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Results: 1-14 |
Results: 14
POTENT AND SPECIFIC-INHIBITION OF HUMAN-LEUKOCYTE ELASTASE, CATHEPSIN-G AND PROTEINASE-3 BY SULFONE DERIVATIVES EMPLOYING THE 1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE SCAFFOLD
Authors: GROUTAS WC KUANG RZ RUAN SM EPP JB VENKATARAMAN R TRUONG TM
Citation: Wc. Groutas et al., POTENT AND SPECIFIC-INHIBITION OF HUMAN-LEUKOCYTE ELASTASE, CATHEPSIN-G AND PROTEINASE-3 BY SULFONE DERIVATIVES EMPLOYING THE 1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE SCAFFOLD, Bioorganic & medicinal chemistry, 6(6), 1998, pp. 661-671
USE OF THE 1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE AND ISOTHIAZOLIDIN-3-ONE 1,1-DIOXIDE SCAFFOLDS IN THE DESIGN OF POTENT INHIBITORS OF SERINE PROTEINASES
Authors: KUANG RZ VENKATARAMAN R RUAN SM GROUTAS WC
Citation: Rz. Kuang et al., USE OF THE 1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE AND ISOTHIAZOLIDIN-3-ONE 1,1-DIOXIDE SCAFFOLDS IN THE DESIGN OF POTENT INHIBITORS OF SERINE PROTEINASES, Bioorganic & medicinal chemistry letters, 8(5), 1998, pp. 539-544
INHIBITION OF NEUROTOXIC ESTERASE IN-VITRO BY NOVEL CARBAMATES
Authors: RANDALL JC AMBROSO JL GROUTAS WC BRUBAKER MJ RICHARDSON RJ
Citation: Jc. Randall et al., INHIBITION OF NEUROTOXIC ESTERASE IN-VITRO BY NOVEL CARBAMATES, Toxicology and applied pharmacology, 143(1), 1997, pp. 173-178
STRUCTURE-BASED DESIGN OF A GENERAL-CLASS OF MECHANISM-BASED INHIBITORS OF THE SERINE PROTEINASES EMPLOYING A NOVEL AMINO ACID-DERIVED HETEROCYCLIC SCAFFOLD
Authors: GROUTAS WC KUANG RZ VENKATARAMAN R EPP JB RUAN SM PRAKASH O
Citation: Wc. Groutas et al., STRUCTURE-BASED DESIGN OF A GENERAL-CLASS OF MECHANISM-BASED INHIBITORS OF THE SERINE PROTEINASES EMPLOYING A NOVEL AMINO ACID-DERIVED HETEROCYCLIC SCAFFOLD, Biochemistry, 36(16), 1997, pp. 4739-4750
INHIBITION OF HUMAN-LEUKOCYTE PROTEINASE-3 BY A NOVEL RECOMBINANT SERINE PROTEINASE-INHIBITOR (LEX032)
Authors: GROUTAS WC RUAN SM KUANG RZ HOOK JB SANDS H
Citation: Wc. Groutas et al., INHIBITION OF HUMAN-LEUKOCYTE PROTEINASE-3 BY A NOVEL RECOMBINANT SERINE PROTEINASE-INHIBITOR (LEX032), Biochemical and biophysical research communications, 233(3), 1997, pp. 697-699
AMINO ACID-DERIVED PHTHALIMIDE AND SACCHARIN DERIVATIVES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, CATHEPSIN-G, AND PROTEINASE-3
Authors: GROUTAS WC CHONG LS VENKATARAMAN R KUANG R EPP JB HOUSERARCHIELD N HUANG H HOIDAL JR
Citation: Wc. Groutas et al., AMINO ACID-DERIVED PHTHALIMIDE AND SACCHARIN DERIVATIVES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, CATHEPSIN-G, AND PROTEINASE-3, Archives of biochemistry and biophysics, 332(2), 1996, pp. 335-340
MECHANISM-BASED INHIBITION OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G BY SUBSTITUTED DIHYDROURACILS
Authors: GROUTAS WC HUANG H EPP JB VENKATARAMAN R MCCLENAHAN JJ TAGUSAGAWA F
Citation: Wc. Groutas et al., MECHANISM-BASED INHIBITION OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G BY SUBSTITUTED DIHYDROURACILS, Biochimica et biophysica acta. Molecular basis of disease, 1227(3), 1994, pp. 130-136
SUBSTITUTED 3-OXO-1,25-THIADIAZOLIDINE 1,1-DIOXIDES - A NEW CLASS OF POTENTIAL MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G
Authors: GROUTAS WC KUANG RZ VENKATARAMAN R
Citation: Wc. Groutas et al., SUBSTITUTED 3-OXO-1,25-THIADIAZOLIDINE 1,1-DIOXIDES - A NEW CLASS OF POTENTIAL MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G, Biochemical and biophysical research communications, 198(1), 1994, pp. 341-349
HETEROCYCLIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE - 3-HYDROXYPYRIDAZOPYRIMIDINE, 3-HYDROXYPYRIDOPYRIMIDINE AND 3-HYDROXYQUINAZOLINE-2,4(1H,3H)DIONE DERIVATIVES
Authors: GROUTAS WC CASTRISOS JC STANGA MA KUANG RZ VENKATARAMAN R EPP JB BRUBAKER MJ CHONG LS
Citation: Wc. Groutas et al., HETEROCYCLIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE - 3-HYDROXYPYRIDAZOPYRIMIDINE, 3-HYDROXYPYRIDOPYRIMIDINE AND 3-HYDROXYQUINAZOLINE-2,4(1H,3H)DIONE DERIVATIVES, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 1163-1168
A GENERAL-APPROACH TOWARD THE DESIGN OF MECHANISM-BASED INACTIVATORS OF SERINE PROTEINASES - INACTIVATION OF HUMAN-LEUKOCYTE ELASTASE BY A PHTHALIMIDE DERIVATIVE
Authors: GROUTAS WC CHONG LS VENKATARAMAN R HUANG H EPP JB KUANG RZ
Citation: Wc. Groutas et al., A GENERAL-APPROACH TOWARD THE DESIGN OF MECHANISM-BASED INACTIVATORS OF SERINE PROTEINASES - INACTIVATION OF HUMAN-LEUKOCYTE ELASTASE BY A PHTHALIMIDE DERIVATIVE, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2745-2750
EFFICIENT INHIBITION OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G BY SACCHARIN DERIVATIVES
Authors: GROUTAS WC HOUSERARCHIELD N CHONG LS VENKATARAMAN R EPP JB HUANG H MCCLENAHAN JJ
Citation: Wc. Groutas et al., EFFICIENT INHIBITION OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G BY SACCHARIN DERIVATIVES, Journal of medicinal chemistry, 36(21), 1993, pp. 3178-3181
3-(ALKYLTHIO)-N-HYDROXYSUCCINIMIDE DERIVATIVES - POTENT INHIBITORS OFHUMAN-LEUKOCYTE ELASTASE
Authors: GROUTAS WC VENKATARAMAN R BRUBAKER MJ EPP JB CHONG LS STANGA MA MCCLENAHAN JJ TAGUSAGAWA F
Citation: Wc. Groutas et al., 3-(ALKYLTHIO)-N-HYDROXYSUCCINIMIDE DERIVATIVES - POTENT INHIBITORS OFHUMAN-LEUKOCYTE ELASTASE, Biochimica et biophysica acta, 1164(3), 1993, pp. 283-288
NOVEL POTENTIAL MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G - DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE
Authors: GROUTAS WC CHONG LS VENKATARAMAN R
Citation: Wc. Groutas et al., NOVEL POTENTIAL MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G - DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE, Biochemical and biophysical research communications, 197(2), 1993, pp. 730-739
MECHANISM-BASED INHIBITORS OF SERINE PROTEINASES BASED ON THE GABRIEL-COLMAN REARRANGEMENT
Authors: GROUTAS WC CHONG LS VENKATARAMAN R EPP JB KUANG RZ BRUBAKER MJ HOUSERARCHIELD N HUANG H MCCLENAHAN JJ
Citation: Wc. Groutas et al., MECHANISM-BASED INHIBITORS OF SERINE PROTEINASES BASED ON THE GABRIEL-COLMAN REARRANGEMENT, Biochemical and biophysical research communications, 194(3), 1993, pp. 1491-1499
Risultati: 1-14 |