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Results: 1-25 | 26-50 | 51-70
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CRYSTAL-STRUCTURE AND QUANTUM-CHEMICAL AB-INITIO CALCULATIONS OF IBOTENIC ACID, AN EXCITATORY AMINO-ACID RECEPTOR AGONIST
Authors: BREHM L FRYDENVANG K KROGSGAARDLARSEN P LILJEFORS T
Citation: L. Brehm et al., CRYSTAL-STRUCTURE AND QUANTUM-CHEMICAL AB-INITIO CALCULATIONS OF IBOTENIC ACID, AN EXCITATORY AMINO-ACID RECEPTOR AGONIST, Structural chemistry, 9(2), 1998, pp. 149-155
ARYL AND CYCLOALKYL ANALOGS OF AMPA - SYNTHETIC, PHARMACOLOGICAL AND STEREOCHEMICAL ASPECTS
Authors: SKJAERBAEK N BREHM L JOHANSEN TN HANSEN LM NIELSEN B EBERT B SOBY KK STENSBOL TB FALCH E KROGSGAARDLARSEN P
Citation: N. Skjaerbaek et al., ARYL AND CYCLOALKYL ANALOGS OF AMPA - SYNTHETIC, PHARMACOLOGICAL AND STEREOCHEMICAL ASPECTS, Bioorganic & medicinal chemistry, 6(1), 1998, pp. 119-131
SYNTHESES OF NOVEL PIPERIDIN-4-YLPHOSPHINIC ACID, AND PIPERIDIN-4-YLPHOSPHONIC ACID ANALOGS OF THE INHIBITORY NEUROTRANSMITTER 4-AMINOBUTYRIC ACID (GABA)
Authors: KEHLER J EBERT B DAHL O KROGSGAARDLARSEN P
Citation: J. Kehler et al., SYNTHESES OF NOVEL PIPERIDIN-4-YLPHOSPHINIC ACID, AND PIPERIDIN-4-YLPHOSPHONIC ACID ANALOGS OF THE INHIBITORY NEUROTRANSMITTER 4-AMINOBUTYRIC ACID (GABA), Journal of the Chemical Society. Perkin transactions. I (Print), (19), 1998, pp. 3241-3243
UNAMBIGUOUS SYNTHESIS OF 1-METHYL-3-HYDROXYPYRAZOLES
Authors: ZIMMERMANN D KROGSGAARDLARSEN P EHRHARDT JD MADSEN U JANIN YL
Citation: D. Zimmermann et al., UNAMBIGUOUS SYNTHESIS OF 1-METHYL-3-HYDROXYPYRAZOLES, Tetrahedron, 54(32), 1998, pp. 9393-9400
PHARMACOLOGY AND TOXICOLOGY OF ATOA, AN AMPA RECEPTOR ANTAGONIST AND A PARTIAL AGONIST AT GLUR5 RECEPTORS
Authors: WAHL P FRANDSEN A MADSEN U SCHOUSBOE A KROGSGAARDLARSEN P
Citation: P. Wahl et al., PHARMACOLOGY AND TOXICOLOGY OF ATOA, AN AMPA RECEPTOR ANTAGONIST AND A PARTIAL AGONIST AT GLUR5 RECEPTORS, Neuropharmacology, 37(10-11), 1998, pp. 1205-1210
ANTAGONIST PROPERTIES OF A PHOSPHONO ISOXAZOLE AMINO-ACID AT GLUTAMATE R1-4 AMINO-3-(3-HYDROXY-5-METHYL-4-ISOXAZOLYL)PROPIONIC ACID RECEPTOR SUBTYPES
Authors: WAHL P ANKER C TRAYNELIS SF EGEBJERG J RASMUSSEN JS KROGSGAARDLARSEN P MADSEN U
Citation: P. Wahl et al., ANTAGONIST PROPERTIES OF A PHOSPHONO ISOXAZOLE AMINO-ACID AT GLUTAMATE R1-4 AMINO-3-(3-HYDROXY-5-METHYL-4-ISOXAZOLYL)PROPIONIC ACID RECEPTOR SUBTYPES, Molecular pharmacology, 53(3), 1998, pp. 590-596
EXCITATORY AMINO-ACID RECEPTOR LIGANDS - RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND ENANTIOPHARMACOLOGY OF -AMINO-3-(4-BUTYL-3-HYDROXYISOXAZOL-5-YL)PROPIONIC ACID
Authors: JOHANSEN TN EBERT B BRAUNEROSBORNE H DIDRIKSEN M CHRISTENSEN IT SOBY KK MADSEN U KROGSGAARDLARSEN P BREHM L
Citation: Tn. Johansen et al., EXCITATORY AMINO-ACID RECEPTOR LIGANDS - RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND ENANTIOPHARMACOLOGY OF -AMINO-3-(4-BUTYL-3-HYDROXYISOXAZOL-5-YL)PROPIONIC ACID, Journal of medicinal chemistry, 41(6), 1998, pp. 930-939
HETEROARYL ANALOGS OF AMPA - 2 - SYNTHESIS, ABSOLUTE STEREOCHEMISTRY,PHOTOCHEMISTRY, AND STRUCTURE-ACTIVITY-RELATIONSHIPS
Authors: FALCH E BREHM L MIKKELSEN I JOHANSEN TN SKJAERBAEK N NIELSEN B STENSBOL TB EBERT B KROGSGAARDLARSEN P
Citation: E. Falch et al., HETEROARYL ANALOGS OF AMPA - 2 - SYNTHESIS, ABSOLUTE STEREOCHEMISTRY,PHOTOCHEMISTRY, AND STRUCTURE-ACTIVITY-RELATIONSHIPS, Journal of medicinal chemistry, 41(14), 1998, pp. 2513-2523
MOLECULAR PHARMACOLOGY OF HOMOLOGS OF IBOTENIC ACID AT CLONED METABOTROPIC GLUTAMIC-ACID RECEPTORS
Authors: BRAUNEROSBORNE H NIELSEN B KROGSGAARDLARSEN P
Citation: H. Braunerosborne et al., MOLECULAR PHARMACOLOGY OF HOMOLOGS OF IBOTENIC ACID AT CLONED METABOTROPIC GLUTAMIC-ACID RECEPTORS, European journal of pharmacology, 350(2-3), 1998, pp. 311-316
PHARMACOLOGY OF (S)-HOMOQUISQUALIC ACID AND (S)-2-AMINO-5-PHOSPHONOPENTANOIC ACID [(S)-AP5] AT CLONED METABOTROPIC GLUTAMATE RECEPTORS
Authors: BRAUNEROSBORNE H KROGSGAARDLARSEN P
Citation: H. Braunerosborne et P. Krogsgaardlarsen, PHARMACOLOGY OF (S)-HOMOQUISQUALIC ACID AND (S)-2-AMINO-5-PHOSPHONOPENTANOIC ACID [(S)-AP5] AT CLONED METABOTROPIC GLUTAMATE RECEPTORS, British Journal of Pharmacology, 123(2), 1998, pp. 269-274
STRUCTURAL FEATURES OF MUSCIMOL, A POTENT GABA(A) RECEPTOR AGONIST, CRYSTAL-STRUCTURE AND QUANTUM-CHEMICAL AB-INITIO CALCULATIONS
Authors: BREHM L FRYDENVANG K HANSEN LM NORRBY PO KROGSGAARDLARSEN P LILJEFORS T
Citation: L. Brehm et al., STRUCTURAL FEATURES OF MUSCIMOL, A POTENT GABA(A) RECEPTOR AGONIST, CRYSTAL-STRUCTURE AND QUANTUM-CHEMICAL AB-INITIO CALCULATIONS, Structural chemistry, 8(6), 1997, pp. 443-451
BIOISOSTERICALLY MODIFIED DIPEPTIDE EXCITATORY AMINO-ACID RECEPTOR ANTAGONISTS CONTAINING 3-OXYGENATED ISOTHIAZOLE RING-SYSTEMS
Authors: MATZEN L EBERT B STENSBOL TB FROLUND B JAROSZEWSKI JW KROGSGAARDLARSEN P
Citation: L. Matzen et al., BIOISOSTERICALLY MODIFIED DIPEPTIDE EXCITATORY AMINO-ACID RECEPTOR ANTAGONISTS CONTAINING 3-OXYGENATED ISOTHIAZOLE RING-SYSTEMS, Bioorganic & medicinal chemistry, 5(8), 1997, pp. 1569-1575
GABA(A) AND GABA(B) RECEPTOR AGONISTS, PARTIAL AGONISTS, ANTAGONISTS AND MODULATORS - DESIGN AND THERAPEUTIC PROSPECTS
Authors: KROGSGAARDLARSEN P FROLUND B KRISTIANSEN U FRYDENVANG K EBERT B
Citation: P. Krogsgaardlarsen et al., GABA(A) AND GABA(B) RECEPTOR AGONISTS, PARTIAL AGONISTS, ANTAGONISTS AND MODULATORS - DESIGN AND THERAPEUTIC PROSPECTS, European journal of pharmaceutical sciences, 5(6), 1997, pp. 355-384
EXCITATORY AMINO-ACID RECEPTOR ANTAGONISTS - RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND PHARMACOLOGY OF MINO-2-(5-TERT-BUTYL-3-HYDROXYISOXAZOL-4-YL)ACETIC AND MINO-2-(5-TERT-BUTYL-3-HYDROXYISOXAZOL-4-YL)ACETIC ACID (ATAA)
Authors: JOHANSEN TN FRYDENVANG K EBERT B MADSEN U KROGSGAARDLARSEN P
Citation: Tn. Johansen et al., EXCITATORY AMINO-ACID RECEPTOR ANTAGONISTS - RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND PHARMACOLOGY OF MINO-2-(5-TERT-BUTYL-3-HYDROXYISOXAZOL-4-YL)ACETIC AND MINO-2-(5-TERT-BUTYL-3-HYDROXYISOXAZOL-4-YL)ACETIC ACID (ATAA), Chirality, 9(5-6), 1997, pp. 529-536
AMPA-RECEPTOR AGONISTS - RESOLUTION, CONFIGURATIONAL ASSIGNMENT, AND PHARMACOLOGY OF 3-[3-HYDROXY-5-(2-PYRIDYL)ISOXAZOL-4-YL]-PROPIONIC AND3-[3-HYDROXY-5-(2-PYRIDYL)ISOXAZOL-4-YL]-PROPIONIC ACID (2-PY-AMPA)())
Authors: JOHANSEN TN EBERT B FALCH E KROGSGAARDLARSEN P
Citation: Tn. Johansen et al., AMPA-RECEPTOR AGONISTS - RESOLUTION, CONFIGURATIONAL ASSIGNMENT, AND PHARMACOLOGY OF 3-[3-HYDROXY-5-(2-PYRIDYL)ISOXAZOL-4-YL]-PROPIONIC AND3-[3-HYDROXY-5-(2-PYRIDYL)ISOXAZOL-4-YL]-PROPIONIC ACID (2-PY-AMPA)()), Chirality, 9(3), 1997, pp. 274-280
STRUCTURAL CHARACTERISTICS OF ISOXAZOL-3-OL AND ISOTHIAZOL-3-OL, CARBOXY GROUP BIOISOSTERES EXAMINED BY X-RAY CRYSTALLOGRAPHY AND AB-INITIOCALCULATIONS
Authors: FRYDENVANG K MATZEN L NORRBY PO SLOK FA LILJEFORS T KROGSGAARDLARSEN P JAROSZEWSKI JW
Citation: K. Frydenvang et al., STRUCTURAL CHARACTERISTICS OF ISOXAZOL-3-OL AND ISOTHIAZOL-3-OL, CARBOXY GROUP BIOISOSTERES EXAMINED BY X-RAY CRYSTALLOGRAPHY AND AB-INITIOCALCULATIONS, Perkin transactions. 2, (9), 1997, pp. 1783-1791
EXCITATORY AMINO-ACID RECEPTOR AGONISTS - SYNTHESIS AND PHARMACOLOGY OF ANALOGS OF AMINO-3-(3-HYDROXY-5-METHYLISOXAZOL-4-YL)PROPIONIC ACID
Authors: SLOK FA EBERT B LANG Y KROGSGAARDLARSEN P LENZ SM MADSEN U
Citation: Fa. Slok et al., EXCITATORY AMINO-ACID RECEPTOR AGONISTS - SYNTHESIS AND PHARMACOLOGY OF ANALOGS OF AMINO-3-(3-HYDROXY-5-METHYLISOXAZOL-4-YL)PROPIONIC ACID, European journal of medicinal chemistry, 32(4), 1997, pp. 329-338
STRUCTURE AND PHARMACOLOGY OF 4,5,6,7-TETRAHYDROISOTHIAZOLO[5,4-C]PYRIDIN-3-OL (THIO-THIP), AN AGONIST ANTAGONIST AT GABA(A) RECEPTORS/
Authors: BREHM L EBERT B KRISTIANSEN U WAFFORD KA KEMP JA KROGSGAARDLARSEN P
Citation: L. Brehm et al., STRUCTURE AND PHARMACOLOGY OF 4,5,6,7-TETRAHYDROISOTHIAZOLO[5,4-C]PYRIDIN-3-OL (THIO-THIP), AN AGONIST ANTAGONIST AT GABA(A) RECEPTORS/, European journal of medicinal chemistry, 32(4), 1997, pp. 357-363
(-)-(R)-5,5-DIMETHYLMORPHOLINYL-2-ACETIC ACID ETHYL-ESTER HYDROCHLORIDE, C10H20NO3-(.CL)
Authors: FRYDENVANG K ENNA SJ KROGSGAARDLARSEN P
Citation: K. Frydenvang et al., (-)-(R)-5,5-DIMETHYLMORPHOLINYL-2-ACETIC ACID ETHYL-ESTER HYDROCHLORIDE, C10H20NO3-(.CL), Acta crystallographica. Section C, Crystal structure communications, 53, 1997, pp. 1088-1091
DIFFERENCES IN AGONIST ANTAGONIST BINDING-AFFINITY AND RECEPTOR TRANSDUCTION USING RECOMBINANT HUMAN GAMMA-AMINOBUTYRIC-ACID TYPE-A RECEPTORS/
Authors: EBERT B THOMPSON SA SAOUNATSOU K MCKERNAN R KROGSGAARDLARSEN P WAFFORD KA
Citation: B. Ebert et al., DIFFERENCES IN AGONIST ANTAGONIST BINDING-AFFINITY AND RECEPTOR TRANSDUCTION USING RECOMBINANT HUMAN GAMMA-AMINOBUTYRIC-ACID TYPE-A RECEPTORS/, Molecular pharmacology, 52(6), 1997, pp. 1150-1156
AMPA RECEPTOR AGONISTS - SYNTHESIS, PROTOLYTIC PROPERTIES, AND PHARMACOLOGY OF 3-ISOTHIAZOLOL BIOISOSTERES OF GLUTAMIC-ACID
Authors: MATZEN L ENGESGAARD A EBERT B DIDRIKSEN M FROLUND B KROGSGAARDLARSEN P JAROSZEWSKI JW
Citation: L. Matzen et al., AMPA RECEPTOR AGONISTS - SYNTHESIS, PROTOLYTIC PROPERTIES, AND PHARMACOLOGY OF 3-ISOTHIAZOLOL BIOISOSTERES OF GLUTAMIC-ACID, Journal of medicinal chemistry, 40(4), 1997, pp. 520-527
(S)-HOMO-AMPA, A SPECIFIC AGONIST AT THE MGLU(6) SUBTYPE OF METABOTROPIC GLUTAMIC-ACID RECEPTORS
Authors: AHMADIAN H NIELSEN B BRAUNEROSBORNE H JOHANSEN TN STENSBOL TB SLOK FA SEKIYAMA N NAKANISHI S KROGSGAARDLARSEN P MADSEN U
Citation: H. Ahmadian et al., (S)-HOMO-AMPA, A SPECIFIC AGONIST AT THE MGLU(6) SUBTYPE OF METABOTROPIC GLUTAMIC-ACID RECEPTORS, Journal of medicinal chemistry, 40(22), 1997, pp. 3700-3705
HETEROARYL ANALOGS OF AMPA - SYNTHESIS AND QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS
Authors: BANGANDERSEN B LENZ SM SKJAERBAEK N SOBY KK HANSEN HO EBERT B BOGESO KP KROGSGAARDLARSEN P
Citation: B. Bangandersen et al., HETEROARYL ANALOGS OF AMPA - SYNTHESIS AND QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS, Journal of medicinal chemistry, 40(18), 1997, pp. 2831-2842
MOLECULAR PHARMACOLOGY OF 4-SUBSTITUTED GLUTAMIC-ACID ANALOGS AT IONOTROPIC AND METABOTROPIC EXCITATORY AMINO-ACID RECEPTORS
Authors: BRAUNEROSBORNE H NIELSEN B STENSBOL TB JOHANSEN TN SKJAERBAEK N KROGSGAARDLARSEN P
Citation: H. Braunerosborne et al., MOLECULAR PHARMACOLOGY OF 4-SUBSTITUTED GLUTAMIC-ACID ANALOGS AT IONOTROPIC AND METABOTROPIC EXCITATORY AMINO-ACID RECEPTORS, European journal of pharmacology, 335(2-3), 1997, pp. 1-3
DIFFERENTIAL-EFFECTS OF NIPECOTIC ACID AND 4,5,6,7-TETRAHYDROISOXAZOLO[4,5-C]PYRIDIN-3-OL ON EXTRACELLULAR GAMMA-AMINOBUTYRATE LEVELS IN RAT THALAMUS
Authors: JUHASZ G KEKESI KA NYITRAI G DOBOLYI A KROGSGAARDLARSEN P SCHOUSBOE A
Citation: G. Juhasz et al., DIFFERENTIAL-EFFECTS OF NIPECOTIC ACID AND 4,5,6,7-TETRAHYDROISOXAZOLO[4,5-C]PYRIDIN-3-OL ON EXTRACELLULAR GAMMA-AMINOBUTYRATE LEVELS IN RAT THALAMUS, European journal of pharmacology, 331(2-3), 1997, pp. 139-144
Risultati: 1-25 | 26-50 | 51-70