Authors:
BONHAUS DW
WEINHARDT KK
TAYLOR M
DESOUZA A
MCNEELEY PM
SZCZEPANSKI K
FONTANA DJ
TRINH J
ROCHA CL
DAWSON MW
FLIPPIN LA
EGLEN RM
Citation: Dw. Bonhaus et al., RS-102221 - A NOVEL HIGH-AFFINITY AND SELECTIVE, 5-HT2C RECEPTOR ANTAGONIST, Neuropharmacology, 36(4-5), 1997, pp. 621-629
Citation: Kk. Weinhardt et al., SOME BENZENESULFONAMIDO-SUBSTITUTED VALEROPHENONES THAT ARE SELECTIVEANTAGONISTS FOR THE 5-HT2C RECEPTOR, Bioorganic & medicinal chemistry letters, 6(22), 1996, pp. 2687-2692
Authors:
CLARK RD
JAHANGIR A
LANGSTON JA
WEINHARDT KK
MILLER AB
LEUNG E
EGLEN RM
Citation: Rd. Clark et al., KETONES RELATED TO THE BENZOATE 5-HT4 RECEPTOR ANTAGONIST RS-23597 ARE HIGH-AFFINITY PARTIAL AGONISTS, Bioorganic & medicinal chemistry letters, 4(20), 1994, pp. 2477-2480
Authors:
CLARK RD
JAHANGIR A
LANGSTON JA
WEINHARDT KK
MILLER AB
LEUNG E
BONHAUS DW
WONG EHF
EGLEN RM
Citation: Rd. Clark et al., SYNTHESIS AND PRELIMINARY PHARMACOLOGICAL EVALUATION OF 2-BENZYLOXY SUBSTITUTED ARYL KETONES AS 5-HT4 RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(20), 1994, pp. 2481-2484
Authors:
CLARK RD
WEINHARDT KK
BERGER J
LEE CH
LEUNG E
WONG EHF
SMITH WL
EGLEN RM
Citation: Rd. Clark et al., N-(QUINUCLIDIN-3-YL)-1,8-NAPHTHALIMIDES WITH 5-HT(3) RECEPTOR ANTAGONIST AND 5-HT(4) RECEPTOR AGONIST PROPERTIES, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 1375-1378
Authors:
CLARK RD
MILLER AB
BERGER J
REPKE DB
WEINHARDT KK
KOWALCZYK BA
EGLEN RM
BONHAUS DW
LEE CH
MICHEL AD
SMITH WL
WONG EHF
Citation: Rd. Clark et al., 2-(QUINUCLIDIN-3-YL)PYRIDO[4,3-B]INDOL-1-ONES AND ISOQUINOLIN-1-ONES - POTENT CONFORMATIONALLY RESTRICTED 5-HT(3) RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(18), 1993, pp. 2645-2657