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Results: 1-25 | 26-27
Results: 1-25/27
ISOXAZOLO-[3,4-D]-PYRIDAZIN-7-(6H)-ONES AND THEIR CORRESPONDING 4,5-DISUBSTITUTED-3-(2H)-PYRIDAZINONE ANALOGS AS NEW SUBSTRATES FOR ALPHA(1)-ADRENOCEPTOR SELECTIVE ANTAGONISTS - SYNTHESIS, MODELING, AND BINDING-STUDIES
Authors: MONTESANO F BARLOCCO D DALPIAZ V LEONARDI A POGGESI E FANELLI F DEBENEDETTI PG
Citation: F. Montesano et al., ISOXAZOLO-[3,4-D]-PYRIDAZIN-7-(6H)-ONES AND THEIR CORRESPONDING 4,5-DISUBSTITUTED-3-(2H)-PYRIDAZINONE ANALOGS AS NEW SUBSTRATES FOR ALPHA(1)-ADRENOCEPTOR SELECTIVE ANTAGONISTS - SYNTHESIS, MODELING, AND BINDING-STUDIES, Bioorganic & medicinal chemistry, 6(7), 1998, pp. 925-935
FREE-ENERGY PERTURBATION STUDIES ON BINDING OF THE INHIBITOR 5,6-DIHYDROBENZO[H]CINNOLIN-3(2H)ONE-2-ACETIC ACID AND ITS METHOXYLATED ANALOGS TO ALDOSE REDUCTASE
Authors: RASTELLI G COSTANTINO L VIANELLO P BARLOCCO D
Citation: G. Rastelli et al., FREE-ENERGY PERTURBATION STUDIES ON BINDING OF THE INHIBITOR 5,6-DIHYDROBENZO[H]CINNOLIN-3(2H)ONE-2-ACETIC ACID AND ITS METHOXYLATED ANALOGS TO ALDOSE REDUCTASE, Tetrahedron, 54(32), 1998, pp. 9415-9428
MONOSUBSTITUTED-3,8-DIAZABICYCLO[3.2.1]OCTANE AND DISUBSTITUTED-3,8-DIAZABICYCLO[3.2.1]OCTANE DERIVATIVES AS ANALGESICS STRUCTURALLY RELATED TO EPIBATIDINE - SYNTHESIS, ACTIVITY, AND MODELING
Authors: BARLOCCO D CIGNARELLA G TONDI D VIANELLO P VILLA S BARTOLINI A GHELARDINI C GALEOTTI N ANDERSON DJ KUNTZWEILER TA COLOMBO D TOMA L
Citation: D. Barlocco et al., MONOSUBSTITUTED-3,8-DIAZABICYCLO[3.2.1]OCTANE AND DISUBSTITUTED-3,8-DIAZABICYCLO[3.2.1]OCTANE DERIVATIVES AS ANALGESICS STRUCTURALLY RELATED TO EPIBATIDINE - SYNTHESIS, ACTIVITY, AND MODELING, Journal of medicinal chemistry, 41(5), 1998, pp. 674-681
PYRIDAZINONES AND THEIR TRICYCLIC CONGENERS - CHEMISTRY AND BIOLOGY
Authors: CIGNARELLA G BARLOCCO D VILLA S CURZU MM PINNA GA
Citation: G. Cignarella et al., PYRIDAZINONES AND THEIR TRICYCLIC CONGENERS - CHEMISTRY AND BIOLOGY, Journal of heterocyclic chemistry, 35(5), 1998, pp. 1161-1170
DEVELOPMENT OF PHARMACOPHORES FOR INHIBITORS OF THE RAPID COMPONENT OF THE CARDIAC DELAYED RECTIFIER POTASSIUM CURRENT
Authors: MATYUS P BOROSY AP VARRO A PAPP JG BARLOCCO D CIGNARELLA G
Citation: P. Matyus et al., DEVELOPMENT OF PHARMACOPHORES FOR INHIBITORS OF THE RAPID COMPONENT OF THE CARDIAC DELAYED RECTIFIER POTASSIUM CURRENT, International journal of quantum chemistry, 69(1), 1998, pp. 21-30
NEW ALDOSE REDUCTASE INHIBITORS AS POTENTIAL AGENTS FOR THE PREVENTION OF LONG-TERM DIABETIC COMPLICATIONS
Authors: COSTANTINO L RASTELLI G CIGNARELLA G VIANELLO P BARLOCCO D
Citation: L. Costantino et al., NEW ALDOSE REDUCTASE INHIBITORS AS POTENTIAL AGENTS FOR THE PREVENTION OF LONG-TERM DIABETIC COMPLICATIONS, Expert opinion on therapeutic patents, 7(8), 1997, pp. 843-858
STUDY OF THE ANTISECRETORY AND ANTIULCER MECHANISMS OF A NEW INDENOPIRYDAZINONE DERIVATIVE IN RATS
Authors: BAROCELLI E CHIAVARINI M BALLABENI V BARLOCCO D VIANELLO P DALPIAZ V IMPICCIATORE M
Citation: E. Barocelli et al., STUDY OF THE ANTISECRETORY AND ANTIULCER MECHANISMS OF A NEW INDENOPIRYDAZINONE DERIVATIVE IN RATS, Pharmacological research, 35(5), 1997, pp. 487-492
STRUCTURE-BASED DESIGN OF AN INHIBITOR MODELED AT THE SUBSTRATE ACTIVE-SITE OF ALDOSE REDUCTASE
Authors: RASTELLI G VIANELLO P BARLOCCO D COSTANTINO L DELCORSO A MURA U
Citation: G. Rastelli et al., STRUCTURE-BASED DESIGN OF AN INHIBITOR MODELED AT THE SUBSTRATE ACTIVE-SITE OF ALDOSE REDUCTASE, Bioorganic & medicinal chemistry letters, 7(14), 1997, pp. 1897-1902
ANTINOCICEPTIVE PROFILE OF THE NEW NICOTINIC AGONIST DBO-83
Authors: GHELARDINI C GALEOTTI N BARLOCCO D BARTOLINI A
Citation: C. Ghelardini et al., ANTINOCICEPTIVE PROFILE OF THE NEW NICOTINIC AGONIST DBO-83, Drug development research, 40(3), 1997, pp. 251-258
2,2,6-TRIMETHYLPIPERAZINE AND 2,3,5-TRIMETHYLPIPERAZINE AS MONOCYCLICANALOGS OF THE MU-OPIOID AGONIST 3,8-DIAZABICYCLO[3.2.1]OCTANES - SYNTHESIS, MODELING, AND ACTIVITY
Authors: BALLABIO M BARLOCCO D CIGNARELLA G COLOMBO D TOMA L
Citation: M. Ballabio et al., 2,2,6-TRIMETHYLPIPERAZINE AND 2,3,5-TRIMETHYLPIPERAZINE AS MONOCYCLICANALOGS OF THE MU-OPIOID AGONIST 3,8-DIAZABICYCLO[3.2.1]OCTANES - SYNTHESIS, MODELING, AND ACTIVITY, Tetrahedron, 53(4), 1997, pp. 1481-1490
ANTINOCICEPTIVE ACTION OF DBO-17 AND DBO-11 IN MICE - 2 3,8-DIAZABICYCLO(3.2.1.)OCTANE DERIVATES WITH SELECTIVE MU-OPIOID RECEPTOR AFFINITY
Authors: FADDA P BARLOCCO D TRONCI S CIGNARELLA G FRATTA W
Citation: P. Fadda et al., ANTINOCICEPTIVE ACTION OF DBO-17 AND DBO-11 IN MICE - 2 3,8-DIAZABICYCLO(3.2.1.)OCTANE DERIVATES WITH SELECTIVE MU-OPIOID RECEPTOR AFFINITY, Naunyn-Schmiedeberg's archives of pharmacology, 356(5), 1997, pp. 596-602
NAPHTHALIMIDO DERIVATIVES AS ANTIFOLATE THYMIDYLATE SYNTHASE INHIBITORS
Authors: COSTI MP TONDI D RINALDI M BARLOCCO D CIGNARELLA G SANTI DV MUSIU C PUDU I VACCA G LACOLLA P
Citation: Mp. Costi et al., NAPHTHALIMIDO DERIVATIVES AS ANTIFOLATE THYMIDYLATE SYNTHASE INHIBITORS, European journal of medicinal chemistry, 31(12), 1996, pp. 1011-1016
4,5-FUNCTIONALIZED 6-PHENYL-3(2H)-PYRIDAZINONES - SYNTHESIS AND EVALUATION OF ANTINOCICEPTIVE ACTIVITY
Authors: DALPIAZ V GIOVANNONI MP CICIANI G BARLOCCO D GIARDINA G PETRONE G CLARKE GD
Citation: V. Dalpiaz et al., 4,5-FUNCTIONALIZED 6-PHENYL-3(2H)-PYRIDAZINONES - SYNTHESIS AND EVALUATION OF ANTINOCICEPTIVE ACTIVITY, European journal of medicinal chemistry, 31(1), 1996, pp. 65-70
TRICYCLIC INDENOPYRIDAZINE DERIVATIVES - SYNTHESIS, CYTOTOXIC ACTIVITY AND DNA-BINDING PROPERTIES
Authors: BARLOCCO D BERGOMI M MENTA E PALUMBO M CIGNARELLA G
Citation: D. Barlocco et al., TRICYCLIC INDENOPYRIDAZINE DERIVATIVES - SYNTHESIS, CYTOTOXIC ACTIVITY AND DNA-BINDING PROPERTIES, Recueil des travaux chimiques des Pays-Bas, 115(1), 1996, pp. 25
SYNTHESIS, ACTIVITY, AND MOLECULAR MODELING OF A NEW SERIES OF TRICYCLIC PYRIDAZINONES AS SELECTIVE ALDOSE REDUCTASE INHIBITORS
Authors: COSTANTINO L RASTELLI G VESCOVINI K CIGNARELLA G VIANELLO P DELCORSO A CAPPIELLO M MURA U BARLOCCO D
Citation: L. Costantino et al., SYNTHESIS, ACTIVITY, AND MOLECULAR MODELING OF A NEW SERIES OF TRICYCLIC PYRIDAZINONES AS SELECTIVE ALDOSE REDUCTASE INHIBITORS, Journal of medicinal chemistry, 39(22), 1996, pp. 4396-4405
SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF A NEW SERIES OF SUBSTITUTED BENZOYL-GAMMA-BUTYROLACTONE DERIVATIVES
Authors: CIGNARELLA G BARLOCCO D POCAR D CLERICI F CURZU MM GESSA GL FADDA F SERRA M BIGGIO G
Citation: G. Cignarella et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF A NEW SERIES OF SUBSTITUTED BENZOYL-GAMMA-BUTYROLACTONE DERIVATIVES, European journal of medicinal chemistry, 30(9), 1995, pp. 721-726
MONOCYCLIC ANALOGS OF THE MU-OPIOID AGONIST 3,8-DIAZABICYCLO-[3.2.1]OCTANES - SYNTHESIS, MODELING, AND ACTIVITY
Authors: BARLOCCO D VILLA S FRATTA W FADDA P COLOMBO D TOMA L
Citation: D. Barlocco et al., MONOCYCLIC ANALOGS OF THE MU-OPIOID AGONIST 3,8-DIAZABICYCLO-[3.2.1]OCTANES - SYNTHESIS, MODELING, AND ACTIVITY, Tetrahedron, 51(42), 1995, pp. 11547-11556
UNEXPECTED BEHAVIOR OF THE OXIDIZING-AGENT SODIUM M-NITROBENZENESULFONATE - SYNTHESIS OF A NEW CLASS OF -HYDROXY[1]BENZOPYRANO-[4-3-C]PYRIDAZIN-3(2H)-ONES
Authors: CIGNARELLA G BARLOCCO D
Citation: G. Cignarella et D. Barlocco, UNEXPECTED BEHAVIOR OF THE OXIDIZING-AGENT SODIUM M-NITROBENZENESULFONATE - SYNTHESIS OF A NEW CLASS OF -HYDROXY[1]BENZOPYRANO-[4-3-C]PYRIDAZIN-3(2H)-ONES, Journal of heterocyclic chemistry, 32(1), 1995, pp. 79-80
SYNTHESIS OF 1,4-DISUBSTITUTED-2-METHYLPIPERAZINES AND STUDY OF THEIRANALGESIC PROPERTIES
Authors: BARLOCCO D BRUNELLO N BERNARDI M CIGNARELLA G
Citation: D. Barlocco et al., SYNTHESIS OF 1,4-DISUBSTITUTED-2-METHYLPIPERAZINES AND STUDY OF THEIRANALGESIC PROPERTIES, Il Farmaco, 50(2), 1995, pp. 119-124
SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF THIENOCINNOLIN-3-(2H)-ONES, BIOISOSTERS OF ANTIHYPERTENSIVE AND ANTITHROMBOTIC BENZO(H)CINNOLINONES
Authors: PINNA GA CURZU MM CIGNARELLA G BARLOCCO D DAMICO M FILIPPELLI A DENOVELLIS V ROSSI F
Citation: Ga. Pinna et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF THIENOCINNOLIN-3-(2H)-ONES, BIOISOSTERS OF ANTIHYPERTENSIVE AND ANTITHROMBOTIC BENZO(H)CINNOLINONES, European journal of medicinal chemistry, 29(6), 1994, pp. 447-454
SYNTHESIS OF A NEW SERIES OF 2,7-DIAZASPIRO[3.5]NONAN-1-ONES AND STUDY OF THEIR CHOLINERGIC PROPERTIES
Authors: CIGNARELLA G VILLA S BARLOCCO D
Citation: G. Cignarella et al., SYNTHESIS OF A NEW SERIES OF 2,7-DIAZASPIRO[3.5]NONAN-1-ONES AND STUDY OF THEIR CHOLINERGIC PROPERTIES, European journal of medicinal chemistry, 29(2), 1994, pp. 115-120
SYNTHESIS OF A NEW SERIES OF 2,8-DISUBSTITUTED-2,8-DIAZASPIRO[4,5]DECAN-1-ONES AS POTENTIAL MUSCARINIC AGONISTS
Authors: CIGNARELLA G VILLA S CATTABENI F RENO F CIMINO M DEBENEDETTI PG BARLOCCO D
Citation: G. Cignarella et al., SYNTHESIS OF A NEW SERIES OF 2,8-DISUBSTITUTED-2,8-DIAZASPIRO[4,5]DECAN-1-ONES AS POTENTIAL MUSCARINIC AGONISTS, European journal of medicinal chemistry, 29(12), 1994, pp. 955-961
COMPUTER-AIDED STRUCTURE AFFINITY RELATIONSHIPS IN A SET OF PIPERAZINE AND 3,8-DIAZABICYCLO[3.2.1]OCTANE DERIVATIVES BINDING TO THE MU-OPIOID RECEPTOR
Authors: BARLOCCO D CIGNARELLA G GRECO G NOVELLINO E
Citation: D. Barlocco et al., COMPUTER-AIDED STRUCTURE AFFINITY RELATIONSHIPS IN A SET OF PIPERAZINE AND 3,8-DIAZABICYCLO[3.2.1]OCTANE DERIVATIVES BINDING TO THE MU-OPIOID RECEPTOR, Journal of computer-aided molecular design, 7(5), 1993, pp. 557-571
SYNTHESIS OF A NEW SERIES OF N-SUBSTITUTED-3-[L-ALKYL(ARYL)- 4-PIPERIDYL]AZETIDIN-2-ONES AS POSSIBLE MUSCARINIC AGENTS
Authors: CIGNARELLA G VILLA S BARLOCCO D
Citation: G. Cignarella et al., SYNTHESIS OF A NEW SERIES OF N-SUBSTITUTED-3-[L-ALKYL(ARYL)- 4-PIPERIDYL]AZETIDIN-2-ONES AS POSSIBLE MUSCARINIC AGENTS, Journal of heterocyclic chemistry, 30(5), 1993, pp. 1337-1340
SYNTHESIS OF A NEW SERIES OF 8-SUBSTITUTED-2,8-DIAZASPIRO[4.5]DECAN-3-ONES
Authors: CIGNARELLA G VILLA S BARLOCCO D
Citation: G. Cignarella et al., SYNTHESIS OF A NEW SERIES OF 8-SUBSTITUTED-2,8-DIAZASPIRO[4.5]DECAN-3-ONES, Journal of heterocyclic chemistry, 30(5), 1993, pp. 1357-1359
Risultati: 1-25 | 26-27