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Results: 1-24 |
Results: 24
Conformation of the tripeptide Cbz-Pro-Leu-Trp-OBzl(CF3)(2) deduced from two-dimensional H-1-NMR and conformational energy calculations is related toits affinity for NK1-receptor
Authors: Millet, R Goossens, L Goossens, JF Chavatte, P Bertrand-Caumont, K Houssin, R Henichart, JP
Citation: R. Millet et al., Conformation of the tripeptide Cbz-Pro-Leu-Trp-OBzl(CF3)(2) deduced from two-dimensional H-1-NMR and conformational energy calculations is related toits affinity for NK1-receptor, J PEPT SCI, 7(6), 2001, pp. 323-330
New bis-catechols 5-lipoxygenase inhibitors
Authors: Dupont, R Goossens, JF Cotelle, N Vrielynck, L Vezin, H Henichart, JP Cotelle, P
Citation: R. Dupont et al., New bis-catechols 5-lipoxygenase inhibitors, BIO MED CH, 9(2), 2001, pp. 229-235
N-Aminoindoline derivatives as inhibitors of 5-lipoxygenase
Authors: Audouin, C Mestdagh, N Lassoie, MA Houssin, R Henichart, JP
Citation: C. Audouin et al., N-Aminoindoline derivatives as inhibitors of 5-lipoxygenase, BIOORG MED, 11(6), 2001, pp. 845-848
Pyrazolidine-3,5-dione angiotensin-II receptor antagonists
Authors: Cauvin, C Le Bourdonnec, B Norberg, B Henichart, JP Durant, F
Citation: C. Cauvin et al., Pyrazolidine-3,5-dione angiotensin-II receptor antagonists, ACT CRYST C, 57, 2001, pp. 1330-1332
A flexible approach to the design of new potent substance P receptor ligands
Authors: Millet, R Goossens, L Bertrand-Caumont, K Goossens, JF Houssin, R Henichart, JP
Citation: R. Millet et al., A flexible approach to the design of new potent substance P receptor ligands, J PHARM PHA, 53(7), 2001, pp. 929-934
Conformational analysis of tripeptide Ac-Lys-Pro-Val-NH2, COOH-terminal sequence of alpha-MSH
Authors: Chavatte, P Yous, S Lesieur, D Henichart, JP
Citation: P. Chavatte et al., Conformational analysis of tripeptide Ac-Lys-Pro-Val-NH2, COOH-terminal sequence of alpha-MSH, J PHARM PHA, 53(7), 2001, pp. 949-953
A synthesis of new Pyrrolo[3,2-c]quinolines
Authors: Dudouit, F Houssin, R Henichart, JP
Citation: F. Dudouit et al., A synthesis of new Pyrrolo[3,2-c]quinolines, J HETERO CH, 38(3), 2001, pp. 755-758
DNA interaction of the tyrosine protein kinase inhibitor PD153035 and its N-methyl analogue
Authors: Goossens, JF Bouey-Bencteux, E Houssin, R Henichart, JP Colson, P Houssier, C Laine, W Baldeyrou, B Bailly, C
Citation: Jf. Goossens et al., DNA interaction of the tyrosine protein kinase inhibitor PD153035 and its N-methyl analogue, BIOCHEM, 40(15), 2001, pp. 4663-4671
Synthesis, DNA binding, topoisomerases inhibition and cytotoxic propertiesof 4-arylcarboxamidopyrrolo-2-carboxyanilides
Authors: Dudouit, F Goossens, JF Houssin, R Henichart, JP Colson, P Houssier, C Gelus, N Bailly, C
Citation: F. Dudouit et al., Synthesis, DNA binding, topoisomerases inhibition and cytotoxic propertiesof 4-arylcarboxamidopyrrolo-2-carboxyanilides, BIOORG MED, 10(6), 2000, pp. 553-557
Relation between intracellular acidification and camptothecin-induced apoptosis in leukemia cells
Authors: Goossens, JF Henichart, JP Dassonneville, L Facompre, M Bailly, C
Citation: Jf. Goossens et al., Relation between intracellular acidification and camptothecin-induced apoptosis in leukemia cells, EUR J PH SC, 10(2), 2000, pp. 125-131
Synthesis and pharmacological evaluation of new pyrazolidine-3,5-diones asAT(1) angiotensin II receptor antagonists
Authors: Le Bourdonnec, B Meulon, E Yous, S Goossens, JF Houssin, R Henichart, JP
Citation: B. Le Bourdonnec et al., Synthesis and pharmacological evaluation of new pyrazolidine-3,5-diones asAT(1) angiotensin II receptor antagonists, J MED CHEM, 43(14), 2000, pp. 2685-2697
Conformationally constrained dipeptides. Obtention of enantiomerically pure 6-acetamido-5-oxo-1,2,3,5,6,7-hexahydro-3-indolizine carboxylic acid
Authors: Millet, R Meulon, E Goossens, L Houssin, R Henichart, JP Rigo, B
Citation: R. Millet et al., Conformationally constrained dipeptides. Obtention of enantiomerically pure 6-acetamido-5-oxo-1,2,3,5,6,7-hexahydro-3-indolizine carboxylic acid, J HETERO CH, 37(6), 2000, pp. 1491-1494
A new synthesis of N-alkyl pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones
Authors: Le Bourdonnec, B Meulon, E Yous, S Houssin, R Henichart, JP
Citation: B. Le Bourdonnec et al., A new synthesis of N-alkyl pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones, J HETERO CH, 37(5), 2000, pp. 1209-1212
Studies on pyrrolidinones. Synthesis and cyclization of N-[alpha-naphthyl-(3,4,5-trimethoxyphenyl)-methyl]pyroglutamic acid
Authors: Legrand, A Rigo, B Henichart, JP Norberg, B Camus, F Durant, F Couturier, D
Citation: A. Legrand et al., Studies on pyrrolidinones. Synthesis and cyclization of N-[alpha-naphthyl-(3,4,5-trimethoxyphenyl)-methyl]pyroglutamic acid, J HETERO CH, 37(2), 2000, pp. 215-227
Studies on pyrrolidinones. Preparation of 1,5,6-10b-tetrahydro-2H-pyrrolo[1,2-c]quinazoline-3-ones from pyroglutamic acid
Authors: El Ghammarti, S Rigo, B Mejdi, H Henichart, JP Couturier, D
Citation: S. El Ghammarti et al., Studies on pyrrolidinones. Preparation of 1,5,6-10b-tetrahydro-2H-pyrrolo[1,2-c]quinazoline-3-ones from pyroglutamic acid, J HETERO CH, 37(1), 2000, pp. 143-150
Cellular uptake and interaction with purified membranes of rebeccamycin derivatives
Authors: Goossens, JF Henichart, JP Anizon, F Prudhomme, M Dugave, C Riou, JF Bailly, C
Citation: Jf. Goossens et al., Cellular uptake and interaction with purified membranes of rebeccamycin derivatives, EUR J PHARM, 389(2-3), 2000, pp. 141-146
Phosphodiesterase 4 inhibitors as airways smooth muscle relaxant agents: Synthesis and biological activities of triazine derivatives
Authors: Leroux, F van Keulen, BJ Daliers, J Pommery, N Henichart, JP
Citation: F. Leroux et al., Phosphodiesterase 4 inhibitors as airways smooth muscle relaxant agents: Synthesis and biological activities of triazine derivatives, BIO MED CH, 7(3), 1999, pp. 509-516
Synthesis and cytotoxicity of analogues of the antibiotic BE 10988 inhibitors of DNA topoisomerase II
Authors: Catrycke, MO Houssin, R Henichart, JP Pfeiffer, B Renard, P Dassonneville, L Bailly, C
Citation: Mo. Catrycke et al., Synthesis and cytotoxicity of analogues of the antibiotic BE 10988 inhibitors of DNA topoisomerase II, BIOORG MED, 9(14), 1999, pp. 2025-2030
Synthesis, mode of action, and biological activities of rebeccamycin bromoderivatives
Authors: Moreau, P Anizon, F Sancelme, M Prudhomme, M Severe, D Riou, JF Goossens, JF Henichart, JP Bailly, C Labourier, E Tazzi, J Fabbro, D Meyer, T Aubertin, AM
Citation: P. Moreau et al., Synthesis, mode of action, and biological activities of rebeccamycin bromoderivatives, J MED CHEM, 42(10), 1999, pp. 1816-1822
Studies on pyrrolidinone. Synthesis of aza analogs of podophyllotoxin and related compounds
Authors: Legrand, A Rigo, B Gautret, P Henichart, JP Couturier, D
Citation: A. Legrand et al., Studies on pyrrolidinone. Synthesis of aza analogs of podophyllotoxin and related compounds, J HETERO CH, 36(5), 1999, pp. 1263-1270
A new scaffold for dipeptide beta-turn mimetics: Expeditious synthesis of an unsaturated 6,5-fused bicyclic lactam
Authors: Millet, R Houssin, R Henichart, JP Rigo, B
Citation: R. Millet et al., A new scaffold for dipeptide beta-turn mimetics: Expeditious synthesis of an unsaturated 6,5-fused bicyclic lactam, J HETERO CH, 36(5), 1999, pp. 1279-1284
Bay-12-9566
Authors: Lansiaux, A Henichart, JP Bailly, C
Citation: A. Lansiaux et al., Bay-12-9566, B CANCER, 86(4), 1999, pp. 337-339
Nitration of 6-hydroxy-1-methylpyridin-2-one
Authors: Bouey-Bencteux, E Houssin, R Dogimont, C Henichart, JP
Citation: E. Bouey-bencteux et al., Nitration of 6-hydroxy-1-methylpyridin-2-one, HETEROCYCLE, 48(12), 1998, pp. 2643-2646
Synthesis and antiproliferative properties of 4-aminoquinazoline derivatives as inhibitors of EGF receptor-associated tyrosine kinase activity
Authors: Bouey-Bencteux, E Loison, C Pommery, N Houssin, R Henichart, JP
Citation: E. Bouey-bencteux et al., Synthesis and antiproliferative properties of 4-aminoquinazoline derivatives as inhibitors of EGF receptor-associated tyrosine kinase activity, ANTI-CAN DR, 13(8), 1998, pp. 893-922
Risultati: 1-24 |