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Results: 1-23 |
Results: 23
COUMARIN 1,4-DIHYDROPYRIDINE DERIVATIVES
Authors: VALENTI P RAMPA A BUDRIESI R BISI A CHIARINI A
Citation: P. Valenti et al., COUMARIN 1,4-DIHYDROPYRIDINE DERIVATIVES, Bioorganic & medicinal chemistry, 6(6), 1998, pp. 803-810
SEARCH FOR ALPHA(1)-ADRENOCEPTOR SUBTYPES SELECTIVE ANTAGONISTS - DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CYSTAZOSIN, AN ALPHA(1D)-ADRENOCEPTOR ANTAGONIST
Authors: MINARINI A BUDRIESI R CHIARINI A LEONARDI A MELCHIORRE C
Citation: A. Minarini et al., SEARCH FOR ALPHA(1)-ADRENOCEPTOR SUBTYPES SELECTIVE ANTAGONISTS - DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CYSTAZOSIN, AN ALPHA(1D)-ADRENOCEPTOR ANTAGONIST, Bioorganic & medicinal chemistry letters, 8(11), 1998, pp. 1353-1358
DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF PRAZOSIN-RELATED ANTAGONISTS - ROLE OF THE PIPERAZINE AND FURAN UNITS OF PRAZOSIN ON THE SELECTIVITY FOR ALPHA(1)-ADRENORECEPTOR SUBTYPES
Authors: BOLOGNESI ML BUDRIESI R CHIARINI A POGGESI E LEONARDI A MELCHIORRE C
Citation: Ml. Bolognesi et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF PRAZOSIN-RELATED ANTAGONISTS - ROLE OF THE PIPERAZINE AND FURAN UNITS OF PRAZOSIN ON THE SELECTIVITY FOR ALPHA(1)-ADRENORECEPTOR SUBTYPES, Journal of medicinal chemistry, 41(24), 1998, pp. 4844-4853
ACETYLCHOLINESTERASE NONCOVALENT INHIBITORS BASED ON A POLYAMINE BACKBONE FOR POTENTIAL USE AGAINST ALZHEIMERS-DISEASE
Authors: MELCHIORRE C ANDRISANO V BOLOGNESI ML BUDRIESI R CAVALLI A CAVRINI V ROSINI M TUMIATTI V RECANATINI M
Citation: C. Melchiorre et al., ACETYLCHOLINESTERASE NONCOVALENT INHIBITORS BASED ON A POLYAMINE BACKBONE FOR POTENTIAL USE AGAINST ALZHEIMERS-DISEASE, Journal of medicinal chemistry, 41(22), 1998, pp. 4186-4189
UNIVERSAL TEMPLATE APPROACH TO DRUG DESIGN - POLYAMINES AS SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS
Authors: BOLOGNESI ML MINARINI A BUDRIESI R CACCIAGUERRA S CHIARINI A SPAMPINATO S TUMIATTI V MELCHIORRE C
Citation: Ml. Bolognesi et al., UNIVERSAL TEMPLATE APPROACH TO DRUG DESIGN - POLYAMINES AS SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4150-4160
SEARCH FOR SELECTIVE ANTAGONISTS AT ALPHA(1)-ADRENORECEPTORS - NEUTRAL OR NEGATIVE ANTAGONISM
Authors: MELCHIORRE C BOLOGNESI ML BUDRIESI R CHIARINI A GIARDINA D MINARINI A QUAGLIA W LEONARDI A
Citation: C. Melchiorre et al., SEARCH FOR SELECTIVE ANTAGONISTS AT ALPHA(1)-ADRENORECEPTORS - NEUTRAL OR NEGATIVE ANTAGONISM, Il Farmaco, 53(4), 1998, pp. 278-286
SELECTIVE CARDIODEPRESSANT ACTIVITY OF FLUODIPINE, A FLUORENONE-1,4-DIHYDROPYRIDINE DERIVATIVE
Authors: BUDRIESI R AICARDI G CAMPANA G SPAMPINATO S ZAZA A BISI A RAMPA A VALENTI P CHIARINI A
Citation: R. Budriesi et al., SELECTIVE CARDIODEPRESSANT ACTIVITY OF FLUODIPINE, A FLUORENONE-1,4-DIHYDROPYRIDINE DERIVATIVE, European journal of pharmacology, 359(2-3), 1998, pp. 161-170
SYNTHESIS AND BIOLOGICAL PROFILE AT MUSCARINIC M(2) AND M(3) RECEPTORSUBTYPES OF SOME ANALOGS OF DIPHENIDOL
Authors: VAROLI L BURNELLI S BUDRIESI R GUARNIERI A CHIARINI A RECANATINI M
Citation: L. Varoli et al., SYNTHESIS AND BIOLOGICAL PROFILE AT MUSCARINIC M(2) AND M(3) RECEPTORSUBTYPES OF SOME ANALOGS OF DIPHENIDOL, Medicinal chemistry research, 6(9), 1996, pp. 571-580
CARDIOVASCULAR CHARACTERIZATION OF PYRROLO[2,1-D][1,5]BENZOTHIAZEPINEDERIVATIVES BINDING SELECTIVELY TO THE PERIPHERAL-TYPE BENZODIAZEPINERECEPTOR (PBR) - FROM DUAL PBR AFFINITY AND CALCIUM-ANTAGONIST ACTIVITY TO NOVEL AND SELECTIVE CALCIUM-ENTRY BLOCKERS
Authors: CAMPIANI G FIORINI I DEFILIPPIS MP CIANI SM GAROFALO A NACCI V GIORGI G SEGA A BOTTA M CHIARINI A BUDRIESI R BRUNI G ROMEO MR MANZONI C MENNINI T
Citation: G. Campiani et al., CARDIOVASCULAR CHARACTERIZATION OF PYRROLO[2,1-D][1,5]BENZOTHIAZEPINEDERIVATIVES BINDING SELECTIVELY TO THE PERIPHERAL-TYPE BENZODIAZEPINERECEPTOR (PBR) - FROM DUAL PBR AFFINITY AND CALCIUM-ANTAGONIST ACTIVITY TO NOVEL AND SELECTIVE CALCIUM-ENTRY BLOCKERS, Journal of medicinal chemistry, 39(15), 1996, pp. 2922-2938
SYNTHESIS AND PHARMACOLOGICAL PROFILE OF SOME CHLOROXANTHONE-1,4-DIHYDROPYRIDINE DERIVATIVES
Authors: BISI A BUDRIESI R RAMPA A FABBRI G CHIARINI A VALENTI P
Citation: A. Bisi et al., SYNTHESIS AND PHARMACOLOGICAL PROFILE OF SOME CHLOROXANTHONE-1,4-DIHYDROPYRIDINE DERIVATIVES, Arzneimittel-Forschung, 46(9), 1996, pp. 848-851
STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF XANTHONE AND FLUORENONE-1,4-DIHYDROPYRIDINE-5-PHOSPHONATES
Authors: BUDRIESI R RAMPA A BISI A FABBRI G CHIARINI A VALENTI P
Citation: R. Budriesi et al., STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF XANTHONE AND FLUORENONE-1,4-DIHYDROPYRIDINE-5-PHOSPHONATES, Arzneimittel-Forschung, 46(4), 1996, pp. 374-377
DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME 4-DAMP-RELATED COMPOUNDS
Authors: TUMIATTI V SPAMPINATO S RECANATINI M MINARINI A MELCHIORRE C CHIARINI A BUDRIESI R
Citation: V. Tumiatti et al., DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME 4-DAMP-RELATED COMPOUNDS, Bioorganic & medicinal chemistry letters, 5(20), 1995, pp. 2325-2330
THE DESIGN OF NOVEL METHOCTRAMINE-RELATED TETRAAMINES AS MUSCARINIC RECEPTOR SUBTYPE-SELECTIVE ANTAGONISTS
Authors: MELCHIORRE C MINARINI A BUDRIESI R CHIARINI A SPAMPINATO S TUMIATTI V
Citation: C. Melchiorre et al., THE DESIGN OF NOVEL METHOCTRAMINE-RELATED TETRAAMINES AS MUSCARINIC RECEPTOR SUBTYPE-SELECTIVE ANTAGONISTS, Life sciences, 56(11-12), 1995, pp. 837-844
PYRROLO[2,1-C][1,4] BENZOTHIAZINES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, MOLECULAR MODELING STUDIES, AND CARDIOVASCULAR ACTIVITY
Authors: CAMPIANI G GAROFALO A FIORINI I BETTA M NACCI V TAFI A CHIARINI A BUDRIESI R BRUNI G ROMEO MR
Citation: G. Campiani et al., PYRROLO[2,1-C][1,4] BENZOTHIAZINES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, MOLECULAR MODELING STUDIES, AND CARDIOVASCULAR ACTIVITY, Journal of medicinal chemistry, 38(22), 1995, pp. 4393-4410
1,4-DIHYDROPYRIDINES CONTAINING R-NNO-AZOXY MOIETIES
Authors: GASCO AM ERMONDI G GASCO A BUDRIESI R CHIARINI A
Citation: Am. Gasco et al., 1,4-DIHYDROPYRIDINES CONTAINING R-NNO-AZOXY MOIETIES, Il Farmaco, 50(1), 1995, pp. 61-64
IN-VITRO CHARACTERIZATION OF TRIPITRAMINE, A POLYMETHYLENE TETRAAMINEDISPLAYING HIGH SELECTIVITY AND AFFINITY FOR MUSCARINIC M(2) RECEPTORS
Authors: CHIARINI A BUDRIESI R BOLOGNESI ML MINARINI A MELCHIORRE C
Citation: A. Chiarini et al., IN-VITRO CHARACTERIZATION OF TRIPITRAMINE, A POLYMETHYLENE TETRAAMINEDISPLAYING HIGH SELECTIVITY AND AFFINITY FOR MUSCARINIC M(2) RECEPTORS, British Journal of Pharmacology, 114(7), 1995, pp. 1507-1517
STRUCTURE-ACTIVITY RELATIONSHIP STUDIES IN THE FIELD OF CALCIUM-ANTAGONISTS - XANTHONE 1,4-DIHYDROPYRIDINES BEARING A 2,3-LACTONE RING
Authors: RAMPA A BUDRIESI R BISI A FABBRI G BARILI PL CHIARINI A VALENTI P
Citation: A. Rampa et al., STRUCTURE-ACTIVITY RELATIONSHIP STUDIES IN THE FIELD OF CALCIUM-ANTAGONISTS - XANTHONE 1,4-DIHYDROPYRIDINES BEARING A 2,3-LACTONE RING, Arzneimittel-Forschung, 45-2(9), 1995, pp. 957-962
SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF SOME BENZAZEPINONE DERIVATIVES
Authors: BUDRIESI R RAMPA A BISI A FABBRI G CHIARINI A VALENTI P
Citation: R. Budriesi et al., SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF SOME BENZAZEPINONE DERIVATIVES, Arzneimittel-Forschung, 45-1(3), 1995, pp. 234-239
SYNTHESIS AND IN-VITRO CARDIOVASCULAR ACTIVITY OF TRAHYDRO-1H-PYRROLO[2,1-C][1,4]BENZOTHIAZIN-1-ONES AND TETRAHYDROPYRROLO[2,1-D][1,5]BENZOTHIAZEPIN-10-ONE
Authors: CAMPIANI G GAROFALO A FIORINI I NACCI V BOTTA M TAFI A CHIARINI A BUDRIESI R BRUNI G ROMEO MR
Citation: G. Campiani et al., SYNTHESIS AND IN-VITRO CARDIOVASCULAR ACTIVITY OF TRAHYDRO-1H-PYRROLO[2,1-C][1,4]BENZOTHIAZIN-1-ONES AND TETRAHYDROPYRROLO[2,1-D][1,5]BENZOTHIAZEPIN-10-ONE, Bioorganic & medicinal chemistry letters, 4(10), 1994, pp. 1235-1240
SEMIRIGID ANALOGS OF THE CALCIUM-ANTAGONIST VERAPAMIL - A MOLECULAR MODELING STUDY
Authors: ROMANELLI MN DEI S SCAPECCHI S TEODORI E GUALTIERI F BUDRIESI R MANNHOLD R
Citation: Mn. Romanelli et al., SEMIRIGID ANALOGS OF THE CALCIUM-ANTAGONIST VERAPAMIL - A MOLECULAR MODELING STUDY, Journal of computer-aided molecular design, 8(2), 1994, pp. 123-134
SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF VERAPAMIL ANALOGS WITH RESTRICTED MOLECULAR FLEXIBILITY
Authors: TEODORI E DEI S ROMANELLI MN SCAPECCHI S GUALTIERI F BUDRIESI R CHIARINI A LEMOINE H MANNHOLD R
Citation: E. Teodori et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF VERAPAMIL ANALOGS WITH RESTRICTED MOLECULAR FLEXIBILITY, European journal of medicinal chemistry, 29(2), 1994, pp. 139-148
DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF METHOCTRAMINE-RELATED TETRAAMINES BEARING AN 1-DIHYDRO-6H-PYRIDO[2,3-B][1,4]BENZODIAZEPIN-6-ONE MOIETY - STRUCTURAL REQUIREMENTS FOR OPTIMUM OCCUPANCY OF MUSCARINIC RECEPTOR SUBTYPES AS REVEALED BY SYMMETRICAL AND UNSYMMETRICAL POLYAMINES
Authors: MINARINI A BOLOGNESI ML BUDRIESI R CANOSSA M CHIARINI A SPAMPINATO S MELCHIORRE C
Citation: A. Minarini et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF METHOCTRAMINE-RELATED TETRAAMINES BEARING AN 1-DIHYDRO-6H-PYRIDO[2,3-B][1,4]BENZODIAZEPIN-6-ONE MOIETY - STRUCTURAL REQUIREMENTS FOR OPTIMUM OCCUPANCY OF MUSCARINIC RECEPTOR SUBTYPES AS REVEALED BY SYMMETRICAL AND UNSYMMETRICAL POLYAMINES, Journal of medicinal chemistry, 37(20), 1994, pp. 3363-3372
SAR STUDIES IN THE FIELD OF CA-ANTAGONISTS - 2-SUBSTITUTED 1,4-DIHYDROPYRIDINES WITH A XANTHONE BACKBONE
Authors: BISI A BUDRIESI R CHIARINI A RAMPA A VALENTI P
Citation: A. Bisi et al., SAR STUDIES IN THE FIELD OF CA-ANTAGONISTS - 2-SUBSTITUTED 1,4-DIHYDROPYRIDINES WITH A XANTHONE BACKBONE, Il Farmaco, 48(11), 1993, pp. 1491-1502
Risultati: 1-23 |