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Results: 1-11 |
Results: 11
CONFORMATIONALLY CONSTRAINED 1,3-DIAMINO KETONES - A SERIES OF POTENTINHIBITORS OF THE CYSTEINE PROTEASE CATHEPSIN-K
Authors: MARQUIS RW YAMASHITA DS RU Y LOCASTRO SM OH HJ ERHARD KF DESJARLAIS RL HEAD MS SMITH WW ZHAO BG JANSON CA ABDELMEGUID SS TOMASZEK TA LEVY MA VEBER DF
Citation: Rw. Marquis et al., CONFORMATIONALLY CONSTRAINED 1,3-DIAMINO KETONES - A SERIES OF POTENTINHIBITORS OF THE CYSTEINE PROTEASE CATHEPSIN-K, Journal of medicinal chemistry, 41(19), 1998, pp. 3563-3567
USE OF X-RAY CO-CRYSTAL STRUCTURES AND MOLECULAR MODELING TO DESIGN POTENT AND SELECTIVE NONPEPTIDE INHIBITORS OF CATHEPSIN-K
Authors: DESJARLAIS RL YAMASHITA DS OH HJ UZINSKAS IN ERHARD KF ALLEN AC HALTIWANGER RC ZHAO BG SMITH WW ABDELMEGUID SS DALESSIO K JANSON CA MCQUENEY MS TOMASZEK TA LEVY MA VEBER DF
Citation: Rl. Desjarlais et al., USE OF X-RAY CO-CRYSTAL STRUCTURES AND MOLECULAR MODELING TO DESIGN POTENT AND SELECTIVE NONPEPTIDE INHIBITORS OF CATHEPSIN-K, Journal of the American Chemical Society, 120(35), 1998, pp. 9114-9115
AN ALTERNATE ENANTIOSPECIFIC SYNTHESIS OF METHYL DRO-4-METHYL-3-OXO-1H-1,4-BENZODIAZEPINE-2-ACETATE
Authors: KU TW ALI FE BONDINELL WE ERHARD KF HUFFMAN WF VENSLAVSKY JW YUAN CCK
Citation: Tw. Ku et al., AN ALTERNATE ENANTIOSPECIFIC SYNTHESIS OF METHYL DRO-4-METHYL-3-OXO-1H-1,4-BENZODIAZEPINE-2-ACETATE, Tetrahedron letters, 38(18), 1997, pp. 3131-3134
ENANTIOSPECIFIC SYNTHESIS OF SB-214857, A POTENT, ORALLY-ACTIVE, NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONIST
Authors: MILLER WH KU TW ALI FE BONDINELL WE CALVO RR DAVIS LD ERHARD KF HALL LB HUFFMAN WF KEENAN RM KWON C NEWLANDER KA ROSS ST SAMANEN JM TAKATA DT YUAN CK
Citation: Wh. Miller et al., ENANTIOSPECIFIC SYNTHESIS OF SB-214857, A POTENT, ORALLY-ACTIVE, NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONIST, Tetrahedron letters, 36(52), 1995, pp. 9433-9436
POTENT NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS WHICH PRESENT AN ALTERNATIVE PHARMACOPHORE
Authors: KU TW MILLER WH BONDINELL WE ERHARD KF KEENAN RM NICHOLS AJ PEISHOFF CE SAMANEN JM WONG AS HUFFMAN WF
Citation: Tw. Ku et al., POTENT NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS WHICH PRESENT AN ALTERNATIVE PHARMACOPHORE, Journal of medicinal chemistry, 38(1), 1995, pp. 9-12
STRUCTURE-ACTIVITY STUDIES OF SYNTHETIC FKBP LIGANDS AS PEPTIDYL-PROLYL ISOMERASE INHIBITORS
Authors: HOLT DA KONIALIANBECK AL OH HJ YEN HK ROZAMUS LW KROG AJ ERHARD KF ORTIZ E LEVY MA BRANDT M BOSSARD MJ LUENGO JI
Citation: Da. Holt et al., STRUCTURE-ACTIVITY STUDIES OF SYNTHETIC FKBP LIGANDS AS PEPTIDYL-PROLYL ISOMERASE INHIBITORS, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 315-320
PREPARATIVE CHIRAL HPLC SEPARATION OF ALL POSSIBLE STEREOISOMERS OF LY191704 AND LY266111 AND THEIR IN-VITRO INHIBITION OF HUMAN TYPE-1 ANDTYPE-2 STEROID 5-ALPHA-REDUCTASES
Authors: ABELL AD ERHARD KF YEN HK YAMASHITA DS BRANDT M MOHAMMED H LEVY MA HOLT DA
Citation: Ad. Abell et al., PREPARATIVE CHIRAL HPLC SEPARATION OF ALL POSSIBLE STEREOISOMERS OF LY191704 AND LY266111 AND THEIR IN-VITRO INHIBITION OF HUMAN TYPE-1 ANDTYPE-2 STEROID 5-ALPHA-REDUCTASES, Bioorganic & medicinal chemistry letters, 4(11), 1994, pp. 1365-1368
PRETREATMENT OF CHIRAL ALPHA-AGP COLUMN WITH TRIETHYLAMINE SIGNIFICANTLY IMPROVES THE DETECTION SENSITIVITY OF AN ENANTIOMERIC LEUKOTRIENE ANTAGONIST
Authors: HO MYK ERHARD KF CHEN TK
Citation: Myk. Ho et al., PRETREATMENT OF CHIRAL ALPHA-AGP COLUMN WITH TRIETHYLAMINE SIGNIFICANTLY IMPROVES THE DETECTION SENSITIVITY OF AN ENANTIOMERIC LEUKOTRIENE ANTAGONIST, Journal of liquid chromatography, 17(4), 1994, pp. 761-772
1,3-DIARYLINDAN-2-CARBOXYLIC ACIDS, POTENT AND SELECTIVE NONPEPTIDE ENDOTHELIN RECEPTOR ANTAGONISTS
Authors: ELLIOTT JD LAGO MA COUSINS RD GAO AM LEBER JD ERHARD KF NAMBI P ELSHOURBAGY NA KUMAR C LEE JA BEAN JW DEBROSSE CW EGGLESTON DS BROOKS DP FEUERSTEIN G RUFFOLO RR WEINSTOCK J GLEASON JG PEISHOFF CE OHLSTEIN EH
Citation: Jd. Elliott et al., 1,3-DIARYLINDAN-2-CARBOXYLIC ACIDS, POTENT AND SELECTIVE NONPEPTIDE ENDOTHELIN RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 37(11), 1994, pp. 1553-1557
RESOLUTION OF HYDROXYUREAS
Authors: GARIGIPATI RS SORENSON ME ERHARD KF ADAMS JL
Citation: Rs. Garigipati et al., RESOLUTION OF HYDROXYUREAS, Tetrahedron letters, 34(35), 1993, pp. 5537-5540
THE CRYSTAL-STRUCTURE, ABSOLUTE-CONFIGURATION, AND PHOSPHODIESTERASE INHIBITORY ACTIVITY OF CLOPENTYLOXY)-4-METHOXYPHENYL)-PYRROLIDIN-2-ONE())
Authors: BAURES PW EGGLESTON DS ERHARD KF CIESLINSKI LB TORPHY TJ CHRISTENSEN SB
Citation: Pw. Baures et al., THE CRYSTAL-STRUCTURE, ABSOLUTE-CONFIGURATION, AND PHOSPHODIESTERASE INHIBITORY ACTIVITY OF CLOPENTYLOXY)-4-METHOXYPHENYL)-PYRROLIDIN-2-ONE()), Journal of medicinal chemistry, 36(22), 1993, pp. 3274-3277
Risultati: 1-11 |