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Results: 1-25 | 26-30
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Lipophilicity behaviour of the zwitterionic antihistamine cetirizine in phosphatidylcholine liposomes/water systems
Authors: van Balen, GP Caron, G Ermondi, G Pagliara, A Grandi, T Bouchard, G Fruttero, R Carrupt, PA Testa, B
Citation: Gp. Van Balen et al., Lipophilicity behaviour of the zwitterionic antihistamine cetirizine in phosphatidylcholine liposomes/water systems, PHARM RES, 18(5), 2001, pp. 694-701
The apparent lipophilicity of quaternary ammonium ions is influenced by Galvani potential difference, not ion-pairing: A cyclic voltammetry study
Authors: Bouchard, G Carrupt, PA Testa, B Gobry, V Girault, HH
Citation: G. Bouchard et al., The apparent lipophilicity of quaternary ammonium ions is influenced by Galvani potential difference, not ion-pairing: A cyclic voltammetry study, PHARM RES, 18(5), 2001, pp. 702-708
The esterase-like activity of serum albumin may be due to cholinesterase contamination
Authors: Chapuis, N Bruhlmann, C Reist, M Carrupt, PA Mayer, JM Testa, B
Citation: N. Chapuis et al., The esterase-like activity of serum albumin may be due to cholinesterase contamination, PHARM RES, 18(10), 2001, pp. 1435-1439
Interaction of psychotropic drugs with monoamine oxidase in rat brain
Authors: Gnerre, C Kosel, M Baumann, P Carrupt, PA Testa, B
Citation: C. Gnerre et al., Interaction of psychotropic drugs with monoamine oxidase in rat brain, J PHARM PHA, 53(8), 2001, pp. 1125-1130
Coumarins derivatives as dual inhibitors of acetylcholinesterase and monoamine oxidase
Authors: Bruhlmann, C Ooms, F Carrupt, PA Testa, B Catto, M Leonetti, F Altomare, C Carotti, A
Citation: C. Bruhlmann et al., Coumarins derivatives as dual inhibitors of acetylcholinesterase and monoamine oxidase, J MED CHEM, 44(19), 2001, pp. 3195-3198
Novel basic isoflavones as inhibitors of bone resorption
Authors: Delcanale, M Amari, G Armani, E Lipreri, M Civelli, M Galbiati, E Giossi, M Caruso, PL Crivori, P Carrupt, PA Testa, B
Citation: M. Delcanale et al., Novel basic isoflavones as inhibitors of bone resorption, HELV CHIM A, 84(8), 2001, pp. 2417-2429
Natural and synthetic xanthones as monoamine oxidase inhibitors: Biological assay and 3D-QSAR
Authors: Gnerre, C Thull, U Gaillard, P Carrupt, PA Testa, B Fernandes, E Silva, F Pinto, M Pinto, MMM Wolfender, JL Hostettmann, K Cruciani, G
Citation: C. Gnerre et al., Natural and synthetic xanthones as monoamine oxidase inhibitors: Biological assay and 3D-QSAR, HELV CHIM A, 84(3), 2001, pp. 552-570
Molecular-dynamics and NMR investigation of the property space of the zwitterionic antihistamine cetirizine
Authors: Ermondi, G Caron, G Bouchard, G van Balen, GP Pagliara, A Grandi, T Carrupt, PA Fruttero, R Testa, B
Citation: G. Ermondi et al., Molecular-dynamics and NMR investigation of the property space of the zwitterionic antihistamine cetirizine, HELV CHIM A, 84(2), 2001, pp. 360-374
Ionic partition diagram of the zwitterionic antihistamine cetirizine
Authors: Bouchard, G Pagliara, A van Balen, GP Carrupt, PA Testa, B Gobry, V Girault, HH Caron, G Ermondi, G
Citation: G. Bouchard et al., Ionic partition diagram of the zwitterionic antihistamine cetirizine, HELV CHIM A, 84(2), 2001, pp. 375-387
Structural damage to proteins caused by free radicals: asessment, protection by antioxidants, and influence of protein binding
Authors: Salvi, A Carrupt, PA Tillement, JP Testa, B
Citation: A. Salvi et al., Structural damage to proteins caused by free radicals: asessment, protection by antioxidants, and influence of protein binding, BIOCH PHARM, 61(10), 2001, pp. 1237-1242
Generalization of ionic partition diagrams to lipophilic compounds and to biphasic systems with variable phase volume ratios
Authors: Gobry, V Ulmeanu, S Reymond, F Bouchard, G Carrupt, PA Testa, B Girault, HH
Citation: V. Gobry et al., Generalization of ionic partition diagrams to lipophilic compounds and to biphasic systems with variable phase volume ratios, J AM CHEM S, 123(43), 2001, pp. 10684-10690
The influence of lipophilicity on the pharmacokinetic behavior of drugs: Concepts and examples
Authors: Testa, B Crivori, P Reist, M Carrupt, PA
Citation: B. Testa et al., The influence of lipophilicity on the pharmacokinetic behavior of drugs: Concepts and examples, PERSP DR D, 19(1), 2000, pp. 179-211
Molecular fields in quantitative structure-permeation relationships: the VolSurf approach
Authors: Cruciani, C Crivori, P Carrupt, PA Testa, B
Citation: C. Cruciani et al., Molecular fields in quantitative structure-permeation relationships: the VolSurf approach, J MOL ST-TH, 503(1-2), 2000, pp. 17-30
Very slow chiral inversion of clopidogrel in rats: A pharmacokinetic and mechanistic investigation
Authors: Reist, M Roy-De Vos, M Montseny, JP Mayer, JM Carrupt, PA Berger, Y Testa, B
Citation: M. Reist et al., Very slow chiral inversion of clopidogrel in rats: A pharmacokinetic and mechanistic investigation, DRUG META D, 28(12), 2000, pp. 1405-1410
Inhibition of monoamine oxidases by functionalized coumarin derivatives: Biological activities, QSARs, and 3D-QSARs
Authors: Gnerre, C Catto, M Leonetti, F Weber, P Carrupt, PA Altomare, C Carotti, A Testa, B
Citation: C. Gnerre et al., Inhibition of monoamine oxidases by functionalized coumarin derivatives: Biological activities, QSARs, and 3D-QSARs, J MED CHEM, 43(25), 2000, pp. 4747-4758
Predicting blood-brain barrier permeation from three-dimensional molecularstructure
Authors: Crivori, P Cruciani, G Carrupt, PA Testa, B
Citation: P. Crivori et al., Predicting blood-brain barrier permeation from three-dimensional molecularstructure, J MED CHEM, 43(11), 2000, pp. 2204-2216
Physicochemical characterization of sildenafil: Ionization, lipophilicity behavior, and ionic-partition diagram sturdied by two-phase titration and electrochemistry
Authors: Gobry, V Bouchard, G Carrupt, PA Testa, B Girault, HH
Citation: V. Gobry et al., Physicochemical characterization of sildenafil: Ionization, lipophilicity behavior, and ionic-partition diagram sturdied by two-phase titration and electrochemistry, HELV CHIM A, 83(7), 2000, pp. 1465-1474
Lipophilicity and related molecular properties as determinants of pharmacokinetic behaviour
Authors: Testa, B Caron, G Crivori, P Rey, S Reist, M Carrupt, PA
Citation: B. Testa et al., Lipophilicity and related molecular properties as determinants of pharmacokinetic behaviour, CHIMIA, 54(11), 2000, pp. 672-677
Ionic partition diagrams of ionisable drugs: pH-lipophilicity profiles, transfer mechanisms and charge effects on solvation
Authors: Reymond, F Chopineaux-Courtois, V Steyaert, G Bouchard, G Carrupt, PA Testa, B Girault, HH
Citation: F. Reymond et al., Ionic partition diagrams of ionisable drugs: pH-lipophilicity profiles, transfer mechanisms and charge effects on solvation, J ELEC CHEM, 462(2), 1999, pp. 235-250
Combined molecular lipophilicity descriptors and their role in understanding intramolecular effects
Authors: Caron, G Reymond, F Carrupt, PA Girault, HH Testa, B
Citation: G. Caron et al., Combined molecular lipophilicity descriptors and their role in understanding intramolecular effects, PHARM SCI T, 2(8), 1999, pp. 327-335
Charge and delocalisation effects on the lipophilicity of protonable drugs
Authors: Reymond, F Carrupt, PA Testa, B Girault, HH
Citation: F. Reymond et al., Charge and delocalisation effects on the lipophilicity of protonable drugs, CHEM-EUR J, 5(1), 1999, pp. 39-47
The pH-partition profile of the anti-ischemic drug trimetazidine may explain its reduction of intracellular acidosis
Authors: Reymond, F Steyaert, G Carrupt, PA Morin, D Tillement, JP Girault, HH Testa, B
Citation: F. Reymond et al., The pH-partition profile of the anti-ischemic drug trimetazidine may explain its reduction of intracellular acidosis, PHARM RES, 16(5), 1999, pp. 616-624
Production and characterization of 22 monoclonal antibodies directed against S 20499, a new potent 5-HT1A chiral agonist: Influence of the hapten structure on specificity and stereorecognition
Authors: Got, P Raimbaud, E Bussey, C Caron, G Carrupt, PA Walther, B Bensussan, A Scherrmann, JM
Citation: P. Got et al., Production and characterization of 22 monoclonal antibodies directed against S 20499, a new potent 5-HT1A chiral agonist: Influence of the hapten structure on specificity and stereorecognition, PHARM RES, 16(5), 1999, pp. 725-735
Evaluation and prediction of drug permeation
Authors: Pagliara, A Reist, M Geinoz, S Carrupt, PA Testa, B
Citation: A. Pagliara et al., Evaluation and prediction of drug permeation, J PHARM PHA, 51(12), 1999, pp. 1339-1357
Structure-lipophilicity relationships of neutral and protonated beta-blockers Part I Intra- and intermolecular effects in isotropic solvent systems
Authors: Caron, G Steyaert, G Pagliara, A Reymond, F Crivori, P Gaillard, P Carrupt, PA Avdeef, A Comer, J Box, KJ Girault, HH Testa, B
Citation: G. Caron et al., Structure-lipophilicity relationships of neutral and protonated beta-blockers Part I Intra- and intermolecular effects in isotropic solvent systems, HELV CHIM A, 82(8), 1999, pp. 1211-1222
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