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Results: 1-25 |
Results: 25
PRACTICAL RESOLUTION OF AN ATROPOISOMERIC ALPHA,ALPHA-DISUBSTITUTED GLYCINE WITH L-PHENYLALANINE CYCLOHEXYLAMIDE AS CHIRAL AUXILIARY
Authors: MAZALEYRAT JP BOUTBOUL A LEBARS Y GAUCHER A WAKSELMAN M
Citation: Jp. Mazaleyrat et al., PRACTICAL RESOLUTION OF AN ATROPOISOMERIC ALPHA,ALPHA-DISUBSTITUTED GLYCINE WITH L-PHENYLALANINE CYCLOHEXYLAMIDE AS CHIRAL AUXILIARY, Tetrahedron : asymmetry, 9(15), 1998, pp. 2701-2713
SYNTHESIS OF ALPHA,ALPHA-DISUBSTITUTED-BETA-AMINO-ACIDS WITH AXIAL CHIRALITY
Authors: GAUCHER A BINTEIN F WAKSELMAN M MAZALEYRAT JP
Citation: A. Gaucher et al., SYNTHESIS OF ALPHA,ALPHA-DISUBSTITUTED-BETA-AMINO-ACIDS WITH AXIAL CHIRALITY, Tetrahedron letters, 39(7), 1998, pp. 575-578
ACYLATION OF SUGAR HYDROXYL-GROUPS WITH N-BOC AMINO-ACID N-CARBOXYANHYDRIDES (BOC-NCAS) - SYNTHESIS OF AMINO-ACID SACCHARIDE CONJUGATES
Authors: CABARET D WAKSELMAN M KABA A ILUNGA L CHANY C
Citation: D. Cabaret et al., ACYLATION OF SUGAR HYDROXYL-GROUPS WITH N-BOC AMINO-ACID N-CARBOXYANHYDRIDES (BOC-NCAS) - SYNTHESIS OF AMINO-ACID SACCHARIDE CONJUGATES, Synthetic communications, 28(14), 1998, pp. 2713-2724
SPECIFIC AND IRREVERSIBLE CYCLOPEPTIDE INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV ACTIVITY OF THE T-CELL ACTIVATION ANTIGEN CD26
Authors: NGUYEN C BLANCO J MAZALEYRAT JP KRUST B CALLEBAUT C JACOTOT E HOVANESSIAN AG WAKSELMAN M
Citation: C. Nguyen et al., SPECIFIC AND IRREVERSIBLE CYCLOPEPTIDE INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV ACTIVITY OF THE T-CELL ACTIVATION ANTIGEN CD26, Journal of medicinal chemistry, 41(12), 1998, pp. 2100-2110
DIPEPTIDYL-PEPTIDASE-IV-BETA - FURTHER CHARACTERIZATION AND COMPARISON TO DIPEPTIDYL-PEPTIDASE-IV ACTIVITY OF CD26
Authors: BLANCO J NGUYEN C CALLEBAUT C JACOTOT E KRUST B MAZALEYRAT JP WAKSELMAN M HOVANESSIAN AG
Citation: J. Blanco et al., DIPEPTIDYL-PEPTIDASE-IV-BETA - FURTHER CHARACTERIZATION AND COMPARISON TO DIPEPTIDYL-PEPTIDASE-IV ACTIVITY OF CD26, European journal of biochemistry, 256(2), 1998, pp. 369-378
HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC SEPARATION OF ENANTIOMERS OF 1,1'-BINAPHTHYL-SUBSTITUTED ALPHA-AMINOISOBUTYRIC-ACID
Authors: PETER A TOROK G MAZALEYRAT JP WAKSELMAN M
Citation: A. Peter et al., HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC SEPARATION OF ENANTIOMERS OF 1,1'-BINAPHTHYL-SUBSTITUTED ALPHA-AMINOISOBUTYRIC-ACID, Journal of chromatography, 790(1-2), 1997, pp. 41-46
INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL-3,3-DIHALOGENOAZETIDIN-2-ONES - STEREOSPECIFIC SYNTHESIS AND CHIRAL RECOGNITION OF DISSYMMETRICALLY C-3-SUBSTITUTED BETA-LACTAMS
Authors: DOUCET C VERGELY I REBOUDRAVAUX M GUILHEM J KOBAITER R JOYEAU R WAKSELMAN M
Citation: C. Doucet et al., INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL-3,3-DIHALOGENOAZETIDIN-2-ONES - STEREOSPECIFIC SYNTHESIS AND CHIRAL RECOGNITION OF DISSYMMETRICALLY C-3-SUBSTITUTED BETA-LACTAMS, Tetrahedron : asymmetry, 8(5), 1997, pp. 739-751
NOVEL ALPHA,ALPHA-DISUBSTITUTED ALPHA-AMINO-ACIDS WITH AXIAL DISSYMMETRY AND THEIR N-PROTECTED OR C-PROTECTED DERIVATIVES
Authors: MAZALEYRAT JP GAUCHER A SAVRDA J WAKSELMAN M
Citation: Jp. Mazaleyrat et al., NOVEL ALPHA,ALPHA-DISUBSTITUTED ALPHA-AMINO-ACIDS WITH AXIAL DISSYMMETRY AND THEIR N-PROTECTED OR C-PROTECTED DERIVATIVES, Tetrahedron : asymmetry, 8(4), 1997, pp. 619-631
N-T-BOC 7-DIHYDRO-5H-DIBENZO[A,C]CYCLOHEPTENE-6-CARBOXYLIC ACID METHYL-ESTER, THE FIRST PROTOTYPE OF A CROWN-CARRIER AXIALLY DISSYMMETRIC-ALPHA,ALPHA-DISUBSTITUTED GLYCINE
Authors: MAZALEYRAT JP GAUCHER A GOUBARD Y SAVRDA J WAKSELMAN M
Citation: Jp. Mazaleyrat et al., N-T-BOC 7-DIHYDRO-5H-DIBENZO[A,C]CYCLOHEPTENE-6-CARBOXYLIC ACID METHYL-ESTER, THE FIRST PROTOTYPE OF A CROWN-CARRIER AXIALLY DISSYMMETRIC-ALPHA,ALPHA-DISUBSTITUTED GLYCINE, Tetrahedron letters, 38(12), 1997, pp. 2091-2094
A NEW CHIRAL ALPHA-AMINO-ACID WITH ONLY AXIAL DISSYMMETRY - SYNTHESISAND X-RAY-ANALYSIS OF A 1,1'-BINAPHTHYL-SUBSTITUTED ALPHA-AMINOISOBUTYRIC-ACID (BIN) AND OF ITS BIPHENYL ANALOG (BIP)
Authors: MAZALEYRAT JP GAUCHER A WAKSELMAN M TCHERTANOV L GUILHEM J
Citation: Jp. Mazaleyrat et al., A NEW CHIRAL ALPHA-AMINO-ACID WITH ONLY AXIAL DISSYMMETRY - SYNTHESISAND X-RAY-ANALYSIS OF A 1,1'-BINAPHTHYL-SUBSTITUTED ALPHA-AMINOISOBUTYRIC-ACID (BIN) AND OF ITS BIPHENYL ANALOG (BIP), Tetrahedron letters, 37(17), 1996, pp. 2971-2974
SYNTHESIS AND INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL AZETIDIN-2-ONES - EFFECT OF DIFFERENT SUBSTITUENTS ON THE AROMATIC RING
Authors: JOYEAU R FELK A GUILAUME S WAKSELMAN M VERGELY I DOUCET C BOGGETTO N REBOUDRAVAUX M
Citation: R. Joyeau et al., SYNTHESIS AND INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL AZETIDIN-2-ONES - EFFECT OF DIFFERENT SUBSTITUENTS ON THE AROMATIC RING, Journal of Pharmacy and Pharmacology, 48(12), 1996, pp. 1218-1230
THE WILLIAMSON REACTION - A NEW AND EFFICIENT METHOD FOR THE ALTERNATE RESOLUTION OF 2,2'-BIS(BROMOMETHYL)-1,1'-BINAPHTHYL AND 1,1'-BINAPHTHALENE-2,2'-DIOL
Authors: MAZALEYRAT JP WAKSELMAN M
Citation: Jp. Mazaleyrat et M. Wakselman, THE WILLIAMSON REACTION - A NEW AND EFFICIENT METHOD FOR THE ALTERNATE RESOLUTION OF 2,2'-BIS(BROMOMETHYL)-1,1'-BINAPHTHYL AND 1,1'-BINAPHTHALENE-2,2'-DIOL, Journal of organic chemistry, 61(8), 1996, pp. 2695-2698
INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL AZETIDIN-2-ONES - SUBSTITUENT EFFECTS AT C-3 AND BENZYLIC POSITIONS
Authors: VERGELY I BOGGETTO N OKOCHI V GOLPAYEGANI S REBOUDRAVAUX M KOBAITER R JOYEAU R WAKSELMAN M
Citation: I. Vergely et al., INHIBITION OF HUMAN-LEUKOCYTE ELASTASE BY FUNCTIONALIZED N-ARYL AZETIDIN-2-ONES - SUBSTITUENT EFFECTS AT C-3 AND BENZYLIC POSITIONS, European journal of medicinal chemistry, 30(3), 1995, pp. 199-208
SYNTHESIS OF NEW DIOXACYCLOPHANES DERIVED FROM 1,1'-BINAPHTHYL-2,2'-DIOL
Authors: MAZALEYRAT JP WAKSELMAN M
Citation: Jp. Mazaleyrat et M. Wakselman, SYNTHESIS OF NEW DIOXACYCLOPHANES DERIVED FROM 1,1'-BINAPHTHYL-2,2'-DIOL, Synthetic communications, 25(23), 1995, pp. 3845-3854
LIQUID-CRYSTAL PROPERTIES OF OCTYL 6'-O-ALKYLMELIBIOSIDES
Authors: WINGERT LM JEFFREY GA CABARET D WAKSELMAN M
Citation: Lm. Wingert et al., LIQUID-CRYSTAL PROPERTIES OF OCTYL 6'-O-ALKYLMELIBIOSIDES, Carbohydrate research, 275(1), 1995, pp. 25-31
SYNTHESIS OF C2-SYMMETRICAL INHIBITORS OF THE HIV-1 PROTEASE, WITH N,N'-SUBSTITUTED ETHYLENEDIAMIDE AND ETHYLENEDIAMINE LINKERS
Authors: MAZALEYRAT JP RAGE I SAVRDA J MOUNA M WAKSELMAN M BOULAY R LELIEVRE Y
Citation: Jp. Mazaleyrat et al., SYNTHESIS OF C2-SYMMETRICAL INHIBITORS OF THE HIV-1 PROTEASE, WITH N,N'-SUBSTITUTED ETHYLENEDIAMIDE AND ETHYLENEDIAMINE LINKERS, Bioorganic & medicinal chemistry letters, 4(5), 1994, pp. 653-656
ANTI-HIV ACTIVITY OF N-(2,3-DIHALOGENOPROPYL)-GLYCINE AND N-ALLYL-GLYCINE CONTAINING PENTAPEPTIDES
Authors: WAKSELMAN M MOUNA AM XIE J MAZALEYRAT JP BOULAY R LELIEVRE Y BOUSSEAU A NACHMANSOHN C HENIN Y
Citation: M. Wakselman et al., ANTI-HIV ACTIVITY OF N-(2,3-DIHALOGENOPROPYL)-GLYCINE AND N-ALLYL-GLYCINE CONTAINING PENTAPEPTIDES, Bioorganic & medicinal chemistry letters, 4(21), 1994, pp. 2533-2537
PEPTOID MIMICS OF A C-2-SYMMETRICAL INHIBITOR OF THE HIV-1 PROTEASE
Authors: MAZALEYRAT JP RAGE I MOUNA AM SAVRDA J WAKSELMAN M BOULAY R LELIEVRE Y
Citation: Jp. Mazaleyrat et al., PEPTOID MIMICS OF A C-2-SYMMETRICAL INHIBITOR OF THE HIV-1 PROTEASE, Bioorganic & medicinal chemistry letters, 4(11), 1994, pp. 1281-1284
URETHANE PROTECTED AMINO-ACID N-CARBOXYANHYDRIDES AND FLUORIDES (U-NCAS AND U(2)AAFS)
Authors: WAKSELMAN M MAZALEYRAT JP SAVRDA J
Citation: M. Wakselman et al., URETHANE PROTECTED AMINO-ACID N-CARBOXYANHYDRIDES AND FLUORIDES (U-NCAS AND U(2)AAFS), Amino acids, 7(1), 1994, pp. 67-77
A LOW-EPIMERIZING PEPTIDE COUPLING REAGENT BASED ON THE REARRANGEMENTOF A CARBOXYLIC-SULFONIC MIXED ANHYDRIDE
Authors: CABARET D WAKSELMAN M
Citation: D. Cabaret et M. Wakselman, A LOW-EPIMERIZING PEPTIDE COUPLING REAGENT BASED ON THE REARRANGEMENTOF A CARBOXYLIC-SULFONIC MIXED ANHYDRIDE, Tetrahedron letters, 35(51), 1994, pp. 9561-9564
ACTIVATION OF N,N-BIS(ALKOXYCARBONYL) AMINO-ACIDS - SYNTHESIS OF N-ALKOXYCARBONYL AMINO-ACID N-CARBOXYANHYDRIDES AND N,N-DIALKOXYCARBONYL AMINO-ACID FLUORIDES, AND THE BEHAVIOR OF THESE AMINO-ACID DERIVATIVES
Authors: SAVRDA J CHERTANOVA L WAKSELMAN M
Citation: J. Savrda et al., ACTIVATION OF N,N-BIS(ALKOXYCARBONYL) AMINO-ACIDS - SYNTHESIS OF N-ALKOXYCARBONYL AMINO-ACID N-CARBOXYANHYDRIDES AND N,N-DIALKOXYCARBONYL AMINO-ACID FLUORIDES, AND THE BEHAVIOR OF THESE AMINO-ACID DERIVATIVES, Tetrahedron, 50(18), 1994, pp. 5309-5322
PREPARATION OF N-BOC N-ALKYL GLYCINES FOR PEPTOID SYNTHESIS
Authors: MOUNA AM NGUYEN C RAGE I XIE J NEE G MAZALEYRAT JP WAKSELMAN M
Citation: Am. Mouna et al., PREPARATION OF N-BOC N-ALKYL GLYCINES FOR PEPTOID SYNTHESIS, Synthetic communications, 24(17), 1994, pp. 2429-2435
AN EFFICIENT SYNTHESIS OF ARYL PHENACETURATES USING ACID-CATALYZED DICYCLOHEXYLCARBODIIMIDE ESTERIFICATION AND TRANSIENT N-TERT-BUTOXYCARBONYLATION
Authors: CABARET D LIU J WAKSELMAN M
Citation: D. Cabaret et al., AN EFFICIENT SYNTHESIS OF ARYL PHENACETURATES USING ACID-CATALYZED DICYCLOHEXYLCARBODIIMIDE ESTERIFICATION AND TRANSIENT N-TERT-BUTOXYCARBONYLATION, Synthesis, (5), 1994, pp. 480-482
CYCLIC-PEPTIDES AS SELECTIVE SUBSTRATES AND SUICIDE SUBSTRATE PRECURSORS OF TRYPSIN-LIKE PROTEINASES
Authors: BOGGETTO N VILAIN AC MONTAGNE JJ REBOUDRAVAUX M MAZALEYRAT JP XIE J WAKSELMAN M
Citation: N. Boggetto et al., CYCLIC-PEPTIDES AS SELECTIVE SUBSTRATES AND SUICIDE SUBSTRATE PRECURSORS OF TRYPSIN-LIKE PROTEINASES, Bulletin de la Societe chimique de France, 131(2), 1994, pp. 152-166
NEW MECHANISM-BASED INACTIVATORS OF TRYPSIN-LIKE PROTEINASES - SELECTIVE INACTIVATION OF UROKINASE BY FUNCTIONALIZED CYCLOPEPTIDES INCORPORATING A SULFONIOMETHYL-SUBSTITUTED M-AMINOBENZOIC ACID RESIDUE
Authors: WAKSELMAN M XIE J MAZALEYRAT JP BOGGETTO N VILAIN AC MONTAGNE JJ REBOUDRAVAUX M
Citation: M. Wakselman et al., NEW MECHANISM-BASED INACTIVATORS OF TRYPSIN-LIKE PROTEINASES - SELECTIVE INACTIVATION OF UROKINASE BY FUNCTIONALIZED CYCLOPEPTIDES INCORPORATING A SULFONIOMETHYL-SUBSTITUTED M-AMINOBENZOIC ACID RESIDUE, Journal of medicinal chemistry, 36(11), 1993, pp. 1539-1547
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