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Results: 1-15 |
Results: 15
DUAL METALLOPROTEASE INHIBITORS - MERCAPTOACETYL-BASED FUSED HETEROCYCLIC DIPEPTIDE MIMETICS AS INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYMEAND NEUTRAL ENDOPEPTIDASE
Authors: ROBL JA SUN CQ STEVENSON J RYONO DE SIMPKINS LM CIMARUSTI MP DEJNEKA T SLUSARCHYK WA CHAO S STRATTON L MISRA RN BEDNARZ MS ASAAD MM CHEUNG HS ABBOAOFFEI BE SMITH PL MATHERS PD FOX M SCHAEFFER TR SEYMOUR AA TRIPPODO NC
Citation: Ja. Robl et al., DUAL METALLOPROTEASE INHIBITORS - MERCAPTOACETYL-BASED FUSED HETEROCYCLIC DIPEPTIDE MIMETICS AS INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYMEAND NEUTRAL ENDOPEPTIDASE, Journal of medicinal chemistry, 40(11), 1997, pp. 1570-1577
PRODRUGS OF BMS-183920 - METABOLISM AND PERMEABILITY CONSIDERATIONS
Authors: OBERMEIER MT CHONG SH DANDO SA MARINO AM RYONO DE STARRETTARROYO A DIDONATO GC WARRACK BM WHITE RE MORRISON RA
Citation: Mt. Obermeier et al., PRODRUGS OF BMS-183920 - METABOLISM AND PERMEABILITY CONSIDERATIONS, Journal of pharmaceutical sciences, 85(8), 1996, pp. 828-833
DUAL METALLOPROTEASE INHIBITORS .6. INCORPORATION OF BICYCLIC AND SUBSTITUTED MONOCYCLIC AZEPINONES AS DIPEPTIDE SURROGATES IN ANGIOTENSIN-CONVERTING ENZYME NEUTRAL ENDOPEPTIDASE INHIBITORS
Authors: ROBL JA CIMARUSTI MP SIMPKINS LM BROWN B RYONO DE BIRD JE ASAAD MM SCHAEFFER TR TRIPPODO NC
Citation: Ja. Robl et al., DUAL METALLOPROTEASE INHIBITORS .6. INCORPORATION OF BICYCLIC AND SUBSTITUTED MONOCYCLIC AZEPINONES AS DIPEPTIDE SURROGATES IN ANGIOTENSIN-CONVERTING ENZYME NEUTRAL ENDOPEPTIDASE INHIBITORS, Journal of medicinal chemistry, 39(2), 1996, pp. 494-502
AMINODIOL HIV PROTEASE INHIBITORS - SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF P-1 P-1' COMPOUNDS - CORRELATION BETWEEN LIPOPHILICITY AND CYTOTOXICITY/
Authors: CHEN P CHENG PTW ALAM M BEYER BD BISACCHI GS DEJNEKA T EVANS AJ GREYTOK JA HERMSMEIER MA HUMPHREYS WG JACOBS GA KOCY O LIN PF LIS KA MARELLA MA RYONO DE SHEAFFER AK SPERGEL SH SUN CQ TINO JA VITE G COLONNO RJ ZAHLER R BARRISH JC
Citation: P. Chen et al., AMINODIOL HIV PROTEASE INHIBITORS - SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF P-1 P-1' COMPOUNDS - CORRELATION BETWEEN LIPOPHILICITY AND CYTOTOXICITY/, Journal of medicinal chemistry, 39(10), 1996, pp. 1991-2007
ALPHA-HYDROXY PHOSPHINYL-BASED INHIBITORS OF HUMAN RENIN
Authors: PATEL DV RIELLYGAUVIN K RYONO DE FREE CA ROGERS WL SMITH SA DEFORREST JM OEHL RS PETRILLO EW
Citation: Dv. Patel et al., ALPHA-HYDROXY PHOSPHINYL-BASED INHIBITORS OF HUMAN RENIN, Journal of medicinal chemistry, 38(22), 1995, pp. 4557-4569
DUAL METALLOPROTEASE INHIBITORS .4. UTILIZATION OF THIAZEPINES AND THIAZINES AS CONSTRAINED PEPTIDOMIMETIC SURROGATES IN MERCAPTOACYL DIPEPTIDES
Authors: DAS J ROBL JA REID JA SUN CQ MISRA RN BROWN BR RYONO DE ASAAD MM BIRD JE TRIPPODO NC PETRILLO EW KARANEWSKY DS
Citation: J. Das et al., DUAL METALLOPROTEASE INHIBITORS .4. UTILIZATION OF THIAZEPINES AND THIAZINES AS CONSTRAINED PEPTIDOMIMETIC SURROGATES IN MERCAPTOACYL DIPEPTIDES, Bioorganic & medicinal chemistry letters, 4(18), 1994, pp. 2193-2198
DUAL METALLOPROTEASE INHIBITORS .3. UTILIZATION OF BICYCLIC AND MONOCYCLIC DIAZEPINONE BASED MERCAPTOACETYLS
Authors: ROBL JA SUN CQ SIMPKINS LM RYONO DE BARRISH JC KARANEWSKY DS ASAAD MM SCHAEFFER TR TRIPPODO NC
Citation: Ja. Robl et al., DUAL METALLOPROTEASE INHIBITORS .3. UTILIZATION OF BICYCLIC AND MONOCYCLIC DIAZEPINONE BASED MERCAPTOACETYLS, Bioorganic & medicinal chemistry letters, 4(16), 1994, pp. 2055-2060
DUAL METALLOPROTEASE INHIBITORS .2. EFFECT OF SUBSTITUTION AND STEREOCHEMISTRY ON BENZAZEPINONE BASED MERCAPTOACETYLS
Authors: ROBL JA SIMPKINS LM SULSKY R SIEBERMCMASTER E STEVENSON J KELLY YF SUN CQ MISRA RN RYONO DE ASAAD MM BIRD JE TRIPPODO NC KARANEWSKY DS
Citation: Ja. Robl et al., DUAL METALLOPROTEASE INHIBITORS .2. EFFECT OF SUBSTITUTION AND STEREOCHEMISTRY ON BENZAZEPINONE BASED MERCAPTOACETYLS, Bioorganic & medicinal chemistry letters, 4(15), 1994, pp. 1795-1800
1-4-SUBSTITUTED INDOLES - A POTENT AND SELECTIVE CLASS OF ANGIOTENSIN-II RECEPTOR ANTAGONISTS
Authors: POSS MA GU ZX RYONO DE REID JA SIEBERMCMASTER E SPITZMILLER ER DEJNEKA T DICKINSON KEJ WILLIAMS SB MORELAND S DELANEY CL BIRD JE WALDRON TL SCHAEFFER TR HEDBERG SA PETRILLO EW
Citation: Ma. Poss et al., 1-4-SUBSTITUTED INDOLES - A POTENT AND SELECTIVE CLASS OF ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 145-150
QUINOLINE-4-CARBOXYLIC ACIDS AS ANGIOTENSIN-II RECEPTOR ANTAGONISTS
Authors: LLOYD J RYONO DE BIRD JE BUOTE J DELANEY CL DEJNEKA T DICKINSON KEJ MORELAND S NORMANDIN DE SKWISH S SPITZMILLER ER WALDRON TL
Citation: J. Lloyd et al., QUINOLINE-4-CARBOXYLIC ACIDS AS ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 195-200
ORALLY-ACTIVE PRODRUGS OF QUINOLINE-4-CARBOXYLIC ACID ANGIOTENSIN-II RECEPTOR ANTAGONISTS
Authors: RYONO DE LLOYD J POSS MA BIRD JE BUOTE J CHONG S DEJNEKA T DICKINSON KEJ GU Z MATHERS P MORELAND S MORRISON RA PETRILLO EW POWELL JR SCHAEFFER T SPITZMILLER ER WHITE RE
Citation: De. Ryono et al., ORALLY-ACTIVE PRODRUGS OF QUINOLINE-4-CARBOXYLIC ACID ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 201-206
ALPHA-HYDROXY PHOSPHINYL BASED TRANSITION-STATE ANALOG RENIN INHIBITORS - MINIMAL STRUCTURAL REQUIREMENTS FOR GOOD INHIBITORY ACTIVITY
Authors: PATEL DV RIELLYGAUVIN K FREE CA ROGERS WL SMITH SA RYONO DE PETRILLO EW
Citation: Dv. Patel et al., ALPHA-HYDROXY PHOSPHINYL BASED TRANSITION-STATE ANALOG RENIN INHIBITORS - MINIMAL STRUCTURAL REQUIREMENTS FOR GOOD INHIBITORY ACTIVITY, Journal of cellular biochemistry, 1994, pp. 159-159
BMS-180560, AN INSURMOUNTABLE INHIBITOR OF ANGIOTENSIN II-STIMULATED RESPONSES - COMPARISON WITH LOSARTAN AND EXP3174
Authors: DICKINSON KEJ COHEN RB SKWISH S DELANEY CL SERAFINO RP POSS MA GU Z RYONO DE MORELAND S POWELL JR
Citation: Kej. Dickinson et al., BMS-180560, AN INSURMOUNTABLE INHIBITOR OF ANGIOTENSIN II-STIMULATED RESPONSES - COMPARISON WITH LOSARTAN AND EXP3174, British Journal of Pharmacology, 113(1), 1994, pp. 179-189
DIOL SULFONAMIDES - A POTENT AND NOVEL CLASS OF INHIBITORS OF HUMAN RENIN
Authors: POSS MA REID JA FREE CA ROGERS WL WEBER H RYONO DE DEJNEKA T DEFORREST JM WALDRON TL BRITTAIN RJ WELLER HN CIMARUSTI MP PETRILLO EW
Citation: Ma. Poss et al., DIOL SULFONAMIDES - A POTENT AND NOVEL CLASS OF INHIBITORS OF HUMAN RENIN, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2739-2744
ACTIVATED KETONE BASED INHIBITORS OF HUMAN RENIN
Authors: PATEL DV RIELLYGAUVIN K RYONO DE FREE CA SMITH SA PETRILLO EW
Citation: Dv. Patel et al., ACTIVATED KETONE BASED INHIBITORS OF HUMAN RENIN, Journal of medicinal chemistry, 36(17), 1993, pp. 2431-2447
Risultati: 1-15 |