Authors:
LUENGO JI
YAMASHITA DS
DUNNINGTON D
BECK AK
ROZAMUS LW
YEN HK
BOSSARD MJ
LEVY MA
HAND A
NEWMANTARR T
BADGER A
FAUCETTE L
JOHNSON RK
DALESSIO K
PORTER T
SHU AYL
HEYS R
CHOI JW
KONGSAEREE P
CLARDY J
HOLT DA
Citation: Ji. Luengo et al., STRUCTURE-ACTIVITY STUDIES OF RAPAMYCIN ANALOGS - EVIDENCE THAT THE C-7 METHOXY GROUP IS PART OF THE EFFECTOR DOMAIN AND POSITIONED AT THE FKBP12-FRAP INTERFACE, Chemistry & biology, 2(7), 1995, pp. 471-481
Authors:
HOLT DA
KONIALIANBECK AL
OH HJ
YEN HK
ROZAMUS LW
KROG AJ
ERHARD KF
ORTIZ E
LEVY MA
BRANDT M
BOSSARD MJ
LUENGO JI
Citation: Da. Holt et al., STRUCTURE-ACTIVITY STUDIES OF SYNTHETIC FKBP LIGANDS AS PEPTIDYL-PROLYL ISOMERASE INHIBITORS, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 315-320
Authors:
YAMASHITA DS
OH HJ
YEN HK
BOSSARD MJ
BRANDT M
LEVY MA
NEWMANTARR T
BADGER A
LUENGO JI
HOLT DA
Citation: Ds. Yamashita et al., DESIGN, SYNTHESIS AND EVALUATION OF DUAL DOMAIN FKBP LIGANDS, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 325-328
Authors:
ABELL AD
ERHARD KF
YEN HK
YAMASHITA DS
BRANDT M
MOHAMMED H
LEVY MA
HOLT DA
Citation: Ad. Abell et al., PREPARATIVE CHIRAL HPLC SEPARATION OF ALL POSSIBLE STEREOISOMERS OF LY191704 AND LY266111 AND THEIR IN-VITRO INHIBITION OF HUMAN TYPE-1 ANDTYPE-2 STEROID 5-ALPHA-REDUCTASES, Bioorganic & medicinal chemistry letters, 4(11), 1994, pp. 1365-1368
Authors:
HOLT DA
OH HJ
ROZAMUS LW
YEN HK
BRANDT M
LEVY MA
METCALF BW
Citation: Da. Holt et al., SYNTHESIS AND EVALUATION OF 3-CARBOXYMETHYL STEROIDS AS INHIBITORS OFHUMAN PROSTATIC STEROID 5-ALPHA-REDUCTASE, Bioorganic & medicinal chemistry letters, 3(8), 1993, pp. 1735-1738
Authors:
HOLT DA
LUENGO JI
YAMASHITA DS
OH HJ
KONIALIAN AL
YEN HK
ROZAMUS LW
BRANDT M
BOSSARD MJ
LEVY MA
EGGLESTON DS
LIANG J
SCHULTZ LW
STOUT TJ
CLARDY J
Citation: Da. Holt et al., DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS AND THE X-RAY CRYSTAL-STRUCTURES OF THEIR COMPLEXES WITH FKBP12, Journal of the American Chemical Society, 115(22), 1993, pp. 9925-9938