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Results: 1-25 | 26-26
Results: 1-25/26
Indoloparacyclophanes: Synthesis and dopamine receptor binding of a novel arylbioisostere
Authors: Ortner, B Waibel, R Gmeiner, P
Citation: B. Ortner et al., Indoloparacyclophanes: Synthesis and dopamine receptor binding of a novel arylbioisostere, ANGEW CHEM, 40(7), 2001, pp. 1283
Rational molecular design and EPC synthesis of a type VI beta-turn inducing peptide mimetic
Authors: Hoffmann, T Lanig, H Waibel, R Gmeiner, P
Citation: T. Hoffmann et al., Rational molecular design and EPC synthesis of a type VI beta-turn inducing peptide mimetic, ANGEW CHEM, 40(18), 2001, pp. 3361
Dopaminergic 7-aminotetrahydroindolizines: Ex-chiral pool synthesis and preferential D3 receptor binding
Authors: Lehmann, T Hubner, H Gmeiner, P
Citation: T. Lehmann et al., Dopaminergic 7-aminotetrahydroindolizines: Ex-chiral pool synthesis and preferential D3 receptor binding, BIOORG MED, 11(21), 2001, pp. 2863-2866
Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPCsynthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179)
Authors: Einsiedel, J Hubner, H Gmeiner, P
Citation: J. Einsiedel et al., Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPCsynthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179), BIOORG MED, 11(18), 2001, pp. 2533-2536
Synthesis and in vitro evaluation of iodine labelled pyrazolo[1,5-a]pyridines as highly selective dopamine D4 receptor ligands
Authors: Prante, O Lober, S Hubner, H Gmeiner, P Kuwert, T
Citation: O. Prante et al., Synthesis and in vitro evaluation of iodine labelled pyrazolo[1,5-a]pyridines as highly selective dopamine D4 receptor ligands, J LABEL C R, 44(12), 2001, pp. 849-858
Diethoxymethyl protected pyrroles: Synthesis and regioselective transformations
Authors: Bergauer, M Gmeiner, P
Citation: M. Bergauer et P. Gmeiner, Diethoxymethyl protected pyrroles: Synthesis and regioselective transformations, SYNTHESIS-S, (15), 2001, pp. 2281-2288
Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapine
Authors: Lanig, H Utz, W Gmeiner, P
Citation: H. Lanig et al., Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapine, J MED CHEM, 44(8), 2001, pp. 1151-1157
Rationally based efficacy tuning of selective dopamine D4 receptor ligandsleading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-alpha]pyridine (FAUC 213)
Authors: Lober, S Hubner, H Utz, W Gmeiner, P
Citation: S. Lober et al., Rationally based efficacy tuning of selective dopamine D4 receptor ligandsleading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-alpha]pyridine (FAUC 213), J MED CHEM, 44(17), 2001, pp. 2691-2694
Treatment of N,N-dibenzylamino alcohols with sulfonyl chloride leads to rearranged beta-chloro amines, precursors to beta-amino acids, and not to tetrahydroisoquinolines
Authors: Weber, K Kuklinski, S Gmeiner, P
Citation: K. Weber et al., Treatment of N,N-dibenzylamino alcohols with sulfonyl chloride leads to rearranged beta-chloro amines, precursors to beta-amino acids, and not to tetrahydroisoquinolines, ORG LETT, 2(5), 2000, pp. 647-649
Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: Synthesis and dopamine receptor binding profiles
Authors: Einsiedel, J Thomas, C Hubner, H Gmeiner, P
Citation: J. Einsiedel et al., Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: Synthesis and dopamine receptor binding profiles, BIOORG MED, 10(17), 2000, pp. 2041-2044
Traceless linking of indoles: General methodology and application to solidphase supported Mannich and Stille reactions
Authors: Kraxner, J Arlt, M Gmeiner, P
Citation: J. Kraxner et al., Traceless linking of indoles: General methodology and application to solidphase supported Mannich and Stille reactions, SYNLETT, (1), 2000, pp. 125-127
Synthesis of enantiopure 8-aminomethylindolizines from glutamine by stereoelectronically controlled cationic cyclization
Authors: Lehmann, T Gmeiner, P
Citation: T. Lehmann et P. Gmeiner, Synthesis of enantiopure 8-aminomethylindolizines from glutamine by stereoelectronically controlled cationic cyclization, HETEROCYCLE, 53(6), 2000, pp. 1371-1378
Azepino- and diazepinoindoles: Synthesis and dopamine receptor binding profiles
Authors: Kraxner, J Hubner, H Gmeiner, P
Citation: J. Kraxner et al., Azepino- and diazepinoindoles: Synthesis and dopamine receptor binding profiles, ARCH PHARM, 333(9), 2000, pp. 287-292
Regiocontrolled annellation reactions starting from diethoxymethyl protected indole
Authors: Kraxner, J Gmeiner, P
Citation: J. Kraxner et P. Gmeiner, Regiocontrolled annellation reactions starting from diethoxymethyl protected indole, SYNTHESIS-S, (8), 2000, pp. 1081-1083
Effective and variable functionalization of pyrazolo[1,5-a]pyridines involving palladium-catalyzed coupling reactions
Authors: Aboul-Fadl, T Lober, S Gmeiner, P
Citation: T. Aboul-fadl et al., Effective and variable functionalization of pyrazolo[1,5-a]pyridines involving palladium-catalyzed coupling reactions, SYNTHESIS-S, (12), 2000, pp. 1727-1732
Enantiopure 4-and 5-aminopiperidin-2-ones: Regiocontrolled synthesis and conformational characterization as bioactive beta-turn mimetics
Authors: Weber, K Ohnmacht, U Gmeiner, P
Citation: K. Weber et al., Enantiopure 4-and 5-aminopiperidin-2-ones: Regiocontrolled synthesis and conformational characterization as bioactive beta-turn mimetics, J ORG CHEM, 65(22), 2000, pp. 7406-7416
Conjugated enynes as nonaromatic catechol bioisosteres: Synthesis, bindingexperiments, and computational studies of novel dopamine receptor agonistsrecognizing preferentially the D-3 subtype
Authors: Hubner, H Haubmann, C Utz, W Gmeiner, P
Citation: H. Hubner et al., Conjugated enynes as nonaromatic catechol bioisosteres: Synthesis, bindingexperiments, and computational studies of novel dopamine receptor agonistsrecognizing preferentially the D-3 subtype, J MED CHEM, 43(4), 2000, pp. 756-762
Cyanoindole derivatives as highly selective dopamine D-4 receptor partial agonists: Solid-phase synthesis, binding assays, and functional experiments
Authors: Hubner, H Kraxner, J Gmeiner, P
Citation: H. Hubner et al., Cyanoindole derivatives as highly selective dopamine D-4 receptor partial agonists: Solid-phase synthesis, binding assays, and functional experiments, J MED CHEM, 43(23), 2000, pp. 4563-4569
Enantio- and diastereocontrolled dopamine D1, D2, D3 and D4 receptor binding of N-(3-pyrrolidinylmethyl)benzamides synthesized from aspartic acid
Authors: Thomas, C Hubner, H Gmeiner, P
Citation: C. Thomas et al., Enantio- and diastereocontrolled dopamine D1, D2, D3 and D4 receptor binding of N-(3-pyrrolidinylmethyl)benzamides synthesized from aspartic acid, BIOORG MED, 9(6), 1999, pp. 841-846
Piperidinylpyrroles: Design, synthesis and binding properties of novel andselective dopamine D4 receptor ligands
Authors: Haubmann, C Hubner, H Gmeiner, P
Citation: C. Haubmann et al., Piperidinylpyrroles: Design, synthesis and binding properties of novel andselective dopamine D4 receptor ligands, BIOORG MED, 9(21), 1999, pp. 3143-3146
2,2-Dicyanovinyl as a nonaromatic aryl bioisostere: Synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands
Authors: Haubmann, C Hubner, H Gmeiner, P
Citation: C. Haubmann et al., 2,2-Dicyanovinyl as a nonaromatic aryl bioisostere: Synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands, BIOORG MED, 9(14), 1999, pp. 1969-1972
Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps
Authors: Lober, S Hubner, H Gmeiner, P
Citation: S. Lober et al., Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps, BIOORG MED, 9(1), 1999, pp. 97-102
Chemo- and regioselective syntheses of enantiopure aminopyrrolidinones as building blocks for constrained peptidomimetics
Authors: Lehmann, T Michel, D Glanzel, M Waibel, R Gmeiner, P
Citation: T. Lehmann et al., Chemo- and regioselective syntheses of enantiopure aminopyrrolidinones as building blocks for constrained peptidomimetics, HETEROCYCLE, 51(6), 1999, pp. 1389
Ex-chiral pool synthesis of aminooxazepinones as conformationally restricted beta-amino acid analogs
Authors: Michel, D Waibel, R Gmeiner, P
Citation: D. Michel et al., Ex-chiral pool synthesis of aminooxazepinones as conformationally restricted beta-amino acid analogs, HETEROCYCLE, 51(2), 1999, pp. 365-372
Ex-chiral pool synthesis and pharmacological aspects of 3-pyrrolidinylisoxazoles
Authors: Thomas, C Ohnmacht, U Zahn, K Mohr, K Gmeiner, P
Citation: C. Thomas et al., Ex-chiral pool synthesis and pharmacological aspects of 3-pyrrolidinylisoxazoles, PHARMAZIE, 54(4), 1999, pp. 248-250
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