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Results: 1-20 |
Results: 20

Authors: GUIOTTO A HOWARD PW BARALDI PG THURSTON DE
Citation: A. Guiotto et al., SYNTHESIS OF NOVEL C7-ARYL SUBSTITUTED PYRROLO[2,1-C][1,4]BENZODIAZEPINES (PBDS) VIA PRO-N-10-TROC PROTECTION AND SUZUKI COUPLING, Bioorganic & medicinal chemistry letters, 8(21), 1998, pp. 3017-3018

Authors: BARALDI PG CACCIARI B GUIOTTO A LEONI A ROMAGNOLI R SPALLUTO G MONGELLI N HOWARD PW THURSTON DE BIANCHI N GAMBARI R
Citation: Pg. Baraldi et al., DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A PYRROLO[2,1-C][1,4]BENZODIAZEPINE (PBD)-DISTAMYCIN HYBRID, Bioorganic & medicinal chemistry letters, 8(21), 1998, pp. 3019-3024

Authors: KAMAL A HOWARD PW REDDY BSN REDDY BSP THURSTON DE
Citation: A. Kamal et al., SYNTHESIS OF PYRROLO[2,1-C][1,4]BENZODIAZEPINE ANTIBIOTICS - OXIDATION OF CYCLIC SECONDARY AMINE WITH TPAP, Tetrahedron, 53(9), 1997, pp. 3223-3230

Authors: PUVVADA MS FORROW SA HARTLEY JA STEPHENSON P GIBSON I JENKINS TC THURSTON DE
Citation: Ms. Puvvada et al., INHIBITION OF BACTERIOPHAGE-T7 RNA-POLYMERASE IN-VITRO TRANSCRIPTION BY DNA-BINDING PYRROLO[2,1-C][1,4]BENZODIAZEPINES, Biochemistry, 36(9), 1997, pp. 2478-2484

Authors: THURSTON DE MORRIS SJ HARTLEY JA
Citation: De. Thurston et al., SYNTHESIS OF A NOVEL GC-SPECIFIC COVALENT-BINDING DNA AFFINITY-CLEAVAGE AGENT BASED ON PYRROLOBENZODIAZEPINES (PBDS), Chemical communications, (4), 1996, pp. 563-565

Authors: VARVARESOU A TSOTINIS A SIATRAPAPASTAIKOUDI T PAPADAKIVALIRAKI A THURSTON DE JENKINS TC KELLAND LR
Citation: A. Varvaresou et al., NOVEL IMIDAZOTHIOXANTHONES - SYNTHESIS, DNA-BINDING AND CYTOTOXICITY, Bioorganic & medicinal chemistry letters, 6(7), 1996, pp. 865-870

Authors: WALTON MI GODDARD P KELLAND LR THURSTON DE HARRAP KR
Citation: Mi. Walton et al., PRECLINICAL PHARMACOLOGY AND ANTITUMOR-ACTIVITY OF THE NOVEL SEQUENCESELECTIVE DNA MINOR-GROOVE CROSS-LINKING AGENT DSB-120, Cancer chemotherapy and pharmacology, 38(5), 1996, pp. 431-438

Authors: FOLOPPE MP RAULT S THURSTON DE JENKINS TC ROBBA M
Citation: Mp. Foloppe et al., DNA-BINDING PROPERTIES OF PYRROLO[2,1-C][1,4]-BENZODIAZEPINE N-10-C-11 AMIDINES, European journal of medicinal chemistry, 31(5), 1996, pp. 407-410

Authors: THURSTON DE BOSE DS THOMPSON AS HOWARD PW LEONI A CROKER SJ JENKINS TC NEIDLE S HARTLEY JA HURLEY LH
Citation: De. Thurston et al., SYNTHESIS OF SEQUENCE-SELECTIVE C8-LINKED PYRROLO[2,1-C][1,4]BENZODIAZEPINE DNA INTERSTRAND CROSS-LINKING AGENTS, Journal of organic chemistry, 61(23), 1996, pp. 8141-8147

Authors: FOX KR THURSTON DE JENKINS TC VARVARESOU A TSOTINIS A SIATRAPAPASTAIKOUDI T
Citation: Kr. Fox et al., A NOVEL SERIES OF DNA TRIPLE HELIX-BINDING LIGANDS, Biochemical and biophysical research communications, 224(3), 1996, pp. 717-720

Authors: EIFLERLIMA VL URIAC P HUET J JENKINS TC THURSTON DE
Citation: Vl. Eiflerlima et al., RELATIONSHIP BETWEEN CYTOTOXICITY AND DNA-BINDING AFFINITY OF AMIDINEDERIVATIVES OF TETRAHYDROQUINO[4,3-B][1]BENZAZEPINES AND TETRAHYDROBENZO[K]NAPHTHYRIDIN, Bioorganic & medicinal chemistry letters, 5(24), 1995, pp. 3003-3006

Authors: HAFIZ F THURSTON DE CARR AM JONES RW
Citation: F. Hafiz et al., THE CYTOTOXICITY OF ANTHRAMYCIN TO MUTANTS OF SCHIZOSACCHAROMYCES-POMBE DEFICIENT IN DNA-DAMAGE RESPONSES, Biochemical Society transactions, 23(2), 1995, pp. 331-331

Authors: WILSON SC HOWARD PW THURSTON DE
Citation: Sc. Wilson et al., DESIGN AND SYNTHESIS OF A NOVEL EPOXIDE-CONTAINING PYRROLO[2,1-C][1,4]BENZODIAZEPINE (PBD) VIA A NEW CYCLIZATION PROCEDURE, Tetrahedron letters, 36(35), 1995, pp. 6333-6336

Authors: NEIDLE S PUVVADA MS THURSTON DE
Citation: S. Neidle et al., THE RELEVANCE OF DRUG-DNA SEQUENCE SPECIFICITY TO ANTITUMOR-ACTIVITY, European journal of cancer, 30A(4), 1994, pp. 567-568

Authors: BLUNDEN G CURRIE J THURSTON DE
Citation: G. Blunden et al., CLEAVAGE OF DNA BY BROWN ALGAL POLYPHENOLS, Journal of applied phycology, 6(3), 1994, pp. 281-284

Authors: JENKINS TC HURLEY LH NEIDLE S THURSTON DE
Citation: Tc. Jenkins et al., STRUCTURE OF A COVALENT DNA MINOR-GROOVE ADDUCT WITH A PYRROLOBENZODIAZEPINE DIMER - EVIDENCE FOR SEQUENCE-SPECIFIC INTERSTRAND CROSS-LINKING, Journal of medicinal chemistry, 37(26), 1994, pp. 4529-4537

Authors: THURSTON DE BOSE DS
Citation: De. Thurston et Ds. Bose, SYNTHESIS OF DNA-INTERACTIVE PYRROLO[2,1-C][1,4]BENZODIAZEPINES, Chemical reviews, 94(2), 1994, pp. 433-465

Authors: SMELLIE M KELLAND LR THURSTON DE SOUHAMI RL HARTLEY JA
Citation: M. Smellie et al., CELLULAR PHARMACOLOGY OF NOVEL C8-LINKED ANTHRAMYCIN-BASED SEQUENCE-SELECTIVE DNA MINOR-GROOVE CROSS-LINKING AGENTS, British Journal of Cancer, 70(1), 1994, pp. 48-53

Authors: PUVVADA MS HARTLEY JA JENKINS TC THURSTON DE
Citation: Ms. Puvvada et al., A QUANTITATIVE ASSAY TO MEASURE THE RELATIVE DNA-BINDING AFFINITY OF PYRROLO[2,1-C][1,4]BENZODIAZEPINE (PBD) ANTITUMOR ANTIBIOTICS BASED ONTHE INHIBITION OF RESTRICTION-ENDONUCLEASE BAMHI, Nucleic acids research, 21(16), 1993, pp. 3671-3675

Authors: COURTNEY SM THURSTON DE
Citation: Sm. Courtney et De. Thurston, A NEW CONVENIENT PROCEDURE FOR THE SYNTHESIS OF PYRROLO[2,1-C][1,4]BENZODIAZEPINES, Tetrahedron letters, 34(33), 1993, pp. 5327-5328
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