Authors:
TRAIL PA
WILLNER D
KNIPE J
HENDERSON AJ
LASCH SJ
ZOECKLER ME
TRAILSMITH MD
DOYLE TW
KING HD
CASAZZA AM
BRASLAWSKY GR
BROWN J
HOFSTEAD SJ
GREENFIELD RS
FIRESTONE RA
MOSURE K
KADOW KF
YANG MB
HELLSTROM KE
HELLSTROM I
Citation: Pa. Trail et al., EFFECT OF LINKER VARIATION ON THE STABILITY, POTENCY, AND EFFICACY OFCARCINOMA-REACTIVE BR64-DOXORUBICIN IMMUNOCONJUGATES, Cancer research, 57(1), 1997, pp. 100-105
Citation: V. Farina et al., SYNTHESIS OF CEPHEMS BEARING OLEFINIC SULFOXIDE SIDE-CHAINS AS POTENTIAL BETA-LACTAMASE INHIBITORS, Bioorganic & medicinal chemistry letters, 6(13), 1996, pp. 1613-1618
Authors:
FIRESTONE RA
WILLNER D
HOFSTEAD SJ
KING HD
KANEKO T
BRASLAWSKY GR
GREENFIELD RS
TRAIL PA
LASCH SJ
HENDERSON AJ
CASAZZA AM
HELLSTROM I
Citation: Ra. Firestone et al., SYNTHESIS AND ANTITUMOR-ACTIVITY OF THE IMMUNOCONJUGATE BR96-DOX, Journal of controlled release, 39(2-3), 1996, pp. 251-259
Citation: Gm. Dubowchik et Ra. Firestone, A LIPOPHILIC POLYAMINO-BOLAAMPHIPHILE DESIGNED TO DISSIPATE PH GRADIENTS ACROSS A BILAYER-MEMBRANE - SYNTHESIS AND PROTON TRANSPORT, Tetrahedron letters, 37(36), 1996, pp. 6465-6468
Authors:
DUBOWCHIK GM
PADILLA L
EDINGER K
FIRESTONE RA
Citation: Gm. Dubowchik et al., AMINES THAT TRANSPORT PROTONS ACROSS BILAYER-MEMBRANES - SYNTHESIS, LYSOSOMAL NEUTRALIZATION, AND 2-PHASE PK(A) VALUES BY NMR, Journal of organic chemistry, 61(14), 1996, pp. 4676-4684
Citation: Gm. Dubowchik et Ra. Firestone, IMPROVED CYTOTOXICITY OF ANTITUMOR COMPOUNDS DELIVERABLE BY THE LDL PATHWAY, Bioconjugate chemistry, 6(4), 1995, pp. 427-439
Citation: Gm. Dubowchik et al., THE IN-VITRO EFFECTS OF 3 LYSOSOMOTROPIC DETERGENTS AGAINST 3 HUMAN TUMOR-CELL LINES, Bioorganic & medicinal chemistry letters, 5(8), 1995, pp. 893-898
Citation: Ra. Firestone, LOW-DENSITY-LIPOPROTEIN AS A VEHICLE FOR TARGETING ANTITUMOR COMPOUNDS TO CANCER-CELLS, Bioconjugate chemistry, 5(2), 1994, pp. 105-113
Authors:
MAMBER SW
BROOKSHIRE KW
DEAN BJ
FIRESTONE RA
LEET JE
MATSON JA
FORENZA S
Citation: Sw. Mamber et al., INHIBITION OF ANTIBACTERIAL ACTIVITY OF HIMASTATIN, A NEW ANTITUMOR ANTIBIOTIC FROM STREPTOMYCES-HYGROSCOPICUS, BY FATTY-ACID SODIUM-SALTS, Antimicrobial agents and chemotherapy, 38(11), 1994, pp. 2633-2642
Authors:
MAMBER SW
BROOKSHIRE KW
DEAN BJ
FIRESTONE RA
LEET JE
MATSON JA
FORENZA S
Citation: Sw. Mamber et al., INHIBITION OF ANTIBACTERIAL ACTIVITY OF HIMASTATIN, A NEW ANTITUMOR ANTIBIOTIC FROM STREPTOMYCES-HYGROSCOPICUS, BY FATTY-ACID SODIUM-SALTS, Antimicrobial agents and chemotherapy, 38(11), 1994, pp. 2633-2642
Citation: Gm. Dubowchik et Ra. Firestone, THE SYNTHESIS OF BRANCHED STEROIDAL PRODRUGS OF NITROGEN-MUSTARD FOR ANTITUMOR TARGETING VIA RECONSTITUTED LDL, Tetrahedron letters, 35(26), 1994, pp. 4523-4526
Citation: Ta. Montzka et al., REVERSAL OF SYN-ANTI PREFERENCE FOR CARBOXYLIC-ACIDS ALONG THE REACTION COORDINATE FOR PROTON-TRANSFER - IMPLICATIONS FOR INTRAMOLECULAR CATALYSIS, Journal of physical chemistry, 98(50), 1994, pp. 13171-13176
Citation: Ra. Firestone, LEAST-MOTION STEPWISE [2-CYCLOADDUCTS(2] KETENE CYCLOADDITION PATHWAYS PREDICT THE MORE HINDERED CIS), International journal of quantum chemistry, 49(1), 1994, pp. 21-24
Authors:
DUBOWCHIK GM
PADILLA L
EDINGER K
FIRESTONE RA
Citation: Gm. Dubowchik et al., REVERSAL OF DOXORUBICIN RESISTANCE AND CATALYTIC NEUTRALIZATION OF LYSOSOMES BY A LIPOPHILIC IMIDAZOLE, Biochimica et biophysica acta. Biomembranes, 1191(1), 1994, pp. 103-108
Authors:
WILLNER D
TRAIL PA
HOFSTEAD SJ
KING HD
LASCH SJ
BRASLAWSKY GR
GREENFIELD RS
KANEKO T
FIRESTONE RA
Citation: D. Willner et al., (6-MALEIMIDOCAPROYL)HYDRAZONE OF DOXORUBICIN - A NEW DERIVATIVE FOR THE PREPARATION OF IMMUNOCONJUGATES OF DOXORUBICIN, Bioconjugate chemistry, 4(6), 1993, pp. 521-527
Citation: Gm. Dubowchik et al., AN ACID-CLEAVABLE LINKER STABLE AT NEUTRAL PH THAT RELEASES DOXORUBICIN AT LYSOSOMAL PH, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2843-2846