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Results: 1-25 | 26-28
Results: 1-25/28
Crystal structure of 7-chloropyrrolo[1,2-b][1,2,5]benzothiadiazepin-10(11H)-one-5,5-dioxide, C11H7N2O3ClS
Authors: Ettorre, A Silvestri, R Artico, M Massa, S La Colla, P
Citation: A. Ettorre et al., Crystal structure of 7-chloropyrrolo[1,2-b][1,2,5]benzothiadiazepin-10(11H)-one-5,5-dioxide, C11H7N2O3ClS, Z KRIST-NEW, 216(1), 2001, pp. 57-58
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase
Authors: Mai, A Sbardella, G Artico, M Ragno, R Massa, S Novellino, E Greco, G Lavecchia, A Musiu, C La Colla, M Murgioni, C La Colla, P Loddo, R
Citation: A. Mai et al., Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase, J MED CHEM, 44(16), 2001, pp. 2544-2554
Synthesis and anti-HIV-1 activity of new delavirdine analogues carrying arylpyrrole moieties
Authors: Pinna, GA Loriga, G Murineddu, G Grella, G Mura, M Vargiu, L Murgioni, C La Colla, P
Citation: Ga. Pinna et al., Synthesis and anti-HIV-1 activity of new delavirdine analogues carrying arylpyrrole moieties, CHEM PHARM, 49(11), 2001, pp. 1406-1411
Pyrazole related nucleosides 5. Synthesis and biological activity of 2 '-deoxy-2 ',3 '-dideoxy- and acyclo-analogues of 4-iodo-1-beta-D-ribofuranosyl-3-carboxymethyl pyrazole (IPCAR).
Authors: Manfredini, S Baraldi, PG Bazzanini, R Durini, E Vertuani, S Pani, A Marceddu, T Demontis, F Vargiu, L La Colla, P
Citation: S. Manfredini et al., Pyrazole related nucleosides 5. Synthesis and biological activity of 2 '-deoxy-2 ',3 '-dideoxy- and acyclo-analogues of 4-iodo-1-beta-D-ribofuranosyl-3-carboxymethyl pyrazole (IPCAR)., NUCLEOS NUC, 19(4), 2000, pp. 705-722
MDR1, cholesterol esterification and cell growth: a comparative study in normal and multidrug-resistant KB cell Lines
Authors: Pani, A Batetta, B Putzolu, M Sanna, F Spano, O Piras, S Mulas, MF Bonatesta, RR Filippo, CAD Vargiu, L Marceddu, T Sanna, L La Colla, P Dessi, S
Citation: A. Pani et al., MDR1, cholesterol esterification and cell growth: a comparative study in normal and multidrug-resistant KB cell Lines, CELL MOL L, 57(7), 2000, pp. 1094-1102
Does the 2-methylthiomethyl substituent really confer high anti-HIV-1 activity to S-DABOS?
Authors: Sbardella, G Mai, A Artico, M Massa, S Marceddu, T Vargiu, L Marongiu, ME La Colla, P
Citation: G. Sbardella et al., Does the 2-methylthiomethyl substituent really confer high anti-HIV-1 activity to S-DABOS?, MED CHEM RE, 10(1), 2000, pp. 30-39
Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors
Authors: Silvestri, R Artico, M De Martino, G Novellino, E Greco, G Lavecchia, A Massa, S Loi, AG Doratiotto, S La Colla, P
Citation: R. Silvestri et al., Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors, BIO MED CH, 8(9), 2000, pp. 2305-2309
Peptide T-araC conjugates: Solid-phase synthesis and biological activity of N-4-(acylpeptidyl)-araC
Authors: Manfredini, S Marastoni, M Tomatis, R Durini, E Spisani, S Pani, A Marceddu, T Musiu, C Marongiu, ME La Colla, P
Citation: S. Manfredini et al., Peptide T-araC conjugates: Solid-phase synthesis and biological activity of N-4-(acylpeptidyl)-araC, BIO MED CH, 8(3), 2000, pp. 539-547
Synthesis and antimicrobial activity of new 3-(1-R-3(5)-methyl-4-nitroso-1H-5(3)-pyrazolyl)-5-methylisoxazoles
Authors: Aiello, E Aiello, S Mingoia, F Bacchi, A Pelizzi, G Musiu, C Setzu, MG Pani, A La Colla, P Marongiu, ME
Citation: E. Aiello et al., Synthesis and antimicrobial activity of new 3-(1-R-3(5)-methyl-4-nitroso-1H-5(3)-pyrazolyl)-5-methylisoxazoles, BIO MED CH, 8(12), 2000, pp. 2719-2728
1-[2-(Diphenylmethoxy)ethyl]-2-methyl-5-nitroimidazole: a potent lead for the design of novel NNRTIs
Authors: Silvestri, R Artico, M Massa, S Marceddu, T De Montis, F La Colla, P
Citation: R. Silvestri et al., 1-[2-(Diphenylmethoxy)ethyl]-2-methyl-5-nitroimidazole: a potent lead for the design of novel NNRTIs, BIOORG MED, 10(3), 2000, pp. 253-256
Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase
Authors: Costi, R Di Santo, R Artico, M Massa, S Lavecchia, A Marceddu, T Sanna, L La Colla, P Marongiu, ME
Citation: R. Costi et al., Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase, ANTIVIR CHE, 11(2), 2000, pp. 117-133
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines
Authors: Castellano, S Stefancich, G Musiu, C La Colla, P
Citation: S. Castellano et al., A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines, ARCH PHARM, 333(9), 2000, pp. 299-304
Azole antifungal agents related to naftifine and butenafine
Authors: Castellano, S La Colla, P Musiu, C Stefancich, G
Citation: S. Castellano et al., Azole antifungal agents related to naftifine and butenafine, ARCH PHARM, 333(6), 2000, pp. 162-166
Structure-based design, synthesis, and biological evaluation of navel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations
Authors: Artico, M Silvestri, R Pagnozzi, E Bruno, B Novellino, E Greco, G Massa, S Ettorre, A Loi, AG Scintu, F La Colla, P
Citation: M. Artico et al., Structure-based design, synthesis, and biological evaluation of navel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations, J MED CHEM, 43(9), 2000, pp. 1886-1891
Synthesis of tricyclic triazepinones related to nevirapine
Authors: Castellano, S Stefancich, G La Colla, P Musiu, C
Citation: S. Castellano et al., Synthesis of tricyclic triazepinones related to nevirapine, J HETERO CH, 37(6), 2000, pp. 1539-1542
Antiproliferative and antimicrobial activities of pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides and their 5-deoxyderivatives
Authors: Costanzo, A Ciciani, G Guerrini, G Bruni, F Selleri, S Donato, R Sacco, C Musiu, C Milia, C Longu, S Minnei, C La Colla, P
Citation: A. Costanzo et al., Antiproliferative and antimicrobial activities of pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides and their 5-deoxyderivatives, MED CHEM RE, 9(4), 1999, pp. 223-238
Indolo[3,2-c]cinnolines with antiproliferative, antifungal, and antibacterial activity
Authors: Barraja, P Diana, P Lauria, A Passannanti, A Almerico, AM Minnei, C Longu, S Congiu, D Musiu, C La Colla, P
Citation: P. Barraja et al., Indolo[3,2-c]cinnolines with antiproliferative, antifungal, and antibacterial activity, BIO MED CH, 7(8), 1999, pp. 1591-1596
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro
Authors: Artico, M Mai, A Sbardella, G Massa, S Musiu, C Lostia, S Demontis, F La Colla, P
Citation: M. Artico et al., Nitroquinolones with broad-spectrum antimycobacterial activity in vitro, BIOORG MED, 9(12), 1999, pp. 1651-1656
Effect of acyclic nucleoside phosphonates on the HIV-1 integrase in vitro
Authors: Abu Sheika, G Tramontano, E Loi, AG Franchetti, P Grifantini, M La Colla, P
Citation: G. Abu Sheika et al., Effect of acyclic nucleoside phosphonates on the HIV-1 integrase in vitro, NUCLEOS NUC, 18(4-5), 1999, pp. 849-851
Synthesis and antiproliferative activity of 2-triazenothiophenes
Authors: Diana, P Barraja, P Lauria, A Almerico, AM Cirrincione, G Minnei, C Longu, S Congiu, D Musiu, C La Colla, P
Citation: P. Diana et al., Synthesis and antiproliferative activity of 2-triazenothiophenes, ANTICANC R, 19(3A), 1999, pp. 2127-2131
2-triazenopyrroles: synthesis and biological activity
Authors: Diana, P Barraja, P Lauria, A Almerico, AM Cirrincione, G Loi, AG Musiu, C Pani, A La Colla, P Marongiu, ME
Citation: P. Diana et al., 2-triazenopyrroles: synthesis and biological activity, EUR J MED C, 34(4), 1999, pp. 353-360
5-alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives
Authors: Mai, A Artico, M Sbardella, G Massa, S Novellino, E Greco, G Loi, AG Tramontano, E Marongiu, ME La Colla, P
Citation: A. Mai et al., 5-alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives, J MED CHEM, 42(4), 1999, pp. 619-627
Derivatives of the new ring system indolo[1,2-c]benzo[1,2,3]triazine with potent antitumor and antimicrobial activity
Authors: Cirrincione, G Almerico, AM Barraja, P Diana, P Lauria, A Passannanti, A Musiu, C Pani, A Murtas, P Minnei, C Marongiu, ME La Colla, P
Citation: G. Cirrincione et al., Derivatives of the new ring system indolo[1,2-c]benzo[1,2,3]triazine with potent antitumor and antimicrobial activity, J MED CHEM, 42(14), 1999, pp. 2561-2568
Phthalein derivatives as a new tool for selectivity in thymidylate synthase
Authors: Costi, PM Rinaldi, M Tondi, D Pecorari, P Barlocco, D Ghelli, S Stroud, RM Santi, DV Stout, TJ Musiu, C Marangiu, EM Pani, A Congiu, D Loi, GA La Colla, P
Citation: Pm. Costi et al., Phthalein derivatives as a new tool for selectivity in thymidylate synthase, J MED CHEM, 42(12), 1999, pp. 2112-2124
Synthesis and biological evaluation of [alpha-(1,5-disubstituted 1H-pyrazol-4-yl)benzyl]azoles, analogues of bifonazole
Authors: Menozzi, G Mosti, L Bruno, O Lo Presti, E Musiu, C Longu, S La Colla, P Filippelli, W Falcone, G Piucci, B
Citation: G. Menozzi et al., Synthesis and biological evaluation of [alpha-(1,5-disubstituted 1H-pyrazol-4-yl)benzyl]azoles, analogues of bifonazole, FARMACO, 54(6), 1999, pp. 416-422
Risultati: 1-25 | 26-28