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Citation: A. Petit et al., New protease inhibitors prevent gamma-secretase-mediated production of A beta 40/42 without affecting Notch cleavage, NAT CELL BI, 3(5), 2001, pp. 507-511
Authors:
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Citation: P. Vlieghe et al., New 3 '-azido-3 '-deoxythymidin-5 '-yl O-(omega-hydroxyalkyl) carbonate prodrugs: Synthesis and anti-HIV evaluation, J MED CHEM, 44(5), 2001, pp. 777-786
Authors:
Vlieghe, P
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Kraus, JL
Citation: P. Vlieghe et al., New 3 '-azido-3 '-deoxythymidin-5 '-yl O-(4-hydroxyalkyl or -alkenyl or -alkylepoxide) carbonate prodrugs: Synthesis and anti-HIV evaluation, J MED CHEM, 44(18), 2001, pp. 3014-3021
Authors:
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Citation: N. Mourier et al., Synthesis and anti-HIV evaluation of new 2 ',3 '-dideoxy-3 '-thiacytidine prodrugs, NUCLEOS NUC, 19(7), 2000, pp. 1057-1091
Authors:
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Courcambeck, J
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Citation: Jl. Kraus et al., Use of proline bioisosteres in potential HIV protease inhibitors: Phenylalanine-2-thiophenoxy-3-pyrrolidinone: Synthesis and anti-HIV evaluation, BIOORG MED, 10(17), 2000, pp. 2023-2026
Authors:
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Rocheblave, L
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Kraus, JL
Citation: G. Priem et al., Synthesis and chemical reactivity of thiophenoxyphenylalanine bioisosteres, suitable synthons for the design of HIV protease inhibitors, J CHEM S P1, (5), 2000, pp. 819-824
Authors:
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Mourier, N
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Kraus, JL
Citation: M. Camplo et al., Synthesis and biological evaluation of polyaminated 2 ',3 '-dideoxy-3 '-thiacytidine prodrugs, NUCLEOS NUC, 18(4-5), 1999, pp. 879-880
Authors:
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Vlieghe, P
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Kraus, JL
Citation: J. Dessolin et al., New polyazamacrocycle-nucleoside conjugates : Synthesis, anti-HIV evaluation and interaction with CXCR-4 coreceptor, NUCLEOS NUC, 18(4-5), 1999, pp. 881-882
Authors:
Rocheblave, L
Priem, G
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Citation: L. Rocheblave et al., Potent HIV protease inhibitors containing a novel (2-phenylsulfanyl-1-hydroxyethyl)amide isostere, TETRAHEDR L, 40(22), 1999, pp. 4173-4176
Authors:
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Vlieghe, P
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Kraus, JL
Citation: J. Dessolin et al., New Bicyclam-AZT conjugates: Design, synthesis, Anti-HIV evaluation, and their interaction with CXCR-4 coreceptor, J MED CHEM, 42(2), 1999, pp. 229-241