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Results: 76-97/97

Authors: ZHANG MQ STEINBUSCH HWM KOOIJ PJ TIMMERMAN H
Citation: Mq. Zhang et al., SYNTHESIS AND PRELIMINARY EVALUATION OF HYDROQUINONE-SUBSTITUTED HISTIDINE DERIVATIVES AS PUTATIVE HISTAMINERGIC NEUROTOXINS, European journal of medicinal chemistry, 29(7-8), 1994, pp. 503-511

Authors: CHRISTIAANS JAM WINDHORST AD VANDERGOOT H TIMMERMAN H
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF A SERIES OF HYBRID MOLECULES POSSESSING 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL BLOCKING ACTIVITY AND HISTAMINE H-2-AGONISTIC PROPERTIES, European journal of medicinal chemistry, 29(7-8), 1994, pp. 579-593

Authors: YAN ZQ KRAMER K BAST A TIMMERMAN H
Citation: Zq. Yan et al., THE INVOLVEMENT OF NITRIC-OXIDE SYNTHASE IN THE EFFECT OF HISTAMINE ON GUINEA-PIG AIRWAY SMOOTH-MUSCLE IN-VITRO, Agents and actions, 41, 1994, pp. 30000111-30000112

Authors: ZHANG MQ CALDIROLA P TIMMERMAN H
Citation: Mq. Zhang et al., CHIRAL MANIPULATION OF DRUG SELECTIVITY - STUDIES ON A SERIES OF TERFENADINE-DERIVED DUAL ANTAGONISTS ON H-1-RECEPTORS AND CALCIUM CHANNELS, Agents and actions, 41, 1994, pp. 30000140-30000142

Authors: VOLLINGA RC DEKONING JP JANSEN FP LEURS R MENGE WMPB TIMMERMAN H
Citation: Rc. Vollinga et al., A NEW POTENT AND SELECTIVE HISTAMINE H-3 RECEPTOR AGONIST, 4-(1H-IMIDAZOL-4-YLMETHYL)PIPERIDINE, Journal of medicinal chemistry, 37(3), 1994, pp. 332-333

Authors: YOKOYAMA H ONODERA K MAEYAMA K SAKURAI E IINUMA K LEURS R TIMMERMAN H WATANABE T
Citation: H. Yokoyama et al., CLOBENPROPIT (VUF-9153), A NEW HISTAMINE H-3 RECEPTOR ANTAGONIST, INHIBITS ELECTRICALLY-INDUCED CONVULSIONS IN MICE, European journal of pharmacology, 260(1), 1994, pp. 23-28

Authors: SEYDEL JK VANDERGOOT H TIMMERMAN H
Citation: Jk. Seydel et al., INFLUENCE OF MEMBRANE-COMPOSITION OF VARIOUS PARASITES ON THE INHIBITORY ACTIVITY OF A SERIES OF BIPYRIDYL ANALOGS, Chemotherapy, 40(2), 1994, pp. 124-135

Authors: JANSEN FP WU TS VOSS HP STEINBUSCH HWM VOLLINGA RC RADEMAKER B BAST A TIMMERMAN H
Citation: Fp. Jansen et al., CHARACTERIZATION OF THE BINDING OF THE FIRST SELECTIVE RADIOLABELED HISTAMINE H-3 RECEPTOR ANTAGONIST, [I-125] IODOPHENPROPIT, TO RAT-BRAIN, British Journal of Pharmacology, 113(2), 1994, pp. 355-362

Authors: LEURS R SMIT MJ MENGE WMBP TIMMERMAN H
Citation: R. Leurs et al., PHARMACOLOGICAL CHARACTERIZATION OF THE HUMAN HISTAMINE H-2-RECEPTOR STABLY EXPRESSED IN CHINESE-HAMSTER OVARY CELLS, British Journal of Pharmacology, 112(3), 1994, pp. 847-854

Authors: LEURS R SMIT MJ TENSEN CP TERLAAK AM TIMMERMAN H
Citation: R. Leurs et al., SITE-DIRECTED MUTAGENESIS OF THE HISTAMINE H-1-RECEPTOR REVEALS A SELECTIVE INTERACTION OF ASPARAGINE(207) WITH SUBCLASSES OF H-1-RECEPTOR AGONISTS, Biochemical and biophysical research communications, 201(1), 1994, pp. 295-301

Authors: TIMMERMAN H
Citation: H. Timmerman, PHARMACOTHERAPY OF VERTIGO - ANY NEWS TO BE EXPECTED, Acta oto-laryngologica, 1994, pp. 28-32

Authors: ZHANG MQ TIMMERMAN H
Citation: Mq. Zhang et H. Timmerman, TERFENADINE - A MIXTURE OF EQUIPOTENT ANTIHISTAMINE ENANTIOMERS WITHOUT A CLEAR ISOMERIC BALLAST, Pharmacy world & science, 15(5), 1993, pp. 186-192

Authors: SMIT MJ LEURS R BLOEMERS SM TERTOOLEN LGJ BAST A DELAAT SW TIMMERMAN H
Citation: Mj. Smit et al., EXTRACELLULAR ATP ELEVATES CYTOPLASMATIC FREE CA2-CELLS BY THE INTERACTION WITH A 5'-NUCLEOTIDE RECEPTOR( IN HELA), European journal of pharmacology. Molecular pharmacology section, 247(2), 1993, pp. 223-226

Authors: MANNHOLD R CALDIROLA P BIJLOO GJ TIMMERMAN H
Citation: R. Mannhold et al., NEW CALMODULIN ANTAGONISTS OF THE DIPHENYLALKYLAMINE TYPE .1. BIOLOGICAL-ACTIVITY, SAR AND THE ROLE OF LIPOPHILICITY, European journal of medicinal chemistry, 28(9), 1993, pp. 727-734

Authors: CALDIROLA P ZANDBERG P MANNHOLD R TIMMERMAN H
Citation: P. Caldirola et al., NEW PRENYLAMINE-ANALOGS - INVESTIGATIONS OF THEIR INFLUENCE ON CALCIUM-DEPENDENT BIOLOGICAL-SYSTEMS, European journal of medicinal chemistry, 28(7-8), 1993, pp. 555-568

Authors: ZHANG MQ TERLAAK AM TIMMERMAN H
Citation: Mq. Zhang et al., STRUCTURE-ACTIVITY-RELATIONSHIPS WITHIN A SERIES OF ANALOGS OF THE HISTAMINE H-1-ANTAGONIST TERFENADINE, European journal of medicinal chemistry, 28(2), 1993, pp. 165-173

Authors: CHRISTIAANS JAM VANDERGOOT H TIMMERMAN H
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF A SERIES OF NEW 1,4-DIHYDROPYRIDINES .2. DIETHYL ,6-DIMETHYL-1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLATES AND THEIR CORRESPONDING ISOTHIOUREAS AS TOOLS FOR DETERMINING STRUCTURE-ACTIVITY-RELATIONSHIPS, European journal of medicinal chemistry, 28(12), 1993, pp. 935-941

Authors: CHRISTIAANS JAM WINDHORST AD GROENENBERG PM VANDERGOOT H TIMMERMAN H
Citation: Jam. Christiaans et al., SYNTHESIS AND IN-VITRO PHARMACOLOGY OF NEW 1,4-DIHYDROPYRIDINES .1. -(OMEGA-AMINOALKYLTHIOMETHYL)-1,4-DIHYDROPYRIDINES AS POTENT CALCIUM-CHANNEL BLOCKERS, European journal of medicinal chemistry, 28(11), 1993, pp. 859-867

Authors: CALDIROLA P COATS E MANNHOLD R VANDERGOOT H TIMMERMAN H
Citation: P. Caldirola et al., NEW CALMODULIN-ANTAGONISTS OF THE DIPHENYLALKYLAMINE TYPE .2. QSAR INVESTIGATIONS BY MEANS OF PARTIAL LEAST-SQUARE (PLS) ANALYSIS, European journal of medicinal chemistry, 28(10), 1993, pp. 783-790

Authors: POLI E POZZOLI C CORUZZI G BERTACCINI G TIMMERMAN H
Citation: E. Poli et al., IN-VITRO CARDIAC PHARMACOLOGY OF THE NEW HISTAMINE H-2-RECEPTOR AGONIST AMTHAMINE - COMPARISONS WITH HISTAMINE AND DIMAPRIT, Agents and actions, 40(1-2), 1993, pp. 44-49

Authors: KATHMANN M SCHLICKER E DETZNER M TIMMERMAN H
Citation: M. Kathmann et al., NORDIMAPRIT, HOMODIMAPRIT, CLOBENPROPIT AND IMETIT - AFFINITIES FOR H-3 BINDING-SITES AND POTENCIES IN A FUNCTIONAL H-3 RECEPTOR MODEL, Naunyn-Schmiedeberg's archives of pharmacology, 348(5), 1993, pp. 498-503

Authors: ERIKS JC VANDERGOOT H TIMMERMAN H
Citation: Jc. Eriks et al., NEW ACTIVATION MODEL FOR THE HISTAMINE-H(2) RECEPTOR, EXPLAINING THE ACTIVITY OF THE DIFFERENT CLASSES OF HISTAMINE-H(2) RECEPTOR AGONISTS, Molecular pharmacology, 44(4), 1993, pp. 886-894
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