Authors:
MANFREDINI S
SIMONI D
CAMINITI G
VERTUANI S
INVIDIATA F
MOSCATO B
HATSE S
DECLERCQ E
BALZARINI J
Citation: S. Manfredini et al., RETINOIDS AS POTENTIAL CHEMOTHERAPEUTIC-AGENTS - SYNTHESIS, CYTOSTATIC AND DIFFERENTIATING ACTIVITIES OF NEW HETEROCYCLIC-ANALOGS OF RETINOIC ACID, Medicinal chemistry research, 8(6), 1998, pp. 291-304
Authors:
MAY EL
JACOBSON AE
MATTSON MV
COOP A
ACETO MD
BOWMAN ER
TRAYNOR JR
WOODS JH
HARRIS LS
Citation: El. May et al., SYNTHESIS, IN-VITRO, AND IN-VIVO ACTIVITY OF N-P-SUBSTITUTEDBENZYL- (-)- AND (-N-NORMETAZOCINES, (-)- AND (+)-N-NORMORPHINANS, N-NORKETOBEMIDONES, AND (-)-N-NOR-4,5-EPOXYMORPHINANS()), Medicinal chemistry research, 8(6), 1998, pp. 311-321
Authors:
BUCHOLTZ EC
WYRICK SD
OWENS CE
MCPHAIL AT
BOOTH RG
Citation: Ec. Bucholtz et al., ENYL-3-DIMETHYLAMINO-1,2,3,4-TETRAHYDRONAPHTHALENE (H-2-PAT) - EFFECTOF STEREOCHEMISTRY ON BINDING AND FUNCTION AT BRAIN HISTAMINE-RECEPTORS, Medicinal chemistry research, 8(6), 1998, pp. 322-332
Authors:
COFFEN DL
BALDINO CM
LANGE M
TILTON RF
TU C
Citation: Dl. Coffen et al., MOLECULAR DIVERSITY, BIOLOGICAL-ACTIVITY AND COMMON GROUND SHARED BY BOTH, Medicinal chemistry research, 8(4-5), 1998, pp. 206-218
Authors:
ILLIG C
EISENNAGEL S
BONE R
RADZICKA A
MURPHY L
RANDLE T
SPURLINO J
SALEMME FR
SOLL RM
Citation: C. Illig et al., EXPANDING THE ENVELOPE OF STRUCTURE-BASED DRUG DESIGN USING CHEMICAL LIBRARIES - APPLICATION TO SMALL-MOLECULE INHIBITORS OF THROMBIN, Medicinal chemistry research, 8(4-5), 1998, pp. 244-260
Citation: Dp. Curran et Zy. Luo, RAPID, PARALLEL SYNTHESIS OF HOMOALLYLIC ALCOHOLS BY LEWIS-ACID MEDIATED ALLYLATIONS OF ALDEHYDES WITH NEW FLUOROUS ALLYL STANNANES, Medicinal chemistry research, 8(4-5), 1998, pp. 261-265
Citation: M. Deutsch, STRUCTURE-ACTIVITY-RELATIONSHIPS FOR METHYLPHENIDATE ANALOGS AND COMPARISONS TO COCAINE AND TROPANES. (VOL 8, PG 91, 1998), Medicinal chemistry research, 8(4-5), 1998, pp. 276-276
Authors:
YANG B
JOHNSTON DE
LUEDTKE RR
HAMMOND PS
MACH RH
Citation: B. Yang et al., SYNTHESIS AND IN-VITRO BINDING OF N-ALKYL-2,3-DIMETHOXY-[3.3.1]AZABICYCLONONANE BENZAMIDES AT DOPAMINE D-2 AND D-3 RECEPTORS, Medicinal chemistry research, 8(3), 1998, pp. 115-131
Citation: M. Lamothe et al., SYNTHESIS OF NEW BENZOTHIENYLPIPERAZINE DERIVATIVES AND THEIR CHARACTERIZATION AT BOTH 5HT(1A) AND 5HT(1B) RECEPTOR-SITES, Medicinal chemistry research, 8(3), 1998, pp. 132-142
Citation: I. Doytchinova et S. Petrova, N6-N7 - A MODIFICATION OF THE N6-C8 MODEL FOR THE BINDING-SITE ON ADENOSINE-A1-RECEPTORS WITH IMPROVED STERIC AND ELECTROSTATIC FIT, Medicinal chemistry research, 8(3), 1998, pp. 143-152
Authors:
BRYANS JS
HORWELL DC
MCGUFFOG J
MORRELL AI
ONIELL JA
RATCLIFFE GS
Citation: Js. Bryans et al., BIOACTIVE CONFORMATIONS OF LIGANDS FOR THE CALCIUM-CHANNEL ALPHA(2)DELTA GABAPENTIN BINDING-SITE, Medicinal chemistry research, 8(3), 1998, pp. 153-162
Authors:
ELMOSELHY TF
ELKERSH MA
NYBERG F
HEDE R
ELDAWY MA
Citation: Tf. Elmoselhy et al., PREPARATION AND EVALUATION OF SOME ANTIARRHYTHMIC AND CARDIAC INOTROPIC AGENTS AS COLD ANALOGS OF POTENTIAL MYOCARDIAL IMAGING AGENTS, Medicinal chemistry research, 8(3), 1998, pp. 163-170
Citation: Pc. Meltzer et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF INHIBITION OF THE DOPAMINE TRANSPORTER BY 3-ARYLBICYCLO[3.2.1]OCTANES, Medicinal chemistry research, 8(1-2), 1998, pp. 12-34
Authors:
LOMENZO SA
IZENWASSER S
KATZ JL
TRUDELL ML
Citation: Sa. Lomenzo et al., THE EFFECTS OF ALKYL SUBSTITUENTS AT THE 6-POSITION OF COCAINE ANALOGS ON DOPAMINE TRANSPORTER BINDING-AFFINITY AND DOPAMINE UPTAKE INHIBITION, Medicinal chemistry research, 8(1-2), 1998, pp. 35-42
Authors:
PRAKASH KRC
ARALDI GL
SMITH MP
ZHANG M
JOHNSON KM
KOZIKOWSKI AP
Citation: Krc. Prakash et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF NEW 6-SUBSTITUTED AND 7-SUBSTITUTED 2-BETA-BUTYL-3-PHENYLTROPANES AS LIGANDS FOR THE DOPAMINE TRANSPORTER, Medicinal chemistry research, 8(1-2), 1998, pp. 43-58