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Results: 1-8 |
Results: 8
Azepanone-based inhibitors of human and rat cathepsin K
Authors: Marquis, RW Ru, Y LoCastro, SM Zeng, J Yamashita, DS Oh, HJ Erhard, KF Davis, LD Tomaszek, TA Tew, D Salyers, K Proksch, J Ward, K Smith, B Levy, M Cummings, MD Haltiwanger, RC Trescher, G Wang, B Hemling, ME Quinn, CJ Cheng, HY Lin, F Smith, WW Janson, CA Zhao, BG McQueney, MS D'Alessio, K Lee, CP Marzulli, A Dodds, RA Blake, S Hwang, SM James, IE Gress, CJ Bradley, BR Lark, MW Gowen, M Veber, DF
Citation: Rw. Marquis et al., Azepanone-based inhibitors of human and rat cathepsin K, J MED CHEM, 44(9), 2001, pp. 1380-1395
Potent and selective cathepsin L inhibitors do not inhibit human osteoclast resorption in vitro
Authors: James, IE Marquis, RW Blake, SM Hwang, SM Gress, CJ Ru, Y Zembryki, D Yamashita, DS McQueney, MS Tomaszek, TA Oh, HJ Gowen, M Veber, DF Lark, MW
Citation: Ie. James et al., Potent and selective cathepsin L inhibitors do not inhibit human osteoclast resorption in vitro, J BIOL CHEM, 276(15), 2001, pp. 11507-11511
Solid-phase synthesis of a combinatorial array of 1,3-bis(acylamino)-2-butanones, inhibitors of the cysteine proteases cathepsins K and L
Authors: Yamashita, DS Dong, XY Oh, HJ Brook, CS Tomaszek, TA Szewczuk, L Tew, DG Veber, DF
Citation: Ds. Yamashita et al., Solid-phase synthesis of a combinatorial array of 1,3-bis(acylamino)-2-butanones, inhibitors of the cysteine proteases cathepsins K and L, J COMB CHEM, 1(3), 1999, pp. 207-215
Potent dipeptidylketone inhibitors of the cysteine protease cathepsin K
Authors: Marquis, RW Ru, Y Yamashita, DS Oh, HJ Yen, J Thompson, SK Carr, TJ Levy, MA Tomaszek, TA Ijames, CF Smith, WW Zhao, BG Janson, CA Abdel-Meguid, SS D'Alessio, KJ McQueney, MS Veber, DF
Citation: Rw. Marquis et al., Potent dipeptidylketone inhibitors of the cysteine protease cathepsin K, BIO MED CH, 7(4), 1999, pp. 581-588
Structure-based design of non-peptide, carbohydrazide-based cathepsin K inhibitors
Authors: Thompson, SK Halbert, SM DesJarlais, RL Tomaszek, TA Levy, MA Tew, DG Ijames, CF Veber, DF
Citation: Sk. Thompson et al., Structure-based design of non-peptide, carbohydrazide-based cathepsin K inhibitors, BIO MED CH, 7(4), 1999, pp. 599-605
Design and synthesis of diaminopyrrolidinone inhibitors of human osteoclast cathepsin K
Authors: Duffy, KJ Ridgers, LH DesJarlais, RL Tomaszek, TA Bossard, MJ Thompson, SK Keenan, RM Veber, DF
Citation: Kj. Duffy et al., Design and synthesis of diaminopyrrolidinone inhibitors of human osteoclast cathepsin K, BIOORG MED, 9(14), 1999, pp. 1907-1910
Development and characterization of a human in vitro resorption assay: Demonstration of utility using novel antiresorptive agents
Authors: James, IE Lark, MW Zembryki, D Lee-Rykaczewski, EV Hwang, SM Tomaszek, TA Belfiore, P Gowen, M
Citation: Ie. James et al., Development and characterization of a human in vitro resorption assay: Demonstration of utility using novel antiresorptive agents, J BONE MIN, 14(9), 1999, pp. 1562-1569
Mechanism of inhibition of cathepsin K by potent, selective 1,5-diacylcarbohydrazides: A new class of mechanism-based inhibitors of thiol proteases
Authors: Bossard, MJ Tomaszek, TA Levy, MA Ijames, CF Huddleston, MJ Briand, J Thompson, S Halpert, S Veber, DF Carr, SA Meek, TD Tew, DG
Citation: Mj. Bossard et al., Mechanism of inhibition of cathepsin K by potent, selective 1,5-diacylcarbohydrazides: A new class of mechanism-based inhibitors of thiol proteases, BIOCHEM, 38(48), 1999, pp. 15893-15902
Risultati: 1-8 |