Zoukhri et al., Cholinergic-induced Ca2+ elevation in rat lacrimal gland acini is negatively modulated by PKC delta and PKC epsilon, INV OPHTH V, 41(2), 2000, pp. 386-392
Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): Influence of the linker
Authors: Girault, S Grellier, P Berecibar, A Maes, L Mouray, E Lemiere, P Debreu, MA Davioud-Charvet, E Sergheraert, C
Citation: S. Girault et al., Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): Influence of the linker, J MED CHEM, 43(14), 2000, pp. 2646-2654
Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4-bis{3-[N-(cyclohexyl methyl)amino]propyl}piperazine
Authors: Florenta, I Mouray, E Ali, FD Drobecq, H Girault, S Schrevel, J Sergheraert, C Grellier, P
Citation: I. Florenta et al., Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4-bis{3-[N-(cyclohexyl methyl)amino]propyl}piperazine, FEBS LETTER, 484(3), 2000, pp. 246-252
Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors
Authors: Vendeville, S Bourel, L Davioud-Charvet, E Grellier, P Deprez, B Sergheraert, C
Citation: S. Vendeville et al., Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors, BIOORG MED, 9(3), 1999, pp. 437-442
Synthesis of polyamine derivatives for the preparation of affinity chromatography columns for the search of new Trypanosoma cruzi targets
Authors: Davioud-Charvet, E Berecibar, A Girault, S Landry, V Drobecq, H Sergheraert, C
Citation: E. Davioud-charvet et al., Synthesis of polyamine derivatives for the preparation of affinity chromatography columns for the search of new Trypanosoma cruzi targets, BIOORG MED, 9(11), 1999, pp. 1567-1572
PyBroP: a convenient activator for the synthesis of formamidines
Authors: Delarue, S Sergheraert, C
Citation: S. Delarue et C. Sergheraert, PyBroP: a convenient activator for the synthesis of formamidines, TETRAHEDR L, 40(30), 1999, pp. 5487-5490
Characterization of aggregates of hepatitis C virus glycoproteins
Authors: Choukhi, A Pillez, A Drobecq, H Sergheraert, C Wychowski, C Dubuisson, J
Citation: A. Choukhi et al., Characterization of aggregates of hepatitis C virus glycoproteins, J GEN VIROL, 80, 1999, pp. 3099-3107
Direct evidence of cytoplasmic delivery of PKC-alpha, -epsilon and -zeta pseudosubstrate lipopeptides: study of their implication in the induction ofapoptosis
Authors: Thiam, K Loing, E Zoukhri, D Rommens, C Hodges, R Dartt, D Verwaerde, C Auriault, C Gras-Masse, H Sergheraert, C
Citation: K. Thiam et al., Direct evidence of cytoplasmic delivery of PKC-alpha, -epsilon and -zeta pseudosubstrate lipopeptides: study of their implication in the induction ofapoptosis, FEBS LETTER, 459(3), 1999, pp. 285-290
Identification of inhibitors of an 80 kDa protease from Trypanosoma cruzi through the screening of a combinatorial peptide library
Authors: Vendeville, S Buisine, E Williard, X Schrevel, J Grellier, P Santana, J Sergheraert, C
Citation: S. Vendeville et al., Identification of inhibitors of an 80 kDa protease from Trypanosoma cruzi through the screening of a combinatorial peptide library, CHEM PHARM, 47(2), 1999, pp. 194-198
Synthesis of 5,5 '-dithiobis(2-nitrobenzamides) as alternative substrates for trypanothione reductase and thioredoxin reductase: A microtiter colorimetric assay for inhibitor screening
Authors: Davioud-Charvet, E Becker, K Landry, V Gromer, S Loge, C Sergheraert, C
Citation: E. Davioud-charvet et al., Synthesis of 5,5 '-dithiobis(2-nitrobenzamides) as alternative substrates for trypanothione reductase and thioredoxin reductase: A microtiter colorimetric assay for inhibitor screening, ANALYT BIOC, 268(1), 1999, pp. 1-8
Risultati: 1-23 |