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Results: 1-25 |
Results: 25

Authors: CHEN SH FARINA V VYAS DM DOYLE TW
Citation: Sh. Chen et al., SYNTHESIS OF A PACLITAXEL ISOMER - C-2-ACETOXY-C-4-BENZOATE PACLITAXEL, Bioorganic & medicinal chemistry letters, 8(16), 1998, pp. 2227-2230

Authors: ALTSTADT TJ GAO Q WITTMAN MD KADOW JF VYAS DM
Citation: Tj. Altstadt et al., CRYSTALLOGRAPHIC DETERMINATION OF THE STEREOCHEMISTRY OF C-6,7 EPOXY PACLITAXEL, Tetrahedron letters, 39(28), 1998, pp. 4965-4966

Authors: GOLIK J WONG HSL CHEN SH DOYLE TW WRIGHT JJK KNIPE J ROSE WC CASAZZA AM VYAS DM
Citation: J. Golik et al., SYNTHESIS AND ANTITUMOR EVALUATION OF PACLITAXEL PHOSPHONOOXYMETHYL ETHERS - A NOVEL CLASS OF WATER-SOLUBLE PACLITAXEL PRO-DRUGS, Bioorganic & medicinal chemistry letters, 6(15), 1996, pp. 1837-1842

Authors: MASTALERZ H DOYLE TW KADOW JF VYAS DM
Citation: H. Mastalerz et al., SYNTHESIS OF AN ESPERAMICIN CORE ANALOG WITH AN EPOXIDE TRIGGER, Tetrahedron letters, 37(48), 1996, pp. 8683-8686

Authors: MASTALERZ H DOYLE TW KADOW JF VYAS DM
Citation: H. Mastalerz et al., SYNTHESIS OF A HYBRID ANALOG OF THE ESPERAMICIN AND DYNEMICIN CORES, Tetrahedron letters, 37(48), 1996, pp. 8687-8690

Authors: CHEN SH FARINA V VYAS DM DOYLE TW
Citation: Sh. Chen et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF C-13 AMIDE-LINKED PACLITAXEL (TAXOL) ANALOGS, Journal of organic chemistry, 61(6), 1996, pp. 2065-2070

Authors: UEDA Y MATISKELLA JD MIKKILINENI AB FARINA V KNIPE JO ROSE WC CASAZZA AM VYAS DM
Citation: Y. Ueda et al., NOVEL, WATER-SOLUBLE PHOSPHATE DERIVATIVES OF 2'-ETHOXY CARBONYLPACLITAXEL AS POTENTIAL PRODRUGS OF PACLITAXEL - SYNTHESIS AND ANTITUMOR EVALUATION, Bioorganic & medicinal chemistry letters, 5(3), 1995, pp. 247-252

Authors: CHEN SH WEI JM LONG BH FAIRCHILD CA CARBONI J MAMBER SW ROSE WC JOHNSTON K CASAZZA AM KADOW JF FARINA V VYAS DM DOYLE TW
Citation: Sh. Chen et al., NOVEL C-4 PACLITAXEL (TAXOL(R)) ANALOGS - POTENT ANTITUMOR AGENTS, Bioorganic & medicinal chemistry letters, 5(22), 1995, pp. 2741-2746

Authors: WITTMAN MD KADOW JF LANGLEY DR VYAS DM ROSE WC SOLOMON W ZEIN N
Citation: Md. Wittman et al., THE SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ENEDIYNE MINOR-GROOVE BINDING HYBRIDS, Bioorganic & medicinal chemistry letters, 5(10), 1995, pp. 1049-1052

Authors: VYAS DM DOYLE TW
Citation: Dm. Vyas et Tw. Doyle, NEWER STRATEGIES FOR ANTITUMOR DRUG DISCOVERY, Drug development research, 34(2), 1995, pp. 89-90

Authors: SAULNIER MG FRENNESSON DB DESHPANDE MS VYAS DM
Citation: Mg. Saulnier et al., SYNTHESIS OF A REBECCAMYCIN-RELATED INDOLO[2,3-A]CARBAZOLE BY PALLADIUM(0) CATALYZED POLYANNULATION, Tetrahedron letters, 36(43), 1995, pp. 7841-7844

Authors: WITTMAN MD KADOW JF PHAM K LEUNG K MASTALERZ HA VYAS DM ROSE WC SOLOMON W ZEIN N
Citation: Md. Wittman et al., THE EFFECT OF PROPARGYLIC SUBSTITUTION ON THE ACTIVATION AND AROMATIZATION OF ENEDIYNES, Bioorganic & medicinal chemistry letters, 4(24), 1994, pp. 2925-2928

Authors: SAULNIER MG LANGLEY DR KADOW JF SENTER PD KNIPE JO TUN MM VYAS DM DOYLE TW
Citation: Mg. Saulnier et al., SYNTHESIS OF ETOPOSIDE PHOSPHATE, BMY-40481 - A WATER-SOLUBLE CLINICALLY ACTIVE PRODRUG OF ETOPOSIDE, Bioorganic & medicinal chemistry letters, 4(21), 1994, pp. 2567-2572

Authors: CHEN SH KANT J MAMBER SW ROTH GP WEI JM MARSHALL D VYAS DM FARINA V CASAZZA A LONG BH ROSE WC JOHNSTON K FAIRCHILD C
Citation: Sh. Chen et al., TAXOL(R) STRUCTURE-ACTIVITY-RELATIONSHIPS - SYNTHESIS AND BIOLOGICAL EVALUATION OF TAXOL ANALOGS MODIFIED AT C-7, Bioorganic & medicinal chemistry letters, 4(18), 1994, pp. 2223-2228

Authors: SAULNIER MG FRENNESSON DB DESHPANDE MS HANSEL SB VYAS DM
Citation: Mg. Saulnier et al., AN EFFICIENT METHOD FOR THE SYNTHESIS OF GUANIDINO PRODRUGS, Bioorganic & medicinal chemistry letters, 4(16), 1994, pp. 1985-1990

Authors: UEDA Y WONG H MATISKELLA JD MIKKILINENI AB FARINA V FAIRCHILD C ROSE WC MAMBER SW LONG BH KERNS EH CASAZZA AM VYAS DM
Citation: Y. Ueda et al., SYNTHESIS AND ANTITUMOR EVALUATION OF 2'-OXYCARBONYLPACLITAXELS (PACLITAXEL-2'-CARBONATES), Bioorganic & medicinal chemistry letters, 4(15), 1994, pp. 1861-1864

Authors: KANT J FARINA V FAIRCHILD C KADOW JF LANGLEY DR LONG BH ROSE WC VYAS DM
Citation: J. Kant et al., SYNTHESIS AND ANTITUMOR PROPERTIES OF NOVEL 14-BETA-HYDROXYTAXOL AND RELATED ANALOGS, Bioorganic & medicinal chemistry letters, 4(13), 1994, pp. 1565-1570

Authors: YU KL DESHPANDE MS VYAS DM
Citation: Kl. Yu et al., HECK REACTIONS IN SOLID-PHASE SYNTHESIS, Tetrahedron letters, 35(48), 1994, pp. 8919-8922

Authors: KADOW JF COOK DJ DOYLE TW LANGLEY DR PHAM KM VYAS DM WITTMAN MD
Citation: Jf. Kadow et al., FACILE SYNTHESIS OF A SIMPLIFIED BICYCLO[7.3.1] ESPERAMICIN-CALICHEAMICIN ENEDIYNE CORE, Tetrahedron, 50(5), 1994, pp. 1519-1538

Authors: SAULNIER MG LEBOULLUEC KL MCGEE DPC LONG BH CROSSWELL AR VYAS DM
Citation: Mg. Saulnier et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 3',4',5'-TRIHYDROXY ETOPOSIDE, Bioorganic & medicinal chemistry letters, 3(8), 1993, pp. 1619-1624

Authors: UEDA Y MIKKILINENI AB KNIPE JO ROSE WC CASAZZA AM VYAS DM
Citation: Y. Ueda et al., NOVEL WATER-SOLUBLE PHOSPHATE PRODRUGS OF TAXOL(R) POSSESSING IN-VIVOANTITUMOR-ACTIVITY, Bioorganic & medicinal chemistry letters, 3(8), 1993, pp. 1761-1766

Authors: ZEIN N SOLOMON W CASAZZA AM KADOW JF KRISHNAN BS TUN MM VYAS DM DOYLE TW
Citation: N. Zein et al., PROTEIN DAMAGE CAUSED BY A SYNTHETIC ENEDIYNE CORE, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 1351-1356

Authors: VYAS DM WONG H CROSSWELL AR CASAZZA AM KNIPE JO MAMBER SW DOYLE TW
Citation: Dm. Vyas et al., SYNTHESIS AND ANTITUMOR EVALUATION OF WATER-SOLUBLE TAXOL PHOSPHATES, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 1357-1360

Authors: CHEN SH WEI JM VYAS DM DOYLE TW FARINA V
Citation: Sh. Chen et al., A FACILE SYNTHESIS OF 7,10-DIDEOXY TAXOL AND 7-EPI-10-DEOXY TAXOL, Tetrahedron letters, 34(43), 1993, pp. 6845-6848

Authors: ZHANG M WANG YT VYAS DM NEUMAN RS BIEGER D
Citation: M. Zhang et al., NICOTINIC CHOLINOCEPTOR-MEDIATED EXCITATORY POSTSYNAPTIC POTENTIALS IN RAT NUCLEUS AMBIGUUS, Experimental Brain Research, 96(1), 1993, pp. 83-88
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