Authors:
MINARINI A
BUDRIESI R
CHIARINI A
LEONARDI A
MELCHIORRE C
Citation: A. Minarini et al., SEARCH FOR ALPHA(1)-ADRENOCEPTOR SUBTYPES SELECTIVE ANTAGONISTS - DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CYSTAZOSIN, AN ALPHA(1D)-ADRENOCEPTOR ANTAGONIST, Bioorganic & medicinal chemistry letters, 8(11), 1998, pp. 1353-1358
Authors:
BOLOGNESI ML
BUDRIESI R
CHIARINI A
POGGESI E
LEONARDI A
MELCHIORRE C
Citation: Ml. Bolognesi et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF PRAZOSIN-RELATED ANTAGONISTS - ROLE OF THE PIPERAZINE AND FURAN UNITS OF PRAZOSIN ON THE SELECTIVITY FOR ALPHA(1)-ADRENORECEPTOR SUBTYPES, Journal of medicinal chemistry, 41(24), 1998, pp. 4844-4853
Authors:
BOLOGNESI ML
MINARINI A
BUDRIESI R
CACCIAGUERRA S
CHIARINI A
SPAMPINATO S
TUMIATTI V
MELCHIORRE C
Citation: Ml. Bolognesi et al., UNIVERSAL TEMPLATE APPROACH TO DRUG DESIGN - POLYAMINES AS SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4150-4160
Authors:
MELCHIORRE C
BOLOGNESI ML
BUDRIESI R
CHIARINI A
GIARDINA D
MINARINI A
QUAGLIA W
LEONARDI A
Citation: C. Melchiorre et al., SEARCH FOR SELECTIVE ANTAGONISTS AT ALPHA(1)-ADRENORECEPTORS - NEUTRAL OR NEGATIVE ANTAGONISM, Il Farmaco, 53(4), 1998, pp. 278-286
Authors:
BUDRIESI R
AICARDI G
CAMPANA G
SPAMPINATO S
ZAZA A
BISI A
RAMPA A
VALENTI P
CHIARINI A
Citation: R. Budriesi et al., SELECTIVE CARDIODEPRESSANT ACTIVITY OF FLUODIPINE, A FLUORENONE-1,4-DIHYDROPYRIDINE DERIVATIVE, European journal of pharmacology, 359(2-3), 1998, pp. 161-170
Authors:
VAROLI L
BURNELLI S
BUDRIESI R
GUARNIERI A
CHIARINI A
RECANATINI M
Citation: L. Varoli et al., SYNTHESIS AND BIOLOGICAL PROFILE AT MUSCARINIC M(2) AND M(3) RECEPTORSUBTYPES OF SOME ANALOGS OF DIPHENIDOL, Medicinal chemistry research, 6(9), 1996, pp. 571-580
Authors:
GRECO D
SALMASO S
MASTRANTONIO P
GIULIANO M
TOZZI AE
ANEMONA A
ATTI MLCD
GIAMMANCO A
PANEI P
BLACKWELDER WC
KLEIN DL
WASSILAK SGF
STEFANELLI P
BOTTONE M
SOFIA T
LUZI S
BELLOMI G
COBIANCHI F
CANGANELLA G
MEDURI F
SCUDERI G
CHIARINI A
MAGGIO M
TAORMINA S
GENOVESE M
MOIRAGHI A
BARALE A
DITOMMASO S
MALASPINA S
VASILE E
FERRARO P
DALLAGO P
DEMARZI L
ROBINO L
GIRALDO E
COPPOLA N
MATERASSI P
CASTELLANI GT
BASSO F
BARBUTI S
QUARTO M
LOPALCO P
DORAZIO P
SANGUEDOLCE A
Citation: D. Greco et al., A CONTROLLED TRIAL OF 2 ACELLULAR VACCINES AND ONE WHOLE-CELL VACCINEAGAINST PERTUSSIS, The New England journal of medicine, 334(6), 1996, pp. 341-348
Authors:
CAMPIANI G
FIORINI I
DEFILIPPIS MP
CIANI SM
GAROFALO A
NACCI V
GIORGI G
SEGA A
BOTTA M
CHIARINI A
BUDRIESI R
BRUNI G
ROMEO MR
MANZONI C
MENNINI T
Citation: G. Campiani et al., CARDIOVASCULAR CHARACTERIZATION OF PYRROLO[2,1-D][1,5]BENZOTHIAZEPINEDERIVATIVES BINDING SELECTIVELY TO THE PERIPHERAL-TYPE BENZODIAZEPINERECEPTOR (PBR) - FROM DUAL PBR AFFINITY AND CALCIUM-ANTAGONIST ACTIVITY TO NOVEL AND SELECTIVE CALCIUM-ENTRY BLOCKERS, Journal of medicinal chemistry, 39(15), 1996, pp. 2922-2938
Authors:
BISI A
BUDRIESI R
RAMPA A
FABBRI G
CHIARINI A
VALENTI P
Citation: A. Bisi et al., SYNTHESIS AND PHARMACOLOGICAL PROFILE OF SOME CHLOROXANTHONE-1,4-DIHYDROPYRIDINE DERIVATIVES, Arzneimittel-Forschung, 46(9), 1996, pp. 848-851
Authors:
BUDRIESI R
RAMPA A
BISI A
FABBRI G
CHIARINI A
VALENTI P
Citation: R. Budriesi et al., STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF XANTHONE AND FLUORENONE-1,4-DIHYDROPYRIDINE-5-PHOSPHONATES, Arzneimittel-Forschung, 46(4), 1996, pp. 374-377
Authors:
TUMIATTI V
SPAMPINATO S
RECANATINI M
MINARINI A
MELCHIORRE C
CHIARINI A
BUDRIESI R
Citation: V. Tumiatti et al., DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME 4-DAMP-RELATED COMPOUNDS, Bioorganic & medicinal chemistry letters, 5(20), 1995, pp. 2325-2330
Authors:
MELCHIORRE C
MINARINI A
BUDRIESI R
CHIARINI A
SPAMPINATO S
TUMIATTI V
Citation: C. Melchiorre et al., THE DESIGN OF NOVEL METHOCTRAMINE-RELATED TETRAAMINES AS MUSCARINIC RECEPTOR SUBTYPE-SELECTIVE ANTAGONISTS, Life sciences, 56(11-12), 1995, pp. 837-844
Authors:
CAMPIANI G
GAROFALO A
FIORINI I
BETTA M
NACCI V
TAFI A
CHIARINI A
BUDRIESI R
BRUNI G
ROMEO MR
Citation: G. Campiani et al., PYRROLO[2,1-C][1,4] BENZOTHIAZINES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, MOLECULAR MODELING STUDIES, AND CARDIOVASCULAR ACTIVITY, Journal of medicinal chemistry, 38(22), 1995, pp. 4393-4410
Authors:
CHIARINI A
BUDRIESI R
BOLOGNESI ML
MINARINI A
MELCHIORRE C
Citation: A. Chiarini et al., IN-VITRO CHARACTERIZATION OF TRIPITRAMINE, A POLYMETHYLENE TETRAAMINEDISPLAYING HIGH SELECTIVITY AND AFFINITY FOR MUSCARINIC M(2) RECEPTORS, British Journal of Pharmacology, 114(7), 1995, pp. 1507-1517
Authors:
RAMPA A
BUDRIESI R
BISI A
FABBRI G
BARILI PL
CHIARINI A
VALENTI P
Citation: A. Rampa et al., STRUCTURE-ACTIVITY RELATIONSHIP STUDIES IN THE FIELD OF CALCIUM-ANTAGONISTS - XANTHONE 1,4-DIHYDROPYRIDINES BEARING A 2,3-LACTONE RING, Arzneimittel-Forschung, 45-2(9), 1995, pp. 957-962
Authors:
BUDRIESI R
RAMPA A
BISI A
FABBRI G
CHIARINI A
VALENTI P
Citation: R. Budriesi et al., SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF SOME BENZAZEPINONE DERIVATIVES, Arzneimittel-Forschung, 45-1(3), 1995, pp. 234-239
Authors:
CAMPIANI G
GAROFALO A
FIORINI I
NACCI V
BOTTA M
TAFI A
CHIARINI A
BUDRIESI R
BRUNI G
ROMEO MR
Citation: G. Campiani et al., SYNTHESIS AND IN-VITRO CARDIOVASCULAR ACTIVITY OF TRAHYDRO-1H-PYRROLO[2,1-C][1,4]BENZOTHIAZIN-1-ONES AND TETRAHYDROPYRROLO[2,1-D][1,5]BENZOTHIAZEPIN-10-ONE, Bioorganic & medicinal chemistry letters, 4(10), 1994, pp. 1235-1240
Authors:
TEODORI E
DEI S
ROMANELLI MN
SCAPECCHI S
GUALTIERI F
BUDRIESI R
CHIARINI A
LEMOINE H
MANNHOLD R
Citation: E. Teodori et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF VERAPAMIL ANALOGS WITH RESTRICTED MOLECULAR FLEXIBILITY, European journal of medicinal chemistry, 29(2), 1994, pp. 139-148
Authors:
VENERANDO B
FIORILLI A
DIFRANCESCO L
CHIARINI A
MONTI E
ZIZIOLI D
TETTAMANTI G
Citation: B. Venerando et al., CYTOSOLIC SIALIDASE FROM PIG BRAIN - A PROTEIN COMPLEX CONTAINING CATALYTIC AND PROTECTIVE UNITS, Biochimica et biophysica acta. Protein structure and molecular enzymology, 1208(2), 1994, pp. 229-237
Authors:
MINARINI A
BOLOGNESI ML
BUDRIESI R
CANOSSA M
CHIARINI A
SPAMPINATO S
MELCHIORRE C
Citation: A. Minarini et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF METHOCTRAMINE-RELATED TETRAAMINES BEARING AN 1-DIHYDRO-6H-PYRIDO[2,3-B][1,4]BENZODIAZEPIN-6-ONE MOIETY - STRUCTURAL REQUIREMENTS FOR OPTIMUM OCCUPANCY OF MUSCARINIC RECEPTOR SUBTYPES AS REVEALED BY SYMMETRICAL AND UNSYMMETRICAL POLYAMINES, Journal of medicinal chemistry, 37(20), 1994, pp. 3363-3372
Authors:
TETTAMANTI G
DIFRANCESCO L
CHIARINI A
FIORILLI A
MONTI E
ZIZIOLI D
VENERANDO B
Citation: G. Tettamanti et al., BRAIN CYTOSOLIC SIALIDASE - A PROTEIN COMPLEX CONTAINING A CATALYTIC AND A PROTECTIVE UNIT, Glycoconjugate journal, 10(4), 1993, pp. 294-294
Authors:
CHIARINI A
FIORILLI A
DIFRANCESCO L
VENERANDO B
TETTAMANTI G
Citation: A. Chiarini et al., HUMAN ERYTHROCYTE SIALIDASE IS LINKED TO THE PLASMA-MEMBRANE BY A GLYCOSYLPHOSPHATIDYLINOSITOL ANCHOR AND PARTLY LOCATED ON THE OUTER SURFACE, Glycoconjugate journal, 10(1), 1993, pp. 64-71
Authors:
MELCHIORRE C
BOLOGNESI ML
CHIARINI A
MINARINI A
SPAMPINATO S
Citation: C. Melchiorre et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME METHOCTRAMINE-RELATED TETRAAMINES BEARING A -DIHYDRO-6H-PYRIDO[2,3-B][1,4]-BENZODIAZEPIN-6-ONE MOIETY AS ANTIMUSCARINICS - A 2ND-GENERATION OF HIGHLY SELECTIVE M(2)-MUSCARINIC RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(23), 1993, pp. 3734-3737