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Results: 1-25 | 26-27
Results: 1-25/27
SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL NAPHTHALENIC AND BIOISOSTERIC RELATED AMIDIC DERIVATIVES AS MELATONIN RECEPTOR LIGANDS
Authors: LECLERC V FOURMAINTRAUX E DEPREUX P LESIEUR D MORGAN P HOWELL HE RENARD P CAIGNARD DH PFEIFFER B DELAGRANGE P GUARDIOLALEMAITRE B ANDRIEUX J
Citation: V. Leclerc et al., SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL NAPHTHALENIC AND BIOISOSTERIC RELATED AMIDIC DERIVATIVES AS MELATONIN RECEPTOR LIGANDS, Bioorganic & medicinal chemistry, 6(10), 1998, pp. 1875-1887
TETRAHYDRONAPHTHALENIC DERIVATIVES AS NEW AGONIST AND ANTAGONIST LIGANDS FOR MELATONIN RECEPTORS
Authors: FOURMAINTRAUX E DEPREUX P LESIEUR D GUARDIOLALEMAITRE B BENNEJEAN C DELAGRANGE P HOWELL HE
Citation: E. Fourmaintraux et al., TETRAHYDRONAPHTHALENIC DERIVATIVES AS NEW AGONIST AND ANTAGONIST LIGANDS FOR MELATONIN RECEPTORS, Bioorganic & medicinal chemistry, 6(1), 1998, pp. 9-13
A HIGH-CONCENTRATION OF MELATONIN INHIBITS IN-VITRO LDL PEROXIDATION BUT NOT OXIDIZED LDL TOXICITY TOWARD CULTURED ENDOTHELIAL-CELLS
Authors: WALTERSLAPORTE E FURMAN C FOUQUET S MARTINNIZARD F LESTAVEL S GOZZO A LESIEUR D FRUCHART JC DURIEZ P TEISSIER E
Citation: E. Walterslaporte et al., A HIGH-CONCENTRATION OF MELATONIN INHIBITS IN-VITRO LDL PEROXIDATION BUT NOT OXIDIZED LDL TOXICITY TOWARD CULTURED ENDOTHELIAL-CELLS, Journal of cardiovascular pharmacology, 32(4), 1998, pp. 582-592
FRIES LIKE REARRANGEMENT - A NOVEL AND EFFICIENT METHOD FOR THE SYNTHESIS OF 6-ACYL-2(3H)-BENZOXAZOLONES AND 6-ACYL-2(3H)-BENZOTHIAZOLONES
Authors: UCAR H VANDERPOORTEN K DEPOVERE P LESIEUR D ISA M MASEREEL B DELARGE J POUPAERT JH
Citation: H. Ucar et al., FRIES LIKE REARRANGEMENT - A NOVEL AND EFFICIENT METHOD FOR THE SYNTHESIS OF 6-ACYL-2(3H)-BENZOXAZOLONES AND 6-ACYL-2(3H)-BENZOTHIAZOLONES, Tetrahedron, 54(9), 1998, pp. 1763-1772
PHARMACOPHORIC SEARCH AND 3D-QSAR COMPARATIVE MOLECULAR-FIELD ANALYSIS STUDIES ON AGONISTS OF MELATONIN SHEEP RECEPTORS
Authors: MAROT C CHAVATTE P MORINALLORY L VIAUD MC GUILLAUMET G RENARD P LESIEUR D MICHEL A
Citation: C. Marot et al., PHARMACOPHORIC SEARCH AND 3D-QSAR COMPARATIVE MOLECULAR-FIELD ANALYSIS STUDIES ON AGONISTS OF MELATONIN SHEEP RECEPTORS, Journal of medicinal chemistry, 41(23), 1998, pp. 4453-4465
NOVEL BENZOTHIAZOLIN-2-ONE AND BENZOXAZIN-3-ONE ARYLPIPERAZINE DERIVATIVES WITH MIXED 5HT(1A) D-2 AFFINITY AS POTENTIAL ATYPICAL ANTIPSYCHOTICS/
Authors: TAVERNE T DIOUF O DEPREUX P POUPAERT JH LESIEUR D GUARDIOLALEMAITRE B RENARD P RETTORI MC CAIGNARD DH PFEIFFER B
Citation: T. Taverne et al., NOVEL BENZOTHIAZOLIN-2-ONE AND BENZOXAZIN-3-ONE ARYLPIPERAZINE DERIVATIVES WITH MIXED 5HT(1A) D-2 AFFINITY AS POTENTIAL ATYPICAL ANTIPSYCHOTICS/, Journal of medicinal chemistry, 41(12), 1998, pp. 2010-2018
5-HT1A AND 5-HT2A LIGANDS WITH ANXIOLYTIC AND ANTIPANIC-LIKE PROPERTIES
Authors: DIOUF O CARATO P DEPREUX P BONTE JP CAIGNARD DH GUARDIOLALEMAITRE B RETTORI MC BELZUNG C LESIEUR D
Citation: O. Diouf et al., 5-HT1A AND 5-HT2A LIGANDS WITH ANXIOLYTIC AND ANTIPANIC-LIKE PROPERTIES, Bioorganic & medicinal chemistry letters, 7(20), 1997, pp. 2579-2584
ALCL3-DMF COMPLEX AS CATALYST IN THE FRIEDEL-CRAFT REACTION - THE REACTIVITY OF ANHYDRIDES AND CHLORIDES OF DICARBOXYLIC-ACIDS
Authors: TAVERNE T DEPREUX P LESIEUR D HENICHART JP POUPAERT JH
Citation: T. Taverne et al., ALCL3-DMF COMPLEX AS CATALYST IN THE FRIEDEL-CRAFT REACTION - THE REACTIVITY OF ANHYDRIDES AND CHLORIDES OF DICARBOXYLIC-ACIDS, Bulletin des Societes chimiques belges, 106(12), 1997, pp. 791-801
PRIMARY AMINES IN THE WILLGERODT-KINDLER REACTION - AN EFFICIENT CONVERSION OF AROMATIC-ALDEHYDES TO THIOAMIDES
Authors: KANYONYO MR GOZZO A LAMBERT DM LESIEUR D POUPAERT JH
Citation: Mr. Kanyonyo et al., PRIMARY AMINES IN THE WILLGERODT-KINDLER REACTION - AN EFFICIENT CONVERSION OF AROMATIC-ALDEHYDES TO THIOAMIDES, Bulletin des Societes chimiques belges, 106(1), 1997, pp. 39-45
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CONFORMATIONALLY RESTRICTED TRICYCLIC ANALOGS OF THE HORMONE MELATONIN
Authors: LECLERC V DEPREUX P LESIEUR D CAIGNARD DH RENARD P DELAGRANGE P GUARDIOLALEMAITRE B MORGAN P
Citation: V. Leclerc et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CONFORMATIONALLY RESTRICTED TRICYCLIC ANALOGS OF THE HORMONE MELATONIN, Bioorganic & medicinal chemistry letters, 6(10), 1996, pp. 1071-1076
EFFECTS OF BOTH A MELATONIN AGONIST AND ANTAGONIST ON SEASONAL-CHANGES IN BODY-MASS AND ENERGY-INTAKE IN THE GARDEN DORMOUSE
Authors: LEGOUIC S DELAGRANGE P ATGIE C NIBBELINK M HANOUN N CASTEILLA L RENARD P LESIEUR D GUARDIOLALEMAITRE B AMBID L
Citation: S. Legouic et al., EFFECTS OF BOTH A MELATONIN AGONIST AND ANTAGONIST ON SEASONAL-CHANGES IN BODY-MASS AND ENERGY-INTAKE IN THE GARDEN DORMOUSE, International journal of obesity, 20(7), 1996, pp. 661-667
ALCL3-DMF REAGENT IN THE FRIEDEL-CRAFTS REACTION - THE BEHAVIOR OF OMEGA-HALOGENOACID CHLORIDES
Authors: POUPAERT JH KANYONYO M UCAR H MOUITHYS AM DIOUF O LESIEUR D
Citation: Jh. Poupaert et al., ALCL3-DMF REAGENT IN THE FRIEDEL-CRAFTS REACTION - THE BEHAVIOR OF OMEGA-HALOGENOACID CHLORIDES, Bulletin des Societes chimiques belges, 105(7), 1996, pp. 397-401
SYNTHESIS OF 6-BENZOYL-2(3H)-BENZOXAZOLONE AND 6-BENZOYL-2(3H)-BENZOTHIAZOLONE
Authors: UCAR H VANDERPOORTEN K KANYONYO M ISA M LAMBERT D LESIEUR D POUPAERT JH
Citation: H. Ucar et al., SYNTHESIS OF 6-BENZOYL-2(3H)-BENZOXAZOLONE AND 6-BENZOYL-2(3H)-BENZOTHIAZOLONE, Bulletin des Societes chimiques belges, 105(12), 1996, pp. 773-776
SOLVENT EFFECT IN THE WOLLGERODT-KINDLER REACTION
Authors: KANYONYO MR UCAR H ISA M CARATO P LESIEUR D RENARD P POUPAERT JH
Citation: Mr. Kanyonyo et al., SOLVENT EFFECT IN THE WOLLGERODT-KINDLER REACTION, Bulletin des Societes chimiques belges, 105(1), 1996, pp. 17-22
6-(N-IMIDOALKYL)AMINOALKYLBENZOTHIAZOLIN-2-ONES AS LIGANDS OF THE SEROTONINERGIC 5-HT1A RECEPTORS
Authors: DIOUF O DEPREUX P LESIEUR D POUPAERT JH CAIGNARD DH
Citation: O. Diouf et al., 6-(N-IMIDOALKYL)AMINOALKYLBENZOTHIAZOLIN-2-ONES AS LIGANDS OF THE SEROTONINERGIC 5-HT1A RECEPTORS, Heterocycles, 41(6), 1995, pp. 1219-1233
STRUCTURE-ACTIVITY-RELATIONSHIPS OF MELATONIN ANALOGS
Authors: CAIGNARD DH LESIEUR D DEPREUX P RENARD P DELAGRANGE P GUARDIOLALEMAITRE B
Citation: Dh. Caignard et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF MELATONIN ANALOGS, European journal of medicinal chemistry, 30, 1995, pp. 637-642
SYNTHESIS AND EVALUATION OF NEW 2-PIPERAZINYLBENZOTHIAZOLES WITH HIGH5-HT1A AND 5-HT3 AFFINITIES
Authors: DIOUF O DEPREUX P LESIEUR D POUPAERT JH CAIGNARD DH
Citation: O. Diouf et al., SYNTHESIS AND EVALUATION OF NEW 2-PIPERAZINYLBENZOTHIAZOLES WITH HIGH5-HT1A AND 5-HT3 AFFINITIES, European journal of medicinal chemistry, 30(9), 1995, pp. 715-719
(METHYLAMINOSULFONYLMETHYL)-1-NAPHTHYL]ETHYLAMINE, THE NAPHTHALENIC BIOISOSTERE OF SUMATRIPTAN
Authors: TINANT B DECLERCQ JP ABDELLAOUI H DEPREUX P LESIEUR D
Citation: B. Tinant et al., (METHYLAMINOSULFONYLMETHYL)-1-NAPHTHYL]ETHYLAMINE, THE NAPHTHALENIC BIOISOSTERE OF SUMATRIPTAN, Acta crystallographica. Section C, Crystal structure communications, 51, 1995, pp. 916-918
SYNTHESIS OF THE NAPHTHALENIC BIOISOSTERE OF THE ANTIMIGRAINE DRUG SUMATRIPTAN
Authors: ABDELLAOUI H DEPREUX P LESIEUR D PFEIFFER B BONTEMPELLI P
Citation: H. Abdellaoui et al., SYNTHESIS OF THE NAPHTHALENIC BIOISOSTERE OF THE ANTIMIGRAINE DRUG SUMATRIPTAN, Synthetic communications, 25(9), 1995, pp. 1303-1311
S14080, A PERIPHERAL ANALGESIC ACTING BY RELEASE OF AN ENDOGENOUS CIRCULATING OPIOID-LIKE SUBSTANCE
Authors: FERREIRA SH LORENZETTI BB DEVISSAGUET M LESIEUR D TSOUDEROS Y
Citation: Sh. Ferreira et al., S14080, A PERIPHERAL ANALGESIC ACTING BY RELEASE OF AN ENDOGENOUS CIRCULATING OPIOID-LIKE SUBSTANCE, British Journal of Pharmacology, 114(2), 1995, pp. 303-308
N-[2-(7-METHOXY-1-NAPHTHYL)ETHYL]ACETAMIDE, A POTENT MELATONIN ANALOG
Authors: TINANT B DECLERCQ JP POUPAERT JH YOUS S LESIEUR D
Citation: B. Tinant et al., N-[2-(7-METHOXY-1-NAPHTHYL)ETHYL]ACETAMIDE, A POTENT MELATONIN ANALOG, Acta crystallographica. Section C, Crystal structure communications, 50, 1994, pp. 907-910
REGIOSELECTIVE SYNTHESIS OF BENZIMIDAZOLIC BIOISOSTERES OF MELATONIN
Authors: DEPREUX P FOURMAINTRAUX E LESIEUR D RENARD P
Citation: P. Depreux et al., REGIOSELECTIVE SYNTHESIS OF BENZIMIDAZOLIC BIOISOSTERES OF MELATONIN, Synthetic communications, 24(15), 1994, pp. 2123-2132
ALCL3-DMF REAGENT IN THE FRIEDEL-CRAFTS REACTION - APPLICATION TO THEACYLATION REACTION OF 2(3H)-BENZOTHIAZOLONES
Authors: YOUS S POUPAERT JH LESIEUR I DEPREUX P LESIEUR D
Citation: S. Yous et al., ALCL3-DMF REAGENT IN THE FRIEDEL-CRAFTS REACTION - APPLICATION TO THEACYLATION REACTION OF 2(3H)-BENZOTHIAZOLONES, Journal of organic chemistry, 59(6), 1994, pp. 1574-1576
SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL NAPHTHALENIC AND BIOISOSTERIC RELATED AMIDIC DERIVATIVES AS MELATONIN RECEPTOR LIGANDS
Authors: DEPREUX P LESIEUR D MANSOUR HA MORGAN P HOWELL HE RENARD P CAIGNARD DH PFEIFFER B DELAGRANGE P GUARDIOLA B YOUS S DEMARQUE A ADAM G ANDRIEUX J
Citation: P. Depreux et al., SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL NAPHTHALENIC AND BIOISOSTERIC RELATED AMIDIC DERIVATIVES AS MELATONIN RECEPTOR LIGANDS, Journal of medicinal chemistry, 37(20), 1994, pp. 3231-3239
BENZOSELENAZOLINONE DERIVATIVES DESIGNED TO BE GLUTATHIONE-PEROXIDASEMIMETICS FEATURE INHIBITION OF CYCLOOXYGENASE 5-LIPOXYGENASE PATHWAYSAND ANTIINFLAMMATORY ACTIVITY/
Authors: GALET V BERNIER JL HENICHART JP LESIEUR D ABADIE C ROCHETTE L LINDENBAUM A CHALAS J DELAFAVERIE JFR PFEIFFER B RENARD P
Citation: V. Galet et al., BENZOSELENAZOLINONE DERIVATIVES DESIGNED TO BE GLUTATHIONE-PEROXIDASEMIMETICS FEATURE INHIBITION OF CYCLOOXYGENASE 5-LIPOXYGENASE PATHWAYSAND ANTIINFLAMMATORY ACTIVITY/, Journal of medicinal chemistry, 37(18), 1994, pp. 2903-2911
Risultati: 1-25 | 26-27