Authors:
ZHANG MQ
STEINBUSCH HWM
KOOIJ PJ
TIMMERMAN H
Citation: Mq. Zhang et al., SYNTHESIS AND PRELIMINARY EVALUATION OF HYDROQUINONE-SUBSTITUTED HISTIDINE DERIVATIVES AS PUTATIVE HISTAMINERGIC NEUROTOXINS, European journal of medicinal chemistry, 29(7-8), 1994, pp. 503-511
Authors:
CHRISTIAANS JAM
WINDHORST AD
VANDERGOOT H
TIMMERMAN H
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF A SERIES OF HYBRID MOLECULES POSSESSING 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL BLOCKING ACTIVITY AND HISTAMINE H-2-AGONISTIC PROPERTIES, European journal of medicinal chemistry, 29(7-8), 1994, pp. 579-593
Citation: Zq. Yan et al., THE INVOLVEMENT OF NITRIC-OXIDE SYNTHASE IN THE EFFECT OF HISTAMINE ON GUINEA-PIG AIRWAY SMOOTH-MUSCLE IN-VITRO, Agents and actions, 41, 1994, pp. 30000111-30000112
Citation: Mq. Zhang et al., CHIRAL MANIPULATION OF DRUG SELECTIVITY - STUDIES ON A SERIES OF TERFENADINE-DERIVED DUAL ANTAGONISTS ON H-1-RECEPTORS AND CALCIUM CHANNELS, Agents and actions, 41, 1994, pp. 30000140-30000142
Authors:
VOLLINGA RC
DEKONING JP
JANSEN FP
LEURS R
MENGE WMPB
TIMMERMAN H
Citation: Rc. Vollinga et al., A NEW POTENT AND SELECTIVE HISTAMINE H-3 RECEPTOR AGONIST, 4-(1H-IMIDAZOL-4-YLMETHYL)PIPERIDINE, Journal of medicinal chemistry, 37(3), 1994, pp. 332-333
Authors:
YOKOYAMA H
ONODERA K
MAEYAMA K
SAKURAI E
IINUMA K
LEURS R
TIMMERMAN H
WATANABE T
Citation: H. Yokoyama et al., CLOBENPROPIT (VUF-9153), A NEW HISTAMINE H-3 RECEPTOR ANTAGONIST, INHIBITS ELECTRICALLY-INDUCED CONVULSIONS IN MICE, European journal of pharmacology, 260(1), 1994, pp. 23-28
Citation: Jk. Seydel et al., INFLUENCE OF MEMBRANE-COMPOSITION OF VARIOUS PARASITES ON THE INHIBITORY ACTIVITY OF A SERIES OF BIPYRIDYL ANALOGS, Chemotherapy, 40(2), 1994, pp. 124-135
Authors:
JANSEN FP
WU TS
VOSS HP
STEINBUSCH HWM
VOLLINGA RC
RADEMAKER B
BAST A
TIMMERMAN H
Citation: Fp. Jansen et al., CHARACTERIZATION OF THE BINDING OF THE FIRST SELECTIVE RADIOLABELED HISTAMINE H-3 RECEPTOR ANTAGONIST, [I-125] IODOPHENPROPIT, TO RAT-BRAIN, British Journal of Pharmacology, 113(2), 1994, pp. 355-362
Citation: R. Leurs et al., PHARMACOLOGICAL CHARACTERIZATION OF THE HUMAN HISTAMINE H-2-RECEPTOR STABLY EXPRESSED IN CHINESE-HAMSTER OVARY CELLS, British Journal of Pharmacology, 112(3), 1994, pp. 847-854
Authors:
LEURS R
SMIT MJ
TENSEN CP
TERLAAK AM
TIMMERMAN H
Citation: R. Leurs et al., SITE-DIRECTED MUTAGENESIS OF THE HISTAMINE H-1-RECEPTOR REVEALS A SELECTIVE INTERACTION OF ASPARAGINE(207) WITH SUBCLASSES OF H-1-RECEPTOR AGONISTS, Biochemical and biophysical research communications, 201(1), 1994, pp. 295-301
Citation: Mq. Zhang et H. Timmerman, TERFENADINE - A MIXTURE OF EQUIPOTENT ANTIHISTAMINE ENANTIOMERS WITHOUT A CLEAR ISOMERIC BALLAST, Pharmacy world & science, 15(5), 1993, pp. 186-192
Authors:
SMIT MJ
LEURS R
BLOEMERS SM
TERTOOLEN LGJ
BAST A
DELAAT SW
TIMMERMAN H
Citation: Mj. Smit et al., EXTRACELLULAR ATP ELEVATES CYTOPLASMATIC FREE CA2-CELLS BY THE INTERACTION WITH A 5'-NUCLEOTIDE RECEPTOR( IN HELA), European journal of pharmacology. Molecular pharmacology section, 247(2), 1993, pp. 223-226
Authors:
MANNHOLD R
CALDIROLA P
BIJLOO GJ
TIMMERMAN H
Citation: R. Mannhold et al., NEW CALMODULIN ANTAGONISTS OF THE DIPHENYLALKYLAMINE TYPE .1. BIOLOGICAL-ACTIVITY, SAR AND THE ROLE OF LIPOPHILICITY, European journal of medicinal chemistry, 28(9), 1993, pp. 727-734
Authors:
CALDIROLA P
ZANDBERG P
MANNHOLD R
TIMMERMAN H
Citation: P. Caldirola et al., NEW PRENYLAMINE-ANALOGS - INVESTIGATIONS OF THEIR INFLUENCE ON CALCIUM-DEPENDENT BIOLOGICAL-SYSTEMS, European journal of medicinal chemistry, 28(7-8), 1993, pp. 555-568
Citation: Mq. Zhang et al., STRUCTURE-ACTIVITY-RELATIONSHIPS WITHIN A SERIES OF ANALOGS OF THE HISTAMINE H-1-ANTAGONIST TERFENADINE, European journal of medicinal chemistry, 28(2), 1993, pp. 165-173
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF A SERIES OF NEW 1,4-DIHYDROPYRIDINES .2. DIETHYL ,6-DIMETHYL-1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLATES AND THEIR CORRESPONDING ISOTHIOUREAS AS TOOLS FOR DETERMINING STRUCTURE-ACTIVITY-RELATIONSHIPS, European journal of medicinal chemistry, 28(12), 1993, pp. 935-941
Authors:
CHRISTIAANS JAM
WINDHORST AD
GROENENBERG PM
VANDERGOOT H
TIMMERMAN H
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF NEW 1,4-DIHYDROPYRIDINES .1. -(OMEGA-AMINOALKYLTHIOMETHYL)-1,4-DIHYDROPYRIDINES AS POTENT CALCIUM-CHANNEL BLOCKERS, European journal of medicinal chemistry, 28(11), 1993, pp. 859-867
Authors:
CALDIROLA P
COATS E
MANNHOLD R
VANDERGOOT H
TIMMERMAN H
Citation: P. Caldirola et al., NEW CALMODULIN-ANTAGONISTS OF THE DIPHENYLALKYLAMINE TYPE .2. QSAR INVESTIGATIONS BY MEANS OF PARTIAL LEAST-SQUARE (PLS) ANALYSIS, European journal of medicinal chemistry, 28(10), 1993, pp. 783-790
Authors:
POLI E
POZZOLI C
CORUZZI G
BERTACCINI G
TIMMERMAN H
Citation: E. Poli et al., IN-VITRO CARDIAC PHARMACOLOGY OF THE NEW HISTAMINE H-2-RECEPTOR AGONIST AMTHAMINE - COMPARISONS WITH HISTAMINE AND DIMAPRIT, Agents and actions, 40(1-2), 1993, pp. 44-49
Authors:
KATHMANN M
SCHLICKER E
DETZNER M
TIMMERMAN H
Citation: M. Kathmann et al., NORDIMAPRIT, HOMODIMAPRIT, CLOBENPROPIT AND IMETIT - AFFINITIES FOR H-3 BINDING-SITES AND POTENCIES IN A FUNCTIONAL H-3 RECEPTOR MODEL, Naunyn-Schmiedeberg's archives of pharmacology, 348(5), 1993, pp. 498-503
Citation: Jc. Eriks et al., NEW ACTIVATION MODEL FOR THE HISTAMINE-H(2) RECEPTOR, EXPLAINING THE ACTIVITY OF THE DIFFERENT CLASSES OF HISTAMINE-H(2) RECEPTOR AGONISTS, Molecular pharmacology, 44(4), 1993, pp. 886-894