Authors:
ALVESRODRIGUES A
TIMMERMAN H
WILLEMS E
LEMSTRA S
ZUIDERVELD OP
LEURS R
Citation: A. Alvesrodrigues et al., PHARMACOLOGICAL CHARACTERIZATION OF THE HISTAMINE H-3 RECEPTOR IN THERAT HIPPOCAMPUS, Brain research, 788(1-2), 1998, pp. 179-186
Citation: R. Leurs et al., THERAPEUTIC POTENTIAL HISTAMINE H-3 RECEPTOR AGONISTS AND ANTAGONISTS, Trends in pharmacological sciences, 19(5), 1998, pp. 177-183
Authors:
CORUZZI G
POLI E
POZZOLI C
BERTACCINI G
TIMMERMAN H
Citation: G. Coruzzi et al., HISTAMINE RECEPTOR-INDEPENDENT MUSCLE-RELAXATION ELICITED BY A SERIESOF HISTAMINE H-2-RECEPTOR AGONISTS ON THE ISOLATED GUINEA-PIG DUODENUM - A STUDY INTO THE MECHANISM OF ACTION, General pharmacology, 31(4), 1998, pp. 643-651
Authors:
ZWAAGSTRA ME
KORTHOUWER REM
TIMMERMAN H
ZHANG MQ
Citation: Me. Zwaagstra et al., SYNTHESIS OF 3-SUBSTITUTED AND 5'-SUBSTITUTED FLAVONE-8-CARBOXYLIC ACIDS AS 3-ARMED LEUKOTRIENE CYSLT(1) RECEPTOR ANTAGONISTS, European journal of medicinal chemistry, 33(2), 1998, pp. 95-102
Authors:
NEDERKOORN PHJ
TIMMERMAN H
TIMMS D
WILKINSON AJ
KELLY DR
BROADLEY KJ
DAVIES RH
Citation: Phj. Nederkoorn et al., STEPWISE PHOSPHORYLATION MECHANISMS AND SIGNAL TRANSMISSION WITHIN A LIGAND-RECEPTOR-G-ALPHA-BETA-GAMMA-PROTEIN-COMPLEX, Journal of molecular structure. Theochem, 452, 1998, pp. 25-47
Authors:
MOREEUW AM
DECOCK P
TIMMERMAN H
KOZLOWSKI H
Citation: Am. Moreeuw et al., BINDING ABILITY OF IMPROMIDINE, A POTENT H-2 HISTAMINE AGONIST AND ITS ANALOGS, Journal of inorganic biochemistry, 70(2), 1998, pp. 107-111
Authors:
ALEWIJNSE AE
SMIT MJ
HOFFMANN M
TIMMERMAN H
LEURS R
Citation: Ae. Alewijnse et al., CONSTITUTIVE ACTIVITY OF THE HISTAMINE H-2-RECEPTOR, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 116-116
Authors:
ALEWIJNSE AE
TIMMERMAN H
SMIT MJ
ROOVERS E
JACOBS EH
LEURS R
Citation: Ae. Alewijnse et al., MUTATIONAL ANALYSIS OF THE CONSERVED DRY MOTIF IN THE RAT HISTAMINE H-2-RECEPTOR, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 915-915
Authors:
ALEWIJNSE AE
SMIT MJ
HOFFMANN M
TIMMERMAN H
LEURS R
Citation: Ae. Alewijnse et al., CONSTITUTIVE ACTIVITY OF THE HISTAMINE H-2-RECEPTOR, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 928-928
Authors:
ALEWIJNSE AE
SMIT MJ
HOFFMANN M
VERZIJL D
TIMMERMAN H
LEURS R
Citation: Ae. Alewijnse et al., CONSTITUTIVE ACTIVITY AND STRUCTURAL INSTABILITY OF THE WILD-TYPE HUMAN H-2-RECEPTOR, Journal of neurochemistry, 71(2), 1998, pp. 799-807
Authors:
ZWAAGSTRA ME
TIMMERMAN H
VANDESTOLPE AC
DEKANTER FJJ
TAMURA M
WADA Y
ZHANG MQ
Citation: Me. Zwaagstra et al., SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF CARBOXYFLAVONES AS STRUCTURALLY RIGID CYSLT(1) (LTD4) RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 41(9), 1998, pp. 1428-1438
Authors:
ZWAAGSTRA ME
SCHOENMAKERS SHHF
NEDERKOORN PHJ
GELENS E
TIMMERMAN H
ZHANG MQ
Citation: Me. Zwaagstra et al., DEVELOPMENT OF A 3-DIMENSIONAL CYSLT(1) (LTD4) ANTAGONIST MODEL WITH AN INCORPORATED AMINO-ACID RESIDUE FROM THE RECEPTOR, Journal of medicinal chemistry, 41(9), 1998, pp. 1439-1445
Authors:
VANMUIJLWIJKKOEZEN JE
TIMMERMAN H
LINK R
VANDERGOOT H
IJZERMAN AP
Citation: Je. Vanmuijlwijkkoezen et al., A NOVEL CLASS OF ADENOSINE A(3) RECEPTOR LIGANDS - 1 - 3-(2-PYRIDINYL)ISOQUINOLINE DERIVATIVES, Journal of medicinal chemistry, 41(21), 1998, pp. 3987-3993
Authors:
VANMUIJLWIJKKOEZEN JE
TIMMERMAN H
LINK R
VANDERGOOT H
IJZERMANI AP
Citation: Je. Vanmuijlwijkkoezen et al., A NOVEL CLASS OF ADENOSINE A(3) RECEPTOR LIGANDS - 2 - STRUCTURE AFFINITY PROFILE OF A SERIES OF ISOQUINOLINE AND QUINAZOLINE COMPOUNDS, Journal of medicinal chemistry, 41(21), 1998, pp. 3994-4000
Authors:
NEDERKOORN PHJ
DAVIES RH
TIMMS D
TIMMERMAN H
Citation: Phj. Nederkoorn et al., TRIMERIC G-ALPHA-BETA-GAMMA PROTEIN COUPLING TO A 3D MODEL OF G-PROTEIN-COUPLED RECEPTORS CONFIRMING A NEW MOLECULAR MECHANISM FOR ACTIVATION, Receptors & channels, 5(2), 1997, pp. 91
Citation: Mj. Smit et al., FROM HISTAMINE H-2-RECEPTOR REGULATION TO RECLASSIFICATION OF H-2 ANTAGONISTS - INVERSE AGONISM AS THE BASIS FOR H-2-RECEPTOR UP-REGULATION, Receptors & channels, 5(2), 1997, pp. 99-102
Citation: Mq. Zhang et H. Timmerman, LEUKOTRIENE CYSLT(1) (LTD(4)) RECEPTOR ANTAGONISM OF H-1-ANTIHISTAMINES - AN IN-VITRO STUDY, Inflammation research, 46, 1997, pp. 93-94
Authors:
ZHANG MQ
ZWAAGSTRA ME
NEDERKOORN PHJ
TIMMERMAN H
Citation: Mq. Zhang et al., THE ROLE OF ARGININE IN THE BINDING OF LTD4 ANTAGONISTS TO CYSLT(1) RECEPTORS OF GUINEA-PIG LUNG, Bioorganic & medicinal chemistry letters, 7(10), 1997, pp. 1331-1336
Authors:
PAQUAY JBG
TENBOLSCHER M
VOSS HP
TIMMERMAN H
BAST A
Citation: Jbg. Paquay et al., DIFFERENCE IN THE INHIBITION OF NITRIC-OXIDE SYNTHASE AND CYTOCHROME-P-450 BY H-2-ANTAGONISTS, Toxicology in vitro, 11(6), 1997, pp. 775-778
Authors:
SARDJIMAN SS
REKSOHADIPRODJO MS
HAKIM L
VANDERGOOT H
TIMMERMAN H
Citation: Ss. Sardjiman et al., 1,5-DIPHENYL-1,4-PENTADIENE-3-ONES AND CYCLIC ANALOGS AS ANTIOXIDATIVE AGENTS - SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP, European journal of medicinal chemistry, 32(7-8), 1997, pp. 625-630
Authors:
NURFINA AN
REKSOHADIPRODJO MS
TIMMERMAN H
JENIE UA
SUGIYANTO D
VANDERGOOT H
Citation: An. Nurfina et al., SYNTHESIS OF SOME SYMMETRICAL CURCUMIN DERIVATIVES AND THEIR ANTIINFLAMMATORY ACTIVITY, European journal of medicinal chemistry, 32(4), 1997, pp. 321-328
Authors:
ZHANG MQ
VANDESTOLPE A
ZUIDERVELD OP
TIMMERMAN H
Citation: Mq. Zhang et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF SOME AMINO-ACID-CONTAINING CYPROHEPTADINE DERIVATIVES AS DUAL ANTAGONISTS OF HISTAMINE H-1-RECEPTOR AND LEUKOTRIENE D-4-RECEPTOR, European journal of medicinal chemistry, 32(2), 1997, pp. 95-102
Authors:
VACCARI A
SABA PL
CALDIROLA MP
BIJLOO GJ
TIMMERMAN H
Citation: A. Vaccari et al., PRENYLAMINE DERIVATIVES AS BLOCKERS OF THE VESICULAR TRANSPORTER FOR DOPAMINE - A QUANTITATIVE STRUCTURE-ACTIVITY STUDY, European journal of medicinal chemistry, 32(1), 1997, pp. 53-57
Authors:
HILL SJ
GANELLIN CR
TIMMERMAN H
SCHWARTZ JC
SHANKLEY NP
YOUNG JM
SCHUNACK W
LEVI R
HAAS HL
Citation: Sj. Hill et al., INTERNATIONAL UNION OF PHARMACOLOGY .13. CLASSIFICATION OF HISTAMINE-RECEPTORS, Pharmacological reviews, 49(3), 1997, pp. 253-278